5 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp02459 | Chartergellus-CP1 peptide | IIGTILGLLKSLNH2 | Social wasp | Apoptosis inducing; Intracellular ROS formation | MTT assay | MNT-1 | Human melanoma | IC50 : 51.6 µg/mL |
| dbacp07029 | [G10a]-SHa | FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MNT-1 | Skin Cancer | IC50 = 15.25 ± 0.80 µM |
| dbacp07036 | [G10a]2-SHa | FLSGIVGMLaKLFKFLKaLMFLSGIVG | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MNT-1 | Skin Cancer | IC50 = 4.72 ± 0.36 µM |
| dbacp07043 | [G10a]3-SHa | FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MNT-1 | Skin Cancer | IC50 = 2.24 ± 0.05 µM |
| dbacp07049 | Jeff-[G10a]2-SHa | FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MNT-1 | Skin Cancer | IC50 = 57.03 ± 6.09 µM |