31 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp06359 | TsAP-1 | FLSLIPSLVGGSISAFK | Venom-derived cDNAlibrary of the Brazilian yellow scorpion | Not specified | MTT/MTS assay | H-838 | Lung cancer | IC50 : 52.5 µM |
| dbacp06361 | TsAP-2 | FLGMIPGLIGGLISAFK | Venom-derived cDNAlibrary of the Brazilian yellow scorpion | Not specified | MTT/MTS assay | H-838 | Lung cancer | IC50 : 11.0 µM |
| dbacp06369 | TsAP-S1 | FLSLIPKLVKKIIKAFK | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | Not specified | MTT/MTS assay | H-838 | Lung cancer | IC50 : 1.6 µM |
| dbacp06377 | TsAP-S2 | FLGMIPKLIKKLIKAFK | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | Not specified | MTT/MTS assay | H-838 | Lung cancer | IC50 : 1.6 µM |
| dbacp06669 | Crabrolin | FLPLILRKIVTAL | European hornet (Vespa crabro) | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 27.71 μM |
| dbacp06674 | Crabrolin-4R | FLPRILRKIVTAL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 11.40 μM |
| dbacp06679 | Crabrolin-4K | FLPKILRKIVTAL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 22.55 μM |
| dbacp06684 | Crabrolin-TR | FLPRILRKIVRAL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 4.637 μM |
| dbacp06689 | Crabrolin-FR | RLPRILRKIVRAL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 31.51 μM |
| dbacp06694 | Crabrolin-AR | RLPRILRKIVRRL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 41.31 μM |
| dbacp06699 | Crabrolin-PR | RLRRILRKIVRRL | Synthetic Analog of Crabrolin | Not available | MTT assay | H-838 | Lung Cancer | IC50 = 32.32 μM |
| dbacp06723 | L14 | ALWKSILKNAGKALNEINQIVQ | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 64.4 µM |
| dbacp06725 | 14V | ALWKSILKNAGKAVLNEINQIVQ | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 7.0 µM |
| dbacp06727 | 14G | ALWKSILKNAGKAGLNEINQIVQ | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 48.7 µM |
| dbacp06729 | L2V | ALWKSILKNVGKVLNEINQIVQ | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 2.2 µM |
| dbacp06731 | 14V5K | ALWKKILKNAGKAVLNEINQIVQ | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 8.1 µM |
| dbacp06733 | 14VL23 | ALWKSILKNAGKAVLNEINQIV | Dermaseptin-SS1- Analog | Membrane Permeabilization | MTT assay | H-838 | Lung Cancer | IC50 = 5.7 µM |
| dbacp07052 | Temporin-PKE | FLPLIIGALSSLLPKIF | skin secretion of Pelophylax kl. esculentus | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 16.38 μM |
| dbacp07057 | Temporin-PKE-2K | FLPLIIGKLSSLLPKIF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 3.07 μM |
| dbacp07062 | Temporin-PKE-K12 | FLPLIIGALSSKLPKIF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 22.67 μM |
| dbacp07067 | Temporin-PKE-3K | FLPKIIGKLSSLLPKIF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 0.51 μM |
| dbacp07072 | Temporin-PKE-4K | FLPKIIGKLSSKLPKIF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 35.28 μM |
| dbacp07077 | Temporin-PKE-i | FLPLIIGALSSLLPKiF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 5.28 μM |
| dbacp07082 | Temporin-PKE-3i | FLPLiiGALSSLLPKiF | Synthetic | Charge-optimized membranolysis induces apoptosis. | MTT assay | H-838 | Lung Cancer | IC50 = 193.4 μM |
| dbacp07260 | t-DPH1-K4 | GLWKKIKNVAAAAGKAALGAL | Analogue of t-DPH1 | Membrane disruption induces apoptotic signaling. | MTT assay | H-838 | Lung Cancer | IC50 = 10.11 μM |
| dbacp07264 | t-DPH1-5K | GLWKKIKNVAKAAGKAALGAL | Analogue of t-DPH1 | Membrane disruption induces apoptotic signaling. | MTT assay | H-838 | Lung Cancer | IC50 = 1.796 μM |
| dbacp07268 | t-DPH1-6K | GLWKKIKNVAKAAGKAAKGAL | Analogue of t-DPH1 | Membrane disruption induces apoptotic signaling. | MTT assay | H-838 | Lung Cancer | IC50 = 186.1 μM |
| dbacp07272 | t-DPH1-6KW | WLWKKIKNVAKAAGKAAKGAL | Analogue of t-DPH1 | Membrane disruption induces apoptotic signaling. | MTT assay | H-838 | Lung Cancer | IC50 = 180.8 μM |
| dbacp07312 | B1OS-L | FLPLIASLAGNVVPKIFCKITKRC | B-1OS | Not Available | MTT assay | H-838 | Lung Cancer | IC50 = 3.976 µM |
| dbacp07317 | B1OS-D-L | FlPLIASLAGNVVPKIFCKITKRC | B-1OS | Not Available | MTT assay | H-838 | Lung Cancer | IC50 = 2.553 µM |
| dbacp07927 | Phylloseptin-PBa3 | FLSLIPHIVSGVAALANHL | Phyllomedusa burmeisteri | Membrane disruption, apoptosis, selective cytotoxicity | MTT assay | H-838 | Lung Cancer | Cell viability ~ 65% at 10-5 M |