dbACP: A Comprehensive Database of Anti-Cancer Peptides

21 result(s) have been found!

Accession Name Sequence Source/Organism Mechanism Assay Type Cell Line Cancer Type Activity
dbacp04794 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer > 100% cell viability at 5 µM
dbacp04795 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 60% cell viability at 50 µM
dbacp04800 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer > 100% cell viability at 5 µM
dbacp04801 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 60% cell viability at 50 µM
dbacp04806 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 100% cell viability at 5 µM
dbacp04807 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 40% cell viability at 50 µM
dbacp04812 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 100% cell viability at 5 µM
dbacp04813 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 40% cell viability at 50 µM
dbacp04818 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer MIC : 5 µM
dbacp04867 NK-2 KILRGVCKKIMRTFLRRISKDILTGKK NK-lysin Cell membrane disintegration PI-uptake assay SW-480 Leukemia cancer LD50 : 1-4 µM
dbacp06737 Aurein 1.2_mutant (Aurm) GLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 51.63% cell viability
dbacp06739 Aurein 1.2_R5 (R5-Aur) RRRRRGLFDIIKKIAESF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 43.89% cell viability
dbacp06741 Aurein 1.2_mutant_R5 (R5-Aurm) RRRRRGLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 40.62% cell viability
dbacp07085 HB43 FAKLLAKLAKKLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 12 ± 4 μM
dbacp07089 HB43-mut2 FAKLLAKLAKLLK Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 34 ± 2 μM
dbacp07093 HB43-mut3 FAKLLAKLARRLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 8 ± 1 μM
dbacp07287 P264-G274 PARDVLNTTSG Parasporin-2Aa1 h-APN receptor–mediated apoptosis induction. Sulforhodamine B assay SW-480 Colorectal Cancer EC50 = 90.98 ± 0.75 µM
dbacp07289 Loop1-PS2Aa NNETYFNAVKP Parasporin-2Aa1 h-APN receptor–mediated apoptosis induction. Sulforhodamine B assay SW-480 Colorectal Cancer EC50 = 23.76 ± 1.25 µM
dbacp07291 Loop2-PS2Aa TYFNAVKPPITA Parasporin-2Aa1 h-APN receptor–mediated apoptosis induction. Sulforhodamine B assay SW-480 Colorectal Cancer EC50 = 92.99 ± 0.98 µM
dbacp07293 Loop1-HCoV-229E FKPQSGGGKCF Alphacoronavirus (HCoV-229E) h-APN receptor–mediated apoptosis induction. Sulforhodamine B assay SW-480 Colorectal Cancer EC50 = 125.0 ± 1.32 µM
dbacp07294 A4W-GGN5 FLGWLFKVASK Gaegurin 5 h-APN receptor–mediated apoptosis induction. Sulforhodamine B assay SW-480 Colorectal Cancer EC50 = 98.63 ± 1.17 µM