37 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp00774 | A12L | KWKSFLKTFKSLKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 4.3 µMo/L |
| dbacp00782 | A12L/A20L | KWKSFLKTFKSLKKTVLHTLLKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 8.7 µMo/L |
| dbacp00790 | A12L/A20L/A23L | KWKSFLKTFKSLKKTVLHTLLKLISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 7.2 µMo/L |
| dbacp00798 | A20L | KWKSFLKTFKSAKKTVLHTLLKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 6.5 µMo/L |
| dbacp03571 | L17A | KWKSFLKTFKSAKKTVAHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : > 83.6 µMo/L |
| dbacp03579 | L17A/L21A | KWKSFLKTFKSAKKTVAHTAAKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : > 83.6 µMo/L |
| dbacp03590 | L21A | KWKSFLKTFKSAKKTVAHTAAKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 59.8 µMo/L |
| dbacp03614 | L6A | KWKSFAKTFKSAKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 58.7 µMo/L |
| dbacp03622 | L6A/L17A | KWKSFAKTFKSAKKTVAHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : >83.6 µMo/L |
| dbacp05022 | Peptide P | KWKSFLKTFKSAKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | A-375 | Skin cancer | IC50 : 17.8 µMo/L |
| dbacp05043 | P18 | KWKLFKKIPKFLHLAKKF | Synthetic peptide | Necrosis; Cell membrane rupture | MTT/MTS assay | A-375 | Skin cancer | 86 ± 0.57% cell viability at 10 µM |
| dbacp05044 | P18 | KWKLFKKIPKFLHLAKKF | Synthetic peptide | Necrosis; Cell membrane rupture | MTT/MTS assay | A-375 | Skin cancer | 63.8 ± 0.8% cell viability at 20 µM |
| dbacp05045 | P18 | KWKLFKKIPKFLHLAKKF | Synthetic peptide | Necrosis; Cell membrane rupture | MTT/MTS assay | A-375 | Skin cancer | 47.5 ± 1.66% cell viability at 40 µM |
| dbacp05046 | P18 | KWKLFKKIPKFLHLAKKF | Synthetic peptide | Necrosis; Cell membrane rupture | MTT/MTS assay | A-375 | Skin cancer | 26.9 ± 0.5% cell viability at 60 µM |
| dbacp05047 | P18 | KWKLFKKIPKFLHLAKKF | Synthetic peptide | Necrosis; Cell membrane rupture | MTT/MTS assay | A-375 | Skin cancer | 6.5 ± 1.07% cell viability at 80 µM |
| dbacp06802 | A11 | EYVQTVKSSKG | Annexin A1 | Targeting PD-L3 | Biotin Pull Down assay | A-375 | Skin Cancer | Not Available |
| dbacp07008 | ST101 | vaeareelerlearlgqargelkkwkmrrnqfwlklqr | Synthetic | Prevents C/EBPβ dimerization, induces degradation | Annexin V/ PI staining assay | A-375 | Skin Cancer | mean EC50 value of 2.1 ± 0.4 μmol/L |
| dbacp07360 | N-Ter-TAT | RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ | Synthetic | Mitochondrial targeting, VDAC1-HKII dissociation | MTT assay | A-375 | Skin Cancer | IC50 > 50.0 μM |
| dbacp07361 | Pal-N-Ter-TAT | Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ | Analogue of N-terminal fragment of the VDAC1 protein | Mitochondrial targeting, VDAC1-HKII dissociation | MTT assay | A-375 | Skin Cancer | IC50 = 36.67(Supplementary material)/15.2 ± 0.7 μM(Published paper) |
| dbacp07364 | pFL-N-Ter-TAT | FPWWWPFL-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ | Analogue of N-terminal fragment of the VDAC1 protein | Mitochondrial targeting, VDAC1-HKII dissociation | MTT assay | A-375 | Skin Cancer | IC50 = 11.1 ± 0.1 μM |
| dbacp07465 | ΔM4 | NFFKRIRRAWKRIWKWIYSA | Synthetic | Membrane disruption triggers mitochondrial apoptosis | Not Available | A-375 | Skin Cancer | IC50 = 9.31 μM |
| dbacp07578 | R-DIM-P-LF11 | FQWQRNIRKVRPRVKRINRQWQF | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 125.0 ± 16.8 μM |
| dbacp07581 | R-DIM-P-LF11-322 | PFWRIRIRRPRRIRIRWFP | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 4.2 ± 0.2 μM |
| dbacp07584 | DIM-LF11-322 | PFWRIRIRRPFWRIRIRR | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 6.3 ± 0.3 μM |
| dbacp07587 | R-DIM-P-LF11-215 | FWRIRIRRPRRIRIRWF | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 2.7 ± 0.9 μM |
| dbacp07590 | R-DIM-P-LF11-334 | PWRIRIRRPRRIRIWP | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 6.6 ± 0.3 μM |
| dbacp07593 | R-DIM-LF11-334-LF11-334 | PWRIRIRRRRIRIRWPPWRIRIRR | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 < 1 ± 0.1 μM |
| dbacp07596 | DIM-LF11-339 | RRWFWRRRRWFWRR | Synthetic | Peptides target phosphatidylserine, trigger apoptosis | MTS assay | A-375 | Skin Cancer | LC50 = 4.8 ± 0.4 μM |
| dbacp07648 | AP1-Z1 | FLFSLIPHAISGLISAFK | AcrAP1 from the venom of the Arabian scorpion | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | IC50 = 9.478 μM |
| dbacp07651 | AP1-Z5a | FLFKLIPKAIKGLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | Graph Figure 2B |
| dbacp07654 | AP1-Z5b | FLFKLIKHAIKGLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | IC50 = 2.607 μM |
| dbacp07657 | AP1-Z3a | FLFSLIKHAIKGLISAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | Graph Figure 2B |
| dbacp07660 | AP1-Z3b | FLFSLIKHAISKLISAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | Graph Figure 2B |
| dbacp07663 | AP1-Z7 | FLFKLIKKAIKKLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | Graph Figure 2B |
| dbacp07666 | AP1-Z9 | FLFKLIKKKIKKLIKKFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | A-375 | Skin Cancer | Graph Figure 2B |
| dbacp07879 | Nubein6.8 | LKCNQLIPPFWKTCPKGKNLCYKMTMRAAPMVPVKRGCIDVCPKSSLLIKYMCCNTDKCN | Naja nubiae | DNA damage and apoptosis induction | MTT assay | A-375 | Skin Cancer | EC50 = 0.54 ± 0.04 μM |
| dbacp08167 | Bmattacin2 | Not Available | silkworm Bombyx mori | Not Available | MTS assay | A-375 | Skin Cancer | IC50 = 5.23 μM |