24 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp08112 | FR-15 | FRRFFKWFRRFFKFF | Synthetic | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 3.15 μM |
| dbacp08113 | FR-15 | FRRFFKWFRRFFKFF | Synthetic | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 4.9 μM |
| dbacp08114 | FR-15 | FRRFFKWFRRFFKFF | Synthetic | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 6.7 μM |
| dbacp08115 | FR-15 | FRRFFKWFRRFFKFF | Synthetic | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 2.5 μM |
| dbacp08116 | FR4P | FRRPFKWFRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 6.3 μM |
| dbacp08117 | FR4P | FRRPFKWFRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 7.7 μM |
| dbacp08118 | FR4P | FRRPFKWFRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 9.4 μM |
| dbacp08119 | FR4P | FRRPFKWFRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 2.5 μM |
| dbacp08120 | FR8P | FRRFFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 6.4 μM |
| dbacp08121 | FR8P | FRRFFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 10.5 μM |
| dbacp08122 | FR8P | FRRFFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 10.8 μM |
| dbacp08123 | FR8P | FRRFFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 4.2 μM |
| dbacp08124 | FR11P | FRRFFKWFRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 7 μM |
| dbacp08125 | FR11P | FRRFFKWFRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 11 μM |
| dbacp08126 | FR11P | FRRFFKWFRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 12.9 μM |
| dbacp08127 | FR11P | FRRFFKWFRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 4.8 μM |
| dbacp08128 | FR4,8P | FRRPFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 15.4 μM |
| dbacp08129 | FR4,8P | FRRPFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 13.8 μM |
| dbacp08130 | FR4,8P | FRRPFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 15.3 μM |
| dbacp08131 | FR4,8P | FRRPFKWPRRFFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 5 μM |
| dbacp08132 | FR8,11P | FRRFFKWPRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | MDA-MB-231 | Breast Cancer | IC50 = 27 μM |
| dbacp08133 | FR8,11P | FRRFFKWPRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HeLa | Cervical Cancer | IC50 = 18.9 μM |
| dbacp08134 | FR8,11P | FRRFFKWPRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | DLD-1 | Colon Cancer | IC50 = 22 μM |
| dbacp08135 | FR8,11P | FRRFFKWPRRPFKFF | Analogue of FR-15 | Proline-substituted AMP triggers mitochondrial apoptosis | MTT assay | HepG-2 | Liver Cancer | IC50 = 15 μM |