dbACP: A Comprehensive Database of Anti-Cancer Peptides

41 result(s) have been found!

Accession Name Sequence Source/Organism Mechanism Assay Type Cell Line Cancer Type Activity
dbacp00725 6,7-dimethyl-8-ribityllumazine synthase 2 MNQSCPNKTSFKIAFIQARWHADIVDEARKSFVAELAAKTGGSVEVEIFDVPGAYEIPLHAKTLARTGRYAAIVGAAFVIDGGIYRHDFVATAVINGMMQVQLETEVPVLSVVLTPHHFHESKEHHDFFHAHFKVKGVEAAHAALQIVSERSRIAALV Not found Apoptosis inducing Apoptosis assay B16 Melanoma Not found
dbacp01596 BF-30 KFFRKLKKSVKKRAKEFFKKPRVIGVSIPF Banded krait Cytoplasmic membrane permeabilization and DNAspecified-binding Lactate dehydrogenase release assay, DNA retardation assay, Real-time PCR, Western blot, wound healing assay, and chick embryo chorioallantoic membrane assay B16F10 Human Colon cancer IC50 : 7.3 μM
dbacp01597 BF-30 KFFRKLKKSVKKRAKEFFKKPRVIGVSIPF Banded krait Cytoplasmic membrane permeabilization and DNAspecified-binding Lactate dehydrogenase release assay, DNA retardation assay, Real-time PCR, Western blot, wound healing assay, and chick embryo chorioallantoic membrane assay B16 Human Cervical cancer IC50 : 13.9 μM
dbacp01609 Bim EIWIAQELRRIGDEFNAYYAR BH3-only, Direct activators, BIM analogues Inducing apoptosis Not specified B16 Melanoma Not found
dbacp01951 Brevinin-1RL1 FFPLIAGLAARFLPKIFCSITKRC Not found Inducing apoptosis Cell death assay B16F10 Not specified IC50 : 6.65 ± 0.33 μM
dbacp02270 Camel KWKLFKKIGAVLKVL Ceropin-Melittin hybrid Cell swelling and rupture of the plasma membrane MTT/MTS assay B16-F10 Skin cancer LC50 : 1.75 µM
dbacp02480 ChMAP-28 GRFKRFRKKLKRLWHKVGPFVGPILHY Domestic goat Cause cell membrane permeability; Induce necrotic death Cytotoxic Activity assay, Lactate dehydrogenase (LDH)-Releaseassay, MTT assay B16F1 Murine melanoma IC50 : 4.82 ± 1.01μM
dbacp02813 Drosophila Antennapedia homodomain PFV CALNNPFVYLI Fruit fly homodomain PFV Cell membrane disintegration SPR assay B16 Mouse melanoma Not found
dbacp02930 Figainin 1 FIGTLIPLALGALTKLFK Chaco tree frog Membrane disruption and cell lysis MTT/MTS assay B16F10 Leukemia IC50 : 10.5 µM
dbacp02936 Figainin 1 MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG Chaco tree frog Anti-proliferative action MTT/MTS assay B16F10 Skin cancer IC50 : 10.5 µM
dbacp02937 Figainin 1 MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG Chaco tree frog Anti-proliferative action MTT/MTS assay B16F10 Breast cancer IC50 : 10.5 µM
dbacp02938 Figainin 1 MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG Chaco tree frog Anti-proliferative action MTT/MTS assay B16F10 Cervical cancer IC50 : 10.5 µM
dbacp02946 Figainin 1 FIGTLIPLALGALTKLFK Skin secretions, Chaco tree frog, South America Membrane disruption MTT/MTS assay B16F10 Leukemia IC50 : 10.5 µM
dbacp02949 Figainin 2 FLGAILKIGHALAKTVLPMVTNAFKPKQ Skin secretions, Chaco tree frog, South America Cell membrane interaction; Necrosis; Apoptosis MTT/MTS assay B16F10 Murien melanoma IC50 : 12.8 µM
dbacp02951 Figainin 2 MAFLKKSLFLVLFLGIVSLSVCEEEKREGEEKEEKREEEEGKEENEDGNEEHKEKRFLGAILKIGHALAKTVLPMVTNAFKPKQ Chaco tree frog Necrosis; Apoptosis MTT/MTS assay B16F10 Skin cancer IC50 : 12.8 µM
dbacp02952 Figainin 2 MAFLKKSLFLVLFLGIVSLSVCEEEKREGEEKEEKREEEEGKEENEDGNEEHKEKRFLGAILKIGHALAKTVLPMVTNAFKPKQ Chaco tree frog Necrosis; Apoptosis MTT/MTS assay B16F10 Breast cancer IC50 : 12.8 µM
dbacp03328 HSP70 peptide ACFAEKFKEAVKDYFAKFWD-GSG-TKDNNLLGRFELSG Not found Immune response to tumor cell recognition Cytotoxic assay, Lactate dehydrogenase (LDH) release assay B16OVA Necroptotic cancer Not found
dbacp03531 L-amino acid oxidase (CC-LAAO) (LAO) (EC 1.4.3.2) MNVFFMFSLLFLAALESCADDKNPLEEEFFEADYEEFLLIAKNGLQQTSNPKRVVIVGAGMSGLSAAYVLAKTGHEVILLEASERVGGRVSTYRNDQEGWYANLGPMRLPERHRIVREYIRKFGLQLNEFSQENENAWYFIKNIRKRVGEVNKDPGVLEYPVKPSEKGKSAPQLYRDSLQKIIEEYGRSNCSYILNKYDTYSTKDYLIKEGNLSPGAVDMVGDLLNEDSGYYVSFIESLKPDDIFAYENRFDEIVGGFDKLPTSMYQAIQEKVRLNVRVIKIQQDVKEVTVTYQTPAKNLSYVTADYVIVCTTSGAARRIKFEPPLPLKKAHALRSVHYRSGTKIFLTCTKKFWEDDGIHGGKSITDRPSRLIHYPNHNFPNGIGVLVIFTIADDADFFLALDNKTIADIVIHDLSLIHQLPKEKIRDLCYVSMIQKWSLDKYAMGGITTFTPYQFQHFSEALTAPVDRIYFAGEYTAQAHGWIDSTIKSGLTAARDVNRASENPSGIHLSNDNEL Horned desert vip Cytotoxic effects MTT assay B16F10 Not found IC50 : 2 µg/mL
dbacp03539 L-amino-acid oxidase (BatroxLAAO) (LAO) (EC 1.4.3.2) MNVFFTFSLLFLAALGSCADDRNPLEECFRETDYEEFLEIAKNGLSTTSNPKRVVIVGAGMSGLSAAYVLANAGHQVTVLEASERAGGRVKTYRNEKEGWYANLGPMRLPEKHRIVREYIRKFDLQLNEFSQENENAWYFIKNIRKRVGEVNKDPGVLEYPVKPSEVGKSAGQLYEESLQKAVEELRRTNCSYMLNKYDTYSTKEYLLKEGNLSPGAVDMIGDLLNEDSGYYVSFIESLKHDDIFAYEKRFDEIVGGMDKLPTSMYQAIQEKVHLNARVIKIQQDVKEVTVTYQTSEKETLSVTADYVIVCTTSRAARRIKFEPPLPPKKAHALRSVHYRSGTKIFLTCTKKFWEDDGIHGGKSTTDLPSRFIYYPNHNFPNGVGVIIAYGIGDDANYFQALDFEDCGDIVINDLSLIHQLPKEEIQAICRPSMIQRWSLDKYAMGGITTFTPYQFQHFSEALTAPVDRIYFAGEYTAQAHGWIDSTIKSGLRAARDVNRASEIKK Common lancehead Inducing apoptosis MTT assay B16F10 Not found Not found
dbacp03600 l3,10,13K7,8K4R2L9 KLlRLLkkLlRLlLK Diastereomeric peptide Plasma membrane perturbation; Necrosis XTT assay B16-F10 Skin cancer LC50 : 2.5 µM
dbacp03602 l3,4,8,10K5L7 KlllKLKlKlLK Diastereomeric peptide Plasma membrane perturbation; Necrosis XTT assay B16-F10 Skin cancer LC50 : 100 µM
dbacp04302 LTX-315 KKWWKKW-Dip-K Synthetic peptide Necrosis MTT/MTS assay B16F1 Skin cancer IC50 : 13.3 µM
dbacp05094 P7 PLLQATLGGGS Not found Apoptosis inducing WST-1 assay B16-F10 Skin cancer IC50 : 1 µM
dbacp05241 pentadactylin GLLDTLKGAAKNVVGSLASKVMEKL Not found Inducing apoptosis MTT assay B16F10 Melanoma IC50 : 25.7 µM
dbacp05441 Peptide-20 CSSRTMHHC Synthetic Peptide Inducing apoptosis MTT/MTS assay B16F10-Nex 2 Skin cancer At 100 µM 50% viablity
dbacp05505 PHP ITCPQVTQSLAPCVPYLISG Plant sources Inducing apoptosis MTT assay B16 Not found IC50 : 1.47 µM
dbacp05820 R8 CALRRRRRRRR Not found Cell membrane disintegration SPR assay B16 Mouse Melanoma Not found
dbacp05917 Raniseptin-3 AWLDKLKSIGKVVGKVAIGVAKNLLNPQ Skin secretion, Chaco tree frog, South America Disrupting cancer cell membranes MTT and LDH assay B16F10 Murine melanoma IC50 : 6.56 μM
dbacp05919 Raniseptin-6 ALLDKLKSLGKVVGKVALGVVQNYLNPRQ Skin secretion, Chaco tree frog, South America Disrupting cancer cell membranes MTT and LDH assay B16F10 Murine melanoma IC50 : 8.69 μM
dbacp05966 RGD-tachyplesin CRGDCGGKWCFRVCYRGICYRRCR Not found Inducing apoptosis Not specified B16 Prostate cancer Not found
dbacp06157 StigA16 FFKLIPKLVKGLISAF Amino acid substitution, amino acid truncation, animal-derived, natural derivative Disruption of cell membrane MTT assay B16 Human pancreas adenocarcinoma IC 50 : 13.01 μM
dbacp06162 StigA6 FFSLIPKLVKGLISAFK Amino acid substitution, animal-derived, natural derivative Disruption of cell membrane MTT assay B16 Human pancreas adenocarcinoma IC 50 : 14.01 μM
dbacp06202 TAT-Bim (145-165) RKKRRQ(orn)RRREIWIAQELRRIGDEFNAYYAR BH3-only, Direct activators, BIM analogues Inducing apoptosis Not specified B16 Melanoma Not found
dbacp06404 Tyroserleutide YSL Synthetic Peptide Necrosis; Immune regulation MTT/MTS assay B16-F10 Skin cancer 49.4% Cytotoxic at 0.1 µg/ml
dbacp06405 Tyroserleutide YSL Synthetic Peptide Necrosis; Immune regulation MTT/MTS assay B16-F10 Skin cancer 51.2% Cytotoxic at 1 µg/ml
dbacp06406 Tyroserleutide YSL Synthetic Peptide Necrosis; Immune regulation MTT/MTS assay B16-F10 Skin cancer 53.0% Cytotoxic at 10 µg/ml
dbacp06407 Tyroserleutide YSL Synthetic Peptide Necrosis; Immune regulation MTT/MTS assay B16-F10 Skin cancer 61.2% Cytotoxic at 100 µg/ml
dbacp06735 NKL-WT KLKSKLMVVCNKIGLLKSLCRKFVKSH Trematomus bernacchii Apoptosis inducing luciferase-based ATPlite assay B16-F10 Skin Cancer ATP level = 0.753 ± 0.254 at 40 μM
dbacp06736 NKL-MUT KLKSKLMVVANKIGLLKSLARKFVKSH Trematomus bernacchii Apoptosis inducing luciferase-based ATPlite assay B16-F10 Skin Cancer ATP level = 0.023 ± 0.007 at 40 μM
dbacp07239 RB4 MADSERLSAPGCWAACTNFSRTRK Derived from protein PLP2 F-actin modulation induces necrotic death. MTT assay B16-F10-Nex 2 Skin Cancer EC50 = 0.263 ± 0.585 mol/L × 10-3
dbacp07493 Figainin 1 FIGTLIPLALGALTKLFK Boana raniceps Membrane disruption, α-helix mediated MTT assay B16-F10 Skin Cancer IC50 = 10.5 µM