dbACP: A Comprehensive Database of Anti-Cancer Peptides

dbacp06228

General Description

Peptide name : Temporin A

Source/Organism : European common frog

Linear/Cyclic : Linear

Chirality : L

Sequence Information

Sequence : FLPLIGRVLSGIL

Peptide length: 13

C-terminal modification: Linear

N-terminal modification : Amidation

Non-natural peptide information: None

Activity Information

Assay type : MTT/MTS assay

Assay time : 6h

Activity : 15% cytotoxicity at 0.5 µg/ml

Cell line : U-937

Cancer type : Lymphoma cancer

Other activity : Anti-bacterial activity

Physicochemical Properties

Amino acid composition bar chart :

Molecular mass : 1397.7465 Dalton

Aliphatic index : 2.023

Instability index : 32.3308

Hydrophobicity (GRAVY) : 1.8077

Isoelectric point : 9.75

Charge (pH 7) : 0.7601

Aromaticity : 0.076

Molar extinction coefficient (cysteine, cystine): (0, 0)

Hydrophobic/hydrophilic ratio : 5.5

hydrophobic moment : 1.4779

Missing amino acid : C,W,H,Q,T,M,E,K,D,Y,N,A

Most occurring amino acid : L

Most occurring amino acid frequency : 4

Least occurring amino acid : F

Least occurring amino acid frequency : 1

Structural Information

3D structure :

Secondary structure fraction (Helix, Turn, Sheet): (0.3, 0.3, 0.6)

SMILES Notation: CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)Cc1ccccc1)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)O

Secondary Structure :

Method Prediction
GOR ECCEEEEEEEEEE
Chou-Fasman (CF) CEEEEEEEEECCC
Neural Network (NN) CCCCCCCHCCCCE
Joint/Consensus CCCEEEEEEECCC

Molecular Descriptors and ADMET Properties

Molecular Descriptors: Click here to download

ADMET Properties: Click here to download

Cross Referencing databases

Pubmed Id : 9022710

Uniprot : Not available

PDB : Not available

CancerPPD : Click here

ApIAPDB : Not available

CancerPPD2 ID : Not available

Reference

1 : Simmaco M, et al. Temporins, antimicrobial peptides from the European red frog Rana temporaria. Eur J Biochem. 1996; 242:788-92. doi: 10.1111/j.1432-1033.1996.0788r.x

Literature

Paper title : Temporins, antimicrobial peptides from the European red frog Rana temporaria.

Doi : https://doi.org/10.1111/j.1432-1033.1996.0788r.x

Abstract : A cDNA library from the skin of Rana temporaria has been screened using a cDNA fragment probe that encodes the signal peptide of the precursor of esculentin from the skin secretion of Rana esculenta. With this approach, the cDNAs encoding the precursors of three peptides were isolated. Subsequently, the peptides predicted from the sequence of the cloned cDNAs as well as several structurally related peptides could be isolated from the skin secretion of R. temporaria. These peptides, which were named temporins, have a length of 10-13 residues and show some sequence similarity to hemolytic peptides isolated from Vespa venom [Argiolas, A. & Pisano, J. J. (1984) J. Biol. Chem. 259, 10106-10111]. Natural and synthetic temporins have antibacterial activity against gram-positive bacteria, but they are not hemolytic. Temporins are the smallest antibacterial peptides hitherto found in nature.