8 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp02362 | Cecropin B | KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL | Silkmoth | Pore formation at the cytoplasmic membrane | MTT/MTS assay | A-2780 | Ovarian cancer | IC50 : 30.6 µM |
| dbacp02368 | Cecropin B | KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL | Silkmoth | Pore formation at the cytoplasmic membrane | MTT/MTS assay | A-2780R | Ovarian cancer | IC50 : 34.5 µM |
| dbacp07026 | [G10a]-SHa | FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | A-2780 | Ovarian Cancer | IC50 = 14.75 ± 7.35 µM |
| dbacp07033 | [G10a]2-SHa | FLSGIVGMLaKLFKFLKaLMFLSGIVG | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | A-2780 | Ovarian Cancer | IC50 = 4.42 ± 0.06 µM |
| dbacp07040 | [G10a]3-SHa | FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | A-2780 | Ovarian Cancer | IC50 = 2.31 ± 0.08 µM |
| dbacp07046 | Jeff-[G10a]2-SHa | FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | A-2780 | Ovarian Cancer | IC50 = 33.92 ± 5.90 µM |
| dbacp07880 | Nubein6.8 | LKCNQLIPPFWKTCPKGKNLCYKMTMRAAPMVPVKRGCIDVCPKSSLLIKYMCCNTDKCN | Naja nubiae | DNA damage and apoptosis induction | MTT assay | A-2780 | Ovarian Cancer | EC50 = 1.249 ± 0.06 μM |
| dbacp08291 | L-Carnosine | Beta-AH | Synthetic | Not Available | MTT assay | A-2780 | Ovarian Cancer | IC50 = 165 mM |