dbACP: A Comprehensive Database of Anti-Cancer Peptides

22 result(s) have been found!

Accession Name Sequence Source/Organism Mechanism Assay Type Cell Line Cancer Type Activity
dbacp05312 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer 24.2 % inhibition of cell proliferation at 1 nM
dbacp05313 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer 37.8 % inhibition of cell proliferation at 10 nM
dbacp05314 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer 48.2 % inhibition of cell proliferation at 100 nM
dbacp05315 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer 59.6 % inhibition of cell proliferation at 1 µM
dbacp05316 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer 84.5 % inhibition of cell proliferation at 10 µM
dbacp05328 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay MiaPaCa.2 Pancreatic cancer ED50 : 0.210 µM
dbacp05587 PNC-28 ETFSDLWKLL Ant Membrane disruption MTT/MTS assay MiaPaCa.2 Pancreatic cancer Cytotoxicity : 80µg/ml
dbacp06652 LUNA18 Not Available Synthetic Not available CellTiter-Glo Cell Viability assay MiaPaCa.2 Pancreatic Cancer IC50 = 1.4 ± 0.2 nmol/L
dbacp07027 [G10a]-SHa FLSGIVGMLaKLF Analog of temporin SHa Dendrimerization enhances stability, selectivity, anticancer efficacy Resazurin dye assay MiaPaCa.2 Pancreatic Cancer IC50 = 22.36 ± 6.07 µM
dbacp07034 [G10a]2-SHa FLSGIVGMLaKLFKFLKaLMFLSGIVG Analog of temporin SHa Dendrimerization enhances stability, selectivity, anticancer efficacy Resazurin dye assay MiaPaCa.2 Pancreatic Cancer IC50 = 8.71 ± 0.35 µM
dbacp07041 [G10a]3-SHa FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK Analog of temporin SHa Dendrimerization enhances stability, selectivity, anticancer efficacy Resazurin dye assay MiaPaCa.2 Pancreatic Cancer IC50 = 6.94 ± 0.27 µM
dbacp07047 Jeff-[G10a]2-SHa FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF Analog of temporin SHa Dendrimerization enhances stability, selectivity, anticancer efficacy Resazurin dye assay MiaPaCa.2 Pancreatic Cancer IC50 = 57.45 ± 6.03 µM
dbacp08175 Peptide - 1 GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKK Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 = 7.3 µM
dbacp08187 Peptide - 2 GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRR Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 = 5.0 µM
dbacp08195 Peptide - 3 GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- Orn Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 = 3.6 µM
dbacp08203 Peptide - 4 GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-Dab Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 = 4.4 µM
dbacp08211 Peptide - 6 GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM
dbacp08219 Peptide - 7 GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRR Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM
dbacp08227 Peptide - 8 GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKK Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM
dbacp08235 Peptide - 9 GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKK Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM
dbacp08243 Peptide - 10 GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM
dbacp08251 Peptide - 11 KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c) Synthetic Not Available CellTiter-Glo assay MiaPaCa.2 Pancreatic Cancer IC50 > 7.5 µM