28 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp06865 | Pep-1-Phor21 | CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK | Hybrid peptide PEP1 and Phor 21 | Not available | AlamarBlue assay | LNCaP | Liver Cancer | IC50 = 55.13 ± 13.56 µM |
| dbacp06866 | Pep-1-Phor21 | CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK | Hybrid peptide PEP1 and Phor 21 | Not available | AlamarBlue assay | DU-145 | Prostrate Cancer | IC50 = 2.57 ± 2.02 µM |
| dbacp06867 | Pep-1-Phor21 | CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK | Hybrid peptide PEP1 and Phor 21 | Not available | AlamarBlue assay | PC-3 | Prostrate Cancer | IC50 ≤ 0.6 μM |
| dbacp07085 | HB43 | FAKLLAKLAKKLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-480 | Colon Cancer | IC50 = 12 ± 4 μM |
| dbacp07086 | HB43 | FAKLLAKLAKKLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-620 | Colon Cancer | IC50 = 10 ± 1 μM |
| dbacp07087 | HB43 | FAKLLAKLAKKLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | HT-29 | Colon Cancer | IC50 = 11 ± 1 μM |
| dbacp07088 | HB43 | FAKLLAKLAKKLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | MDA-MB-231 | Breast Cancer | 50% cell viability at 20 μM |
| dbacp07089 | HB43-mut2 | FAKLLAKLAKLLK | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-480 | Colon Cancer | IC50 = 34 ± 2 μM |
| dbacp07090 | HB43-mut2 | FAKLLAKLAKLLK | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-620 | Colon Cancer | IC50 = 40 ± 3 μM |
| dbacp07091 | HB43-mut2 | FAKLLAKLAKLLK | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | HT-29 | Colon Cancer | IC50 = 50 ± 3 μM |
| dbacp07092 | HB43-mut2 | FAKLLAKLAKLLK | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | MDA-MB-231 | Breast Cancer | 80% cell viability at 20 μM |
| dbacp07093 | HB43-mut3 | FAKLLAKLARRLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-480 | Colon Cancer | IC50 = 8 ± 1 μM |
| dbacp07094 | HB43-mut3 | FAKLLAKLARRLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | SW-620 | Colon Cancer | IC50 = 9 ± 1 μM |
| dbacp07095 | HB43-mut3 | FAKLLAKLARRLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | HT-29 | Colon Cancer | IC50 = 9 ± 1 μM |
| dbacp07096 | HB43-mut3 | FAKLLAKLARRLL | Synthetic | Motif-driven membrane insertion triggers cytotoxicity | AlamarBlue assay | MDA-MB-231 | Breast Cancer | 75% cell viability at 20 μM |
| dbacp08364 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | RG1 | Glioblastoma | EC50 ~ 7 μM |
| dbacp08365 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | GMB-27 | Glioblastoma | EC50 ~ 7.5 μM |
| dbacp08366 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | 12015 | Glioblastoma | EC50 ~ 10 μM |
| dbacp08367 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | 12089 | Glioblastoma | EC50 ~ 4 μM |
| dbacp08368 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | RG6 | Glioblastoma | EC50 ~ 5 μM |
| dbacp08369 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | RG4 | Glioblastoma | EC50 ~ 5 μM |
| dbacp08370 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | RG5 | Glioblastoma | EC50 ~ 7 μM |
| dbacp08371 | IDP-NS10 | AALVVILKKATEYVHS | Synthetic | Not Available | AlamarBlue assay | 12053 | Glioblastoma | EC50 ~ 50 μM |
| dbacp08372 | IDP-NS02 | RQRRNDLRSSFLTLRDH | Synthetic | Not Available | AlamarBlue assay | NCI-H524 | Lung Cancer | EC50 ~ 5 μM |
| dbacp08373 | IDP-NS16 | RQRRNDLRSSFLTLRDH | Synthetic | Not Available | AlamarBlue assay | RG1 | Glioblastoma | EC50 ~ 15 μM |
| dbacp08374 | IDP-NS16 | RQRRNDLRSSFLTLRDH | Synthetic | Not Available | AlamarBlue assay | 12053 | Glioblastoma | EC50 ~ 10 μM |
| dbacp08375 | IDP-Na05 | RRNDLRSSFLTLRDHVP | Synthetic | Not Available | AlamarBlue assay | RG1 | Glioblastoma | EC50 ~ 10 μM |
| dbacp08376 | IDP-NLCa02 | RQIKIWFQNRRMKWKKRQRRNDLRSSFLTLRDHVP | Synthetic | Not Available | AlamarBlue assay | RG1 | Glioblastoma | EC50 ~ 5 μM |