dbACP: A Comprehensive Database of Anti-Cancer Peptides

dbacp04604

General Description

Peptide name : Maximin H1

Source/Organism : Yunnan firebelly toad, China, Asia

Linear/Cyclic : Linear

Chirality : Not found

Sequence Information

Sequence : ILGPVISTIGGVLGGLLKNL

Peptide length: 20

C-terminal modification: Linear

N-terminal modification : Free

Non-natural peptide information: None

Activity Information

Assay type : MTT assay

Assay time : 6h

Activity : Not found

Cell line : BIU-87

Cancer type : Bladder cancer

Other activity : Anti- microbial activity

Physicochemical Properties

Amino acid composition bar chart :

Molecular mass : 1934.3659 Dalton

Aliphatic index : 1.85

Instability index : 36.855

Hydrophobicity (GRAVY) : 1.42

Isoelectric point : 8.7501

Charge (pH 7) : 0.7591

Aromaticity : 0

Molar extinction coefficient (cysteine, cystine): (0, 0)

Hydrophobic/hydrophilic ratio : 4

hydrophobic moment : 0.0467

Missing amino acid : C,R,W,H,Q,M,E,F,D,Y,A

Most occurring amino acid : L

Most occurring amino acid frequency : 5

Least occurring amino acid : P

Least occurring amino acid frequency : 1

Structural Information

3D structure :

Secondary structure fraction (Helix, Turn, Sheet): (0.3, 0.4, 0.5)

SMILES Notation: CC[C@H](C)[C@H](N)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)NCC(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)O)C(C)C)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC)C(C)C

Secondary Structure :

Method Prediction
GOR EECCEEEEEEEEEEEEEETH
Chou-Fasman (CF) EEEEEEEEEEEEEECCCCCC
Neural Network (NN) CCCCCEEEECCEECHHHCCC
Joint/Consensus EECCEEEEEEEEEECCCCCC

Molecular Descriptors and ADMET Properties

Molecular Descriptors: Click here to download

ADMET Properties: Click here to download

Cross Referencing databases

Pubmed Id : 11835991

Uniprot : Not available

PDB : Not available

CancerPPD : Not available

ApIAPDB : Not available

CancerPPD2 ID : Not available

Reference

1 : Lai R, et al. Antimicrobial peptides from skin secretions of Chinese red belly toad Bombina maxima. Peptides. 2002; 23:427-35. doi: 10.1016/s0196-9781(01)00641-6

Literature

Paper title : Antimicrobial peptides from skin secretions of Chinese red belly toad Bombina maxima.

Doi : https://doi.org/10.1016/s0196-9781(01)00641-6

Abstract : Two groups of antimicrobial peptides have been isolated from skin secretions of Bombina maxima. Peptides in the first group, named maximins 1, 2, 3, 4 and 5, are structurally related to bombinin-like peptides (BLPs). Unlike BLPs, sequence variations in maximins occurred all through the molecules. In addition to the potent antimicrobial activity, cytotoxicity against tumor cells and spermicidal action of maximins, maximin 3 possessed a significant anti-HIV activity. Maximins 1 and 3 were toxic to mice with LD(50) values of 8.2 and 4.3 mg/kg, respectively. Peptides in the second group, termed maximins H1, H2, H3 and H4, are homologous with bombinin H peptides. cDNA sequences revealed that one maximin peptide plus one maximin H peptide derived from a common larger protein.