7 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp07111 | LyeTx-I-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Synergistic autophagic death via AKT inhibition. | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 2.47 µM |
| dbacp07309 | LyeTxI-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Apoptosis induction and immune modulation. | MTT assay | 4T1 | Breast Cancer | IC50 = 6.5 ± 5.30 µM |
| dbacp07310 | LyeTxI-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Apoptosis induction and immune modulation. | MTT assay | MCF-7 | Breast Cancer | IC50 = 7.34 ± 3.09 µM |
| dbacp07311 | LyeTxI-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Apoptosis induction and immune modulation. | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 5.77 ± 0.83 µM |
| dbacp07934 | LyeTx-I-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Membrane disruption, necroptosis, limited apoptosis | MTT/Resazurin dye assay | U-87-MG | Brain Tumor | IC50 = 29.20 ± 7.96 µM |
| dbacp07935 | LyeTx-I-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Membrane disruption, necroptosis, limited apoptosis | MTT/Resazurin dye assay | U-373-MG | Brain Tumor | IC50 = 20.94 ± 5.18 µM |
| dbacp07936 | LyeTx-I-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Membrane disruption, necroptosis, limited apoptosis | MTT/Resazurin dye assay | SH-SY5Y | Brain Tumor | IC50 = 93.80 ± 2.17 µM |