dbACP: A Comprehensive Database of Anti-Cancer Peptides

63 result(s) have been found!

Accession Name Sequence Source/Organism Mechanism Assay Type Cell Line Cancer Type Activity
dbacp01160 Antimicrobial peptide TsAP-1 MQIKHLITLFFLVLIVADQCSAFLSLIPSLVGGSISAFKGRRKREISAQIEQYKDLQKREAELEELLDRLPMY Brazilian scorpion Membrane disruption MTT Cell viability assay NCIeH157 Human squamous carcinoma IC50 : 0.83 - 2.0 μM
dbacp01166 Antimicrobial peptide TsAP- MQIKHLITLFFLVLIVADQCSAFLSLIPSLVGGSISAFKGRRKREISAQIEQYKDLQKREAELEELLDRLPMY Brazilian scorpion Antiproliferative action Not specified H157 Prostate cancer IC50 : 52.5 μM
dbacp01168 Antimicrobial peptide TsAP-2 MQIKHLITIFFLVLIVADHCHAFLGMIPGLIGGLISAFKGRRKREITSQIEQYRNLQKREAELENLLANLPVY Brazilian scorpion Antiproliferative activity Not specified H157 Prostate cancer IC50 : 4.1 μM
dbacp01941 Brevinin-1H FALGAVTKVLPKLFCLITRKC Hainan Torrent Frog Membrane disruption MTT assay H157 Lung cancer IC50 : 3.37 to 5.87 µM
dbacp02108 cMastoparan-C(cMP-C) CLNLKALLAVAKKILC Synthetic construct Apoptosis MTT assay H157 Non-small cell Lung cancer IC50 : 7.02 μM
dbacp02652 Dermaseptin PS4 MDILKKSIFLVLFLGLVSLSICEEEKRENEDEEKQEDDEQSEEKRALWKTLLKHVGKAAGKAALNAVTDMVNQGEQ Sauvage's leaf frog Membrane disruption Lactate dehydrogenase (LDH) cytotoxicity assay, MTT assay H157 Glioma MIC : 10−9 to 10−4 M
dbacp02666 Dermaseptin-PD-1 GMWSKIKETAMAAAKEAAKAAGKTISDMIKQ Skin Secretion, Mexican leaf frog, Mexico, North America Destroy plasma membrane MTT assay H157 Human non-small cell Lung cancer IC50 : 10-4 and 10-9 M
dbacp02669 Dermaseptin-PD-2 GMWSKIKNAGKAAAKAAAKAAGKAALDAVSEAI Skin Secretion, Mexican leaf frog, Mexico, North America Destroy plasma membrane MTT assay H157 Human non-small cell lung cancer IC50 : 6.43 μM
dbacp02672 Dermaseptin-PD1 GMWSKIKETAMAAAKEAAKAAGKTISDMIKQ Mexican leaf frog Destroy plasma membrane MTT assay H157 Neuronal glioblastoma IC50 : 6.43 μM
dbacp02675 Dermaseptin-PD2 GMWSKIKNAGKAAAKAAAKAAGKAALDAVSEAI Mexican leaf frog Destroy plasma membrane MTT assay H157 Neuronal glioblastoma IC50 : 6.43 μM
dbacp02679 Dermaseptin-PH ALWKEVLKNAGKAALNEINNLVQ Northern orange-legged leaf frog Cell membrane permeabilization Bioactivity assessment assay, MTT cell proliferation assay H157 Not specified IC50 : 2.01 μM
dbacp02684 Dermaseptin-PH ALWKEVLKNAGKAALNEINNLV Orange-legged leaf frog, Northern orange-legged leaf frog, South America Cell membrane permeabilization MTT cell proliferation assay H157 Glioma IC50 : 2.01 μM
dbacp02691 Dermaseptin-PH MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay, Lactate dehydrogenase (LDH) assay NCl-H157 Lung cancer IC50 : 17.44 - 49.51 μM
dbacp02703 Dermaseptin-PH (DRS-PH) MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Brain tumor IC50 : 25.51 μM
dbacp02704 Dermaseptin-PH (DRS-PH) MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Breast cancer IC50 : 25.51 μM
dbacp02705 Dermaseptin-PH (DRS-PH) MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Pancreatic cancer IC50 : 25.51 μM
dbacp02706 Dermaseptin-PH (DRS-PH) MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Lung cancer IC50 : 25.51 μM
dbacp02707 Dermaseptin-PH (DRS-PH) MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Prostate cancer IC50 : 25.51 μM
dbacp02725 Dermaseptin-PS3 ALWKDILKNAGKAALNEINQIVQ Skin, the waxy monkey tree frog, South America Membrane rupture MTT assay H157 Lung cancer IC50 : 15.67 μM
dbacp02728 Dermaseptin-PS4 ALWKTLLKHVGKAAGKAALNAVTDMVNQ Waxy monkey tree frog Membrane disruption Lactate dehydrogenase (LDH) cytotoxicity assay, MTT assay H157 Glioma MIC : 10−9 to 10−4 M
dbacp02734 Dermaseptin-PT9 GLWSKIKDAAKTAGKAALGFVNEMV Brownbelly leaf frog Disruption of cell membranes MTT assay, Lactate dehydrogenase (LDH) assay NCl-H157 Lung cancer IC50 : 8.64 - 18.51 μM
dbacp02739 Dermaseptin-PT9 GLWSKIKDAAKTAGKAALGFVNEMV Skin secretion, Brownbelly leaf frog, Purchased in Peru, South America Disruption of cell membranes MTT assay, Lactate dehydrogenase (LDH) assay NCl-H157 Lung cancer IC50 : 8.64 - 18.51 μM
dbacp02779 Distinctin-Like-Peptide-PH NLVSALIEGRKYLKNVLKKLNRLKEKNKAKNSKENN Skin Secretion, Northern orange-legged leaf frog, South America Membrane lysis via pore formation MTT Cell viability assay, LDH assay H157 Prostate carcinoma MIC : ≥ 4.197 μM
dbacp03290 HECI TVLRGCWTFSFPPKPCI Hylarana erythraea Cell membrane disintegration MTT anti-proliferation assay H157 Lung cancer MIC : 1µM
dbacp03495 K8, 23-DPT9 MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Brain tumor IC50 : 9.88μM
dbacp03496 K8, 23-DPT9 MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Breast cancer IC50 : 9.88μM
dbacp03497 K8, 23-DPT9 MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Pancreatic cancer IC50 : 9.88μM
dbacp03498 K8, 23-DPT9 MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Lung cancer IC50 : 9.88μM
dbacp03499 K8, 23-DPT9 MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ Northern orange-legged leaf frog Disruption of cell membranes MTT assay H157 Prostate cancer IC50 : 9.88μM
dbacp03517 Kassiniatuerin-3 FIQHLIPLIPHAIQGIKDIF Senegal running frog, Africa Membranolytic mechanism MTT assay NCI-H157 Non-small cell Lung cancer IC50 : 21.54 µM
dbacp04573 Mastoparan-C LNLKALLAVAKKIL European hornet Apoptosis MTT assay H157 Non-small cell Lung cancer IC50 : 13.57 μM
dbacp04578 Mastoparan-Cimals. XXA; UCLL1c) LNLKALLAVAKKIL Venom, the European Hornet Inducing apoptosis MTT cell viability assay and Lactate dehydrogenase (LDH) leakage assay H157 Lung cancer MIC : 6.26 - 36.65 μM
dbacp04584 Mastoparan-Cimals. XXA; UCLL1c) LNLKALLAVAKKIL Venom, the European Hornet Inducing apoptosis MTT cell viability assay and Lactate dehydrogenase (LDH) leakage assay H157 Lung cancer IC50 : < 4 μM
dbacp05531 Phylloseptin-PBa1 FLSLIPHIASGIASLVKNF Burmeister's leaf frog, Brazil, South America Disruption of cell membranes MTT cell viability assay H157 Lung cancer IC50 : approx. 0.29 µM
dbacp05542 Phylloseptin-PBa2 FLSLLPHIASGIASLVSKF Burmeister's leaf frog, Brazil, South America Disruption of cell membranes MTT cell viability assay H157 Lung cancer IC50 : approx. 0.50 µM
dbacp05547 Phylloseptin-PHa FLSLIPAAISAVSALANHF Skin secretions, Orange-legged Leaf Frog, South America Membrane disruption MTT cell viability assay NCI-H157 Lung cancer IC50 : 14.10 μM
dbacp05549 Phylloseptin-PHa FLSLIPAAISAVSALANHF Northern orange-legged leaf frog Disruption of the membrane MTT assay, Lactate dehydrogenase (LDH) assay NCI-H157 Non-small-cell Lung cancer LD50 : < 5 µM
dbacp05554 Phylloseptin-PTa FLSLIPKIAGGIAALAKHL Skin secretions, the Brown-bellied Leaf Frog, South America Membrane disruption MTT Cell viability assay NCI-H157 Lung cancer IC50 : 6.73 μM
dbacp05793 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Lung cancer IC50 : 843.40 µM
dbacp05794 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Prostate cancer IC50 : 843.40 µM
dbacp05795 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Breast cancer IC50 : 843.40 µM
dbacp05796 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Lung cancer IC50 : 843.40 µM
dbacp05797 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Prostate cancer IC50 : 843.40 µM
dbacp05798 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Breast cancer IC50 : 843.40 µM
dbacp05799 R2PLx-22 GIMDTVKNAAKNLAGQLLDKLK Not found Inducing apoptosis MTT and LDH assay H157 Glioma IC50 : 843.40 µM
dbacp05877 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCKITAC Not found Inducing apoptosis MTT and LDH assay H157 Lung cancer IC50 : 5.90 µM
dbacp05878 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCKITAC Not found Inducing apoptosis MTT and LDH assay H157 Prostate cancer IC50 : 5.90 µM
dbacp05879 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCKITAC Not found Inducing apoptosis MTT and LDH assay H157 Breast cancer IC50 : 5.90 µM
dbacp05880 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCKITAC Not found Inducing apoptosis MTT and LDH assay H157 Glioma IC50 : 5.90 µM
dbacp05901 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCKITAC Gram-negative purple non-sulfur bacteria Inducing apoptosis MTT Cell viability assay and Lactate dehydrogenase (LDH) leakage assay H157 Lung IC50 : 5.90 µM
dbacp05906 Ranatuerin-2PLx GIMDTVKNAAKNLAGQLLDKLKCSITAC Skin secretions, the pickerel frog, North America Inducing apoptosis MTT Cell viability assay and Lactate dehydrogenase (LDH) leakage assay H157 Lung cancer IC50 : 5.90 µM
dbacp05984 S−24-R2PLx GIMDTVKNAAKNLAGQLLDKLKCSITAC Not found Inducing apoptosis MTT and LDH assay H157 Lung cancer IC50 : 58.18 µM
dbacp05985 S−24-R2PLx GIMDTVKNAAKNLAGQLLDKLKCSITAC Not found Inducing apoptosis MTT and LDH assay H157 Prostate cancer IC50 : 58.18 µM
dbacp05986 S−24-R2PLx GIMDTVKNAAKNLAGQLLDKLKCSITAC Not found Inducing apoptosis MTT and LDH assay H157 Breast cancer IC50 : 58.18 µM
dbacp05987 S−24-R2PLx GIMDTVKNAAKNLAGQLLDKLKCSITAC Not found Inducing apoptosis MTT and LDH assay H157 Glioma IC50 : 58.18 µM
dbacp06183 t Mastoparan-C(tMP-C, Tat (49-57)-Mastoparan-C) RKKRRQRRRLNLKALLAVAKKIL Synthetic construct Apoptosis inducing MTT assay H157 Non-small cell Lung cancer IC50 : 2.79 μM
dbacp06267 Temporin-PE FLPIVAKLLSGLL Skin secretions, Common water frog or green frog, Europe Destabilization of membranes MTT assay NCI-H157 Lung cancer TI : 10μM
dbacp06271 Temporin-PE FLPIVAKLLSGLL Skin secretions, Common water frog or green frog, Europe Destabilization of membranes MTT assay NCI-H157 Human neuronal glioblastoma TI : 10μM
dbacp06275 Temporin-PE FLPIVAKLLSGLL Skin secretions, Common water frog or green frog, Europe Destabilization of membranes MTT assay NCI-H157 Human neuronal glioblastoma TI : 10μM
dbacp06279 Temporin-PE FLPIVAKLLSGLL Skin secretions, Common water frog or green frog, Europe Destabilization of membranes MTT assay NCI-H157 Melanoma TI : 10μM
dbacp06283 Temporin-PE FLPIVAKLLSGLL Skin secretions, Common water frog or green frog, Europe Destabilization of membranes MTT assay NCI-H157 Lung cancer TI : approx. 10μM
dbacp06366 TsAP-2 FLGMIPGLIGGLISAFK Venom, the Brazilian yellow scorpion, South America Not specified MTT/MTS assay NCI-H157 Human squamous carcinoma IC50 : 4.1 µM
dbacp06374 TsAP-S1 FLSLIPKLVKKIIKAFK The iNot foundctive natural peptide TsAP-1 was made active by increasing 4 lysines and one leucine, template-based design Not specified MTT/MTS assay NCI-H157 Human squamous carcinoma IC50 : 55.9 µM