dbACP: A Comprehensive Database of Anti-Cancer Peptides

630 result(s) have been found!

Accession Name Sequence Source/Organism Mechanism Assay Type Cell Line Cancer Type Activity
dbacp00003 Citropin modified peptide-3 GLFAVIKKVASVIGGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 6 M
dbacp00012 Citropin modified peptide-5 GLFDVIKAVASVIGGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00021 Citropin modified peptide-7 GLFDVIKKVAAVIGGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00039 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 9.8% inhibition at 10-6 M
dbacp00040 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 1.6% inhibition at 10-5 M
dbacp00041 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 5.4% inhibition at 10-4 M
dbacp00042 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 26.5% inhibition at 10-3 M
dbacp00043 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 12.9% inhibition at 10-6 M
dbacp00044 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 16.5% inhibition at 10-5 M
dbacp00045 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 28.1% inhibition at 10-4 M
dbacp00046 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 58.2% inhibition at 10-3 M
dbacp00047 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 3.5% inhibition at 10-6 M
dbacp00048 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 22.7% inhibition at 10-5 M
dbacp00049 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 18.9% inhibition at 10-4 M
dbacp00050 Enkephalins7 analogue-8 YA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 26.4% inhibition at 10-3 M
dbacp00063 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 4.9% inhibition at 10-6 M
dbacp00064 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 8.9% inhibition at 10-5 M
dbacp00065 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 3.4% inhibition at 10-4 M
dbacp00066 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 20.8% inhibition at 10-3 M
dbacp00067 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 10.5% inhibition at 10-6 M
dbacp00068 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 21.9% inhibition at 10-5 M
dbacp00069 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 11.8% inhibition at 10-4 M
dbacp00070 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 17.9% inhibition at 10-3 M
dbacp00071 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 3.7% inhibition at 10-6 M
dbacp00072 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 16.5% inhibition at 10-5 M
dbacp00073 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.4% inhibition at 10-4 M
dbacp00074 Enkephalins7 analogue-9 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 14.5% inhibition at 10-3 M
dbacp00090 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 0.7% inhibition at 10-6 M
dbacp00091 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 8.3% inhibition at 10-5 M
dbacp00092 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 10.5% inhibition at 10-4 M
dbacp00093 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 21.8% inhibition at 10-3 M
dbacp00094 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 10.7% inhibition at 10-6 M
dbacp00095 Enkephalins7 analogue-10 YSA* Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 10.0% inhibition at 10-5 M
dbacp00100 Citropin modified peptide-11 GLFDVIKKVASVIKGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00109 Citropin modified peptide-13 GLFDVIKKVASVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00118 Citropin modified peptide-14 GLFDVIAKVASVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00137 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 5.4% inhibition at 10-6 M
dbacp00138 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 7.4% inhibition at 10-5 M
dbacp00139 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 9.5% inhibition at 10-4 M
dbacp00140 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 15.7% inhibition at 10-3 M
dbacp00141 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 13.6% inhibition at 10-6 M
dbacp00142 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 20.4% inhibition at 10-5 M
dbacp00143 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 14.4% inhibition at 10-4 M
dbacp00144 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 23.4% inhibition at 10-3 M
dbacp00145 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 2.2% inhibition at 10-6 M
dbacp00146 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 4.2% inhibition at 10-5 M
dbacp00147 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 6.4% inhibition at 10-4 M
dbacp00148 Enkephalins7 analogue-15 YSA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 6.2% inhibition at 10-3 M
dbacp00152 Citropin modified peptide-15 GLFAVIKKVASVIKGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00170 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 7.6% inhibition at 10-6 M
dbacp00171 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 3.8% inhibition at 10-5 M
dbacp00172 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 12.4% inhibition at 10-4 M
dbacp00173 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 22.4% inhibition at 10-3 M
dbacp00174 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 17.0% inhibition at 10-6 M
dbacp00175 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 13.5% inhibition at 10-5 M
dbacp00176 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 13.5% inhibition at 10-4 M
dbacp00177 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 25.3% inhibition at 10-3 M
dbacp00178 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.1% inhibition at 10-6 M
dbacp00179 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 6.9% inhibition at 10-5 M
dbacp00180 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.1% inhibition at 10-4 M
dbacp00181 Enkephalins7 analogue-16 YRA*G Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.6% inhibition at 10-3 M
dbacp00185 Citropin modified peptide-16 GLFAVIKKVASVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00204 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 3.3% inhibition at 10-6 M
dbacp00205 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 11.0% inhibition at 10-5M
dbacp00206 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 7.9% inhibition at 10-4 M
dbacp00207 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 23.7% inhibition at 10-3 M
dbacp00208 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 12.2% inhibition at 10-6 M
dbacp00209 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 15.5% inhibition at 10-5 M
dbacp00210 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 24.7% inhibition at 10-4 M
dbacp00211 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 29.0% inhibition at 10-3 M
dbacp00212 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 3.0% inhibition at 10-6 M
dbacp00213 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.4% inhibition at 10-5 M
dbacp00214 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 18.5% inhibition at 10-4 M
dbacp00215 Enkephalins7 analogue-17 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 10.6% inhibition at 10-3 M
dbacp00219 Citropin modified peptide-17 GLFAVIKKVAAVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00238 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 16.2% inhibition at 10-6 M
dbacp00239 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 6.6% inhibition at 10-5 M
dbacp00240 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 5.1% inhibition at 10-4 M
dbacp00241 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 14.5% inhibition at 10-3 M
dbacp00242 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 26.4% inhibition at 10-6 M
dbacp00243 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 13.1% inhibition at 10-5 M
dbacp00244 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 14.6% inhibition at 10-4 M
dbacp00245 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay SW-620 Colon cancer 38.4% inhibition at 10-3 M
dbacp00246 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 17.7% inhibition at 10-6 M
dbacp00247 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 10.9% inhibition at 10-5 M
dbacp00248 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 12.1% inhibition at 10-4 M
dbacp00249 Enkephalins7 analogue-18 YA*GFM Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 8.1% inhibition at 10-3 M
dbacp00254 Citropin modified peptide-18 GLFAVIKKVAAVIRRL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00263 Citropin modified peptide-19 GLFAVIKKVAKVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00272 Citropin modified peptide-22 GLFKVIKKVASVIGGL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00285 Enkephalins7 analogue-23 YGGFMA* Synthetic Peptide Apoptosis inducing MTT/MTS assay HT-29 Colon cancer 9.2% inhibition at 10-3 M
dbacp00286 Enkephalins7 analogue-23 YGGFMA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 11.08% inhibition at 10-5 M
dbacp00287 Enkephalins7 analogue-23 YGGFMA* Synthetic Peptide Apoptosis inducing MTT/MTS assay CaCo-2 Colon cancer 47.0% inhibition at 10-3 M
dbacp00294 Citropin modified peptide-23 GLFKVIKKVAKVIKKL Amphibian skin secretions Penetration and disruption of the membrane Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp00614 [ribosomal protein uS5]-alanine N-acetyltransferase MPHTPSRLLAEGPRVGIRHFTLADGPEFTARARESKDLHHPWLFPPDSPQTYEAYAARLIEDRTKAGFLVCERDTAGTSEGTRGGGPIAGFVNINNIVEGGFLSGALGYGAFAHAAGRGLMREGLDLVVRYAFGPMRLHRLEINVQPGNAASIALARACGFHLEGFSPRMLHIDGAWRDHQRWALTAETAASG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00714 2,3-dihydroxybenzoate-AMP ligase MTETQPTWSEAESARYRAAGHWQGVTFGARLRQAGAEHAQRVALVDGNRRWTYADLDAEADRVAAGLRGLGVERGDRVVLQLPNCAEFVLAWFGLQRLGAVPVHAMPGHRSREIGHLVRLSDAVACVVPDLHARFDHRRLMSDVRAELGPDGPLRHVVVVGDPGPYDGFVPFDALRESGGRGPSAPVSDSDSADPDPGGLALLLLSGGTTGLPKLIPRTHDDYAYNARACAGVCALDTRSVYLAVLPLGFNFTFACPGVLGTLMAGGTVVIAPDPSPQTAFALIEREGVTLTSLTPPLVPHWTDEAASGSWDLGSLAVVQVGGARLPEDHARRLGPALGARVQQVFGMAEGLINLTRLDDAEDLVCTTQGRPASPDDEILVVDAGGRPVPDGTAGELLTRGPYTLRGYYRAEAHNRTAFTPDGYYRSGDVVRRLPSGHLVVVGRIKDQINRGGEKIPAVEVEEELLTHPAVTAAALVGVPDERWGERSVAFVVCTGTAPGAREVAAHLASRGLAGYKAPDEIVQVPGLPLTAVGKVDKAALARRSEG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00719 3A LTAEHYAAQATS Not found Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : >100 µM
dbacp00766 A specific Eps8/EGFR Inhibitor Peptide 327 EFLDCFQKF A specific Eps8/EGFR Inhibitor Peptide 327 Immune response to tumor cell recognition Lactate dehydrogenase (LDH)-release assay Colo320 Colon cancer IC50 : 83.10 ± 1.41 μM
dbacp00768 A specific Eps8/EGFR Inhibitor Peptide 327 EFLDCFQKF A specific Eps8/EGFR Inhibitor Peptide 327 Immune response to tumor cell recognition Lactate dehydrogenase (LDH)-release assay SW620 Colon cancer IC50 : 102.35 ± 4.66 μM
dbacp00813 A5 KAQIRAMECNIL Cyclin B (285-296) Apoptosis inducing MTT/MTS assay HCT-116 Colon cancer Not found
dbacp00837 ABC transporter ATP-binding protein MTPPKDSTMDPLVRLDGVHVRHRARSGGLLRRDSVHALTDVGLEVRRGEILGLVGESGCGKSTLARVVTGLQRPTEGRVSFRGRDLWTMSGAERRTGFGAAVGVVFQDASTALNPRLPVRRILRDPLDVHDRGTRAEREERVEELLDLVGLPGHTLQALPGQLSGGQRQRVAIARALALEPELIVADEPTSALDVSVRAQILNLLVDLRARLGLGMVFISHDVQTVRHLADRVAVLYLGRVVEEGGASEVLGASRHPYTEALLSATPSLLERPERIVLHGPVPSATNPPSGCPFRTRCWKADDACATAFPAAAEGPGGHRWHCVHPRESGVPREATSAK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00842 ABC transporter ATP-binding protein MTTTGPPTRSDADTPALDVEGLCVELSTPSGTVRAVDGVSFSVRRGRTLALLGESGCGKSMTALSVVGLLDPAAAVTGGAVRVRGDDTLRMSPAQRRRLAGPVLSIVFQDALTALNPVQPVGRQIGEPFRIHRRLSRRQAREKAIELMTRVGIPEPRQRARSYPHQFSGGMRQRLLIAMAVALAPDVLIADEPTTALDVTVQAQIMRLLRDLQDERDMAVVLITHDLAVVAQRADDVVVMYAGTVVENGPVRDVFAAPRHPYTRGLLDSVPEDSVRGRPLPAVPGSPPELSAVPAGCVFQARCPLVRERCVRERPVPRPAGEGRSAACHFSEELDRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00847 ABC transporter ATP-binding protein MTTQTKPEEAPAAAAGNAFLSVRDLKVHFSTEGGVVKAVDGLSFDLERGKTLGIVGESGSGKSVTNLAVLGLHDRRKTAVDGSITLDGQELTDASEKQLETLRGKKMAMIFQDALTALSPYYTVGRQIGEPFMKHNGASKKDARVRAIDLLQKVGIPHPQKRVDDYPHQFSGGMRQRAMIAMALSCDPDLLIADEPTTALDVTVQAQILDLLKDLQQEFGSAIIMITHDLGVVGnMADDILVMYAGRAVERGSVREVLKTPQHPYTWGLLSSMPNLSSDVNEPLMPIPGSPPSLMNPPSGCAFHPRCGFTDLVPGGRCSGERPTLDLGRGAACHLTGDQRQQVFIEKIQPRLG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00852 ABC transporter ATP-binding protein MLLEVRDLHVEFHTRDGVAKAVNGVSYGVDAGETLAVLGESGSGKSVTAQTVMGILDVPPGRITAGEILFEGRDLLKLKEEERRKVRGAEMAMIFQDALSALNPVLTVGAQLAEMFTVHRGMSRKDAHAKAVELMDRVRIPAARERVRQYPHQFSGGMRQRIMIAMAMALEPKLIIADEPTTALDVTVQAQVMDLLAELQRELRMGLILITHDLGVVADVADKIAVMYAGRIVETAPVHDIYKAPAHPYTRGLLESIPRLDQKGQELYAIKGLPPNLTRIPPGCAFHPRCPMAQDVCRTDVPPLYDVTESDAERGSACHFWRECLHA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00857 ABC transporter ATP-binding protein MTEPSKSGAAVGEPTGDAPGSNAFLEVRDLKVHFPTDDGLVKSVDGLSFQLERGKTLGIVGESGSGKSVTSLGIMGLHTAGQYGRRKAQISGEIWLDGTELLSADPDHVRKLRGRQMAMIFQDPLSALHPYYTIGKQIVEAYRIHHDVDKKTARRRAVEMLDRVGIPQPDKRVDSYPHEFSGGMRQRAMIAMSLVNNPELLIADEPTTALDVTVQAQILDLIRDLQKEFGSAVIVITHDLGVVAELADDLLVMYGGRCVERGPAEKVFYEPRHPYTWGLLDSMPRLDRDQQERLIPVKGSPPSLINLPSGCAFNPRCPYADVPKDDVTRTVRPELTEIGSKHWAACHMSQEQRERIWTEEIAPKL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00862 ABC transporter ATP-binding protein MSAVRPPAAPAPDGGHILDLDDLGVVFTTETGTVRAVRGVSLHVAPGETLALVGESGSGKSTVALAAMGLLAGNARATGRAVVDGTDIVGADEEQLSGLRGKTVSMVFQEPATALDPLTRVGRQIAEVIRNHRRVSAADAAAHAVELLRRVGIPEPEQRARAYPFQLSGGQRQRVVIAMAIANEPALLIADEPTTALDVTVQAEILDLLRRLAAETGTGVLLVTHnMGVVADFADRVAVMYQGAVVETGPVEDVLLRPTHDYTKRLLSAVPRLSVSEAAGAGDTAEPAGAGSAGAGSAGAESVEEPAVELRDVSVVFGRGKQAVHALRGVSFAVRPGETLGLVGESGSGKSTASRVALGLVAPTAGSVTLFGADLARTRARARRALRAGVGVVLQDPVASLDPRMTVGECVAEPLRVHRRTLSGRERESLVGDVLDRVRLPREVARRAPRELSGGQRQRVSLARALVLGPRLLVADEPTSALDVSVQEAVLEVIGELQEELGFACLFVSHDLAVVQQFARRVVVMRAGRAEEQGLTSATLLNPETDYTRRLLAAVPVPDPVVQRGRRAERLATLAAGRTEEQG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00867 ABC transporter ATP-binding protein MSLVEVTGLSVAFGSVRAVEDLSFRLEKGAALGLVGESGSGKSTVASALLGLHRGTGAVVDGSVRVAGTDVGAASERELRGLRGGKAAMVFQDPLSSLDPYYAVGDQIAEVYRVHHPASRRAARARAVEVLDRVGIPDAARRSRSRPHEFSGGMRQRALIAMALACEPDLLVADEPTTALDVTVQAQILDLLHALREETGMGLLLVTHDVGVAAESVDEVLVMRHGRAVEHGPVGSVLGSPAEAYTRRLLKSVPRVDTPRPPAPPAGAVADDASRDGVVLEATGLRRVFGRGSKAFTAVDDVSLEVRRGEALGVVGESGSGKTTLGRMLVGLLEPSAGEVRLDGAAVTGVRPDVQMVFQDPVSSLNPRRSVGESVADPLRARGERGPAVRARVAELLERVGLDPAHYDRYPHEFSGGQRQRVGIARALAAGPRVLVCDEPVSALDVTTQAQVVELLDELRRELGLALVFIAHDLAVVRRVSDRLAVMRHGRVVEYGPADGIYESPGDPYTARLLAAVPVLDPGLAALRRAERREPAVT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00872 ABC transporter ATP-binding protein MLSVEGLHVAFPGRRGGADARAVDGVDLDIRRGEIVALVGESGCGKTTLARSLLGLVRPVRGRVTFDGAPLAHSARALKAYRRRAQLVLQDPSGSLNPRHTVYDIVAEGLRIHGRPGDERTAVAEALSRAGLRPPERFFLRYPHELSGGQRQRVVIAGALVLRPELLVADEPVASLDASVRGEILALLLRLRTELGLAALVVTHDLGLAWNIADRVAVMYLGRIVETGAVEQVLTAPRHPYTRALLSVLPEAPGDPVVLTGEPPDPSNIPTGCRFHARCQVLADGTAERAGVADACRSREPAVLHGGGESQVACHWALAAPREVSPAGPAPR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00877 ABC transporter family substrate-binding protein MSHVRVGPRAVTRSVAFLTAGVLAVPALAGCTSDEPAGKPLAAQDVAAAPRSRVADGGTLRWAVDSVPETLNAFQADADDTTNRVAQAVLPSMYRTDDTGRPARNPDYLESAEVVDTEPKQVVVYKLNQQAVWSDGREIGAADFAAQWRALSGKDSAYWTARNAGYDRIEKVERGAGDLEVKVTFSRPYADWQSLFTPLYPKDVTGTPDAFNDGARRELKVTAGPFAVQKVDTKDDEVVLAGNPRWWGEPAKLEQIVLRAVPRDKRVSELVAGKLDLAEVDPETADEVGLAAGPRDAGTGTPLMGPQGTPAAGAPGSPLAGDRGRSAAQALRSWALANGSDEEAAEEEVLAREERRETEAKAQRRQRALSGFEVRKSLEPAYTQLALNGADGPLADERVRRAVARALDRKKLAEAVLKPLGLPAEPVGSHVALAGQPAYADGSGALGDQNAKEARALLADAGWVPGGPVKKTEKGEKAAGAEGDGEKEKDGKKSEDGDDGDDGTYIVGEDGKNPGDGGDGENGEGGAKADAESGEKHSSGKNTAQGGAPGAYAPKGTAAPAAAAAPVAKDGKALTLRFVLPSGPGSEALRTVAGRVSDMLDEIGIDTAITKVPDESYFKDHIASGAYDLALYSWPATAFPATDARPVYAKPVPAADGSLNVAQNYTRVGTDQVDQLFDRAMSTLDRKEARDLLRKADSRIWAAAGSVPLYQRPQLTAARKGLANAGAFGFETPVYEDMGFLKKGAQGPRPAASPSS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00882 ABC transporter permease MLHYALRRCGWTLVQLAVLSLVVFLLTDLLPGDAATVDFNEQAGLDQVAQLREQMGLDRPLVERFADWAHGLLTGDLGTSLVGGGPVRDVLSSSVPVTAALAVVTLVLLVPLAVAVGLLTGLRAGSRTDRTVSAVTLTLTSVPDFVLALLLVGVFALRLGWLPSTWVGADDVWWQRPELFVLPVAVLLARTVCVLSRQIRAGTVTALHAGYTVQARRLGVPPARLVLRHVLPNAAVPGVQELARTGDQLLGGVLVVEAVFAVPGTATALVEAVQNRDVPTVQGLTLTLAAVACLLNLAADLVSHRLAPRTEVLR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00887 ABC transporter permease MLRYALRRSGWTLVQLAALSVIVFLLTDLLPGDAATVDFNEQAGLEQVAQLREQMGLDRPAVERFADWAHGLVTGDLGTSLVGGAPVSEVLTSSIPVTAALAAVTIMLLVPLAVGVGLLTGLRAGSRTDRVVSAVTLTLTSVPDFVLALLLVGVFALRLGWLPSTWVGADDGWWKRPELFVLPVAVLLARTVCVLSRQIRAGTVTALDAGYTVQARRLGVPPARLVLRHVLPNAAVPGVQELARTGDQLLGGVLVVEAVFAVPGTATALVEAVQNRDVPTVQALTLALAAVACLLNLAADLVSHRLAPRTEVLR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00892 ABC transporter permease MNLLAFAGRRLAGAAVLLVLLSAAVFAVTAVLPGDAVSAVAGVDASAAQRADVRAGLGLDRPAAERYAAWAADAVRGDLGHGFVGERPVTDILATRLPNSLLLAGLTLAVTAPLAALLGLWTGLRGGGTADRVVSTGAQVLAAIPEFVVAALLVAVLAVWAGVLPRVSVVPLGGTPLDAPRALVLPVLTLSAVGLAVATRLLRVSVADAAATPYCEAARLGGVRGIRLAVRHVLPNAAGPAVQALTLTTGALVGSAVVVENVFDYPGIGRELQLAVAARDVPMVQGIATALVAVMLLVLLLGDVCARLIGAREGHGR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00897 ABC transporter permease MDLGTSEAATLEQPPGPDGTNPHERPRSLWTDAWHDLRRNPVFIISALVILFLVVISLWPSLIASGSPLKCDLAKAQEGSQPGHPFGFNGQGCDVYTRTVYGARTSVAVGILATLGVALLGSVLGGLAGFFGGAGDAVLSRITDVFFAIPVVLGGLVLLSVITSNTVWPVIGFIVLLGWPQISRIARGSVITAKQNDYVQAARALGASNSRLLLRHIAPNAIAPVIVVATIALGTYISLEATLSFLGVGLKPPSVSWGIDISAAAPYVRNAPHALLWPSGALAVTVLAFIMLGDAVRDALDPKLR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00902 ABC transporter substrate-binding protein MSILRNRTATAAIVAVAAGALTLTACGGGDSDSSSKDNSKQKEDAKSQSKPVQIGDAQASTGPAPDVEGAKSGGVATVYQATDFSHLDPGQIYVSDGKLLSRLIFRGLTQYDEDENGNLTVVGDLATDAGKESDGGKTWTYTLKDNLKDENGNPINSADFRNTVERLYSNYITDGPTFLQQWLSGDGTTYRDAYQGPDKGKHLPDDVLETPDDKTIVFHFDTPRPDLPQMLTMPGYQLVPEETDTKEKYDSAPVSVGPYKISDFKPGKSMTLVKNTQWDPKSDSVRHQYLDGFNISMNHDDEDQTKTLLADQGEAKNAMMFTGQVATTQLQKVVGDKQAMENRTIQGYAPYVWQLNFnMDRIKDKKLRDAISLALPSDAVFKADGGAYGGEVANSLMSPTTPGYDEKFDPFNREKKPNGDVEAAKKLIKEGGFEGKSLVYAYGNTPERQKQAVLIATALEKIGLDIQKKEIDSATWYEQVGKVKNGYDLYMTGWGQDWPSASTVFPPVYDGTQIQDGASNYSHINDDHVNSEIKRIQKITDTDEATKAWAELNEYISKEVNPAAPIYYTKVFQIFGSNIGGIRYSSDSSYVDVTRVFLKK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00907 ABC transporter substrate-binding protein MPVTPTRRSVLAAAVATGAGLLTGCSSANSGSSSPKKGGTLSAAFPGAGVKETMDPHAQRQFVDIARHKAVFDKLVELDSTLRPVPRLARSWSSDDEARVWRFELREARFHDGHVLDADDVLYSLSRILDPDAADHLAKNSLSHVDLANCRKVGRRGVEIALTRPNAELPSQLAMTGTPVVRDGWDDPSKPVGTGPFRFASFTAGRGFTGRRFDDHWNGAPHLDEVRILSAESEARAAAVRSGEVHFAHEMTPTFARTVAHDGRVRVVATKRSGVQGFALKTDRAPFDDPDAALAVKLLVDRKRLVDVVCAGRAEIGNDLYGKGYTYYPDGLEQREQDVAEARRLLRRTGLYNKKVTFYTSTAADGFAQAAHLFTEQAGEAGLKVEVVNGPPESYFTDALSKGTVTNHRCGAMTIPTYIGERLLSDAPQNQTAWKHEDFDDDFTAARAEVDDEKRTARYRSVQTTLRDRGGLVLWGHPEWLNAVSRTAHGVKEAPPNTVDWARFDTVWLD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00912 ABC transporter substrate-binding protein MRYTGAIGVVTATATGLTACGGPASTGGGAGGAGGGGDTVGAGISYPLSTGFDPMITSGATPYAAnMHIFEGLVDLDPATLVARPALATGMPQKINATTYRAVLREGATFHDGSPVTANDVVFSFERVLDEGNASLMAQFVPFVDKVTAVDRSTVEFKLKYPFALFPSRISVVRIVPEKIAGADAKSFDSRPVGSGPYRFVSAVREDKIVMEAYDKYNGPHPAKAGKLVWRLISDPSARVSALKSGRVQAIEDVPYIDVAGFTGKDEVESVQSFGLLFLMFNCADPRFKDKRVRQALHYALDTEKIISTALLGNAEAATGYVPASHPDHHRAATVYGHDPARARKLLAEAGVGKLSFTLLLTDNGWVKDIAPLMKESWAAVGVDAALDIQQSPAQYAKIDQGDFDALAAPGDPSVFGNDADLLLRWFYYGFWPEKRYGWQGSKAYKQTRSLLDKAASEGDEARRKELWGRVTDLVADEAALYPVLHRKLPTAWREGTLTGFEPLPTTGLSFLDVGRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00917 ABC transporter substrate-binding protein MRGATHAKWAACAAAAALAATACGGGGGGGNGGGDSGAVLSSSWGDPQNPLEPANTNEVQGGKVLDMIFRGLKRYDPESGEAQnMLAEKIETSDSQNFTVTVKDGWTFSNGEKVTAQSFVDAWNYGASLKNNQRNAYFFAYIDGYEKAHPEDGGKQSADTLSGLKVTGPRTFTIKLSQKFSTFPDTLGYPAFAPLPKAFFDDHDAWLKKPVGNGPYQVDNYTRGSQMSLRKWEQYPGDDKAQNGGVDLKVYTDNNTAYTDLMAGNLDLVDDVPAAQLKNVKNDLGDRYINTPAGIIQTLAFPYYDDAWNKSGSEKVRKGLSMAINRKQITDTIFQQTRTPATDWTSPVLGEDGGYKAGLCGEACEYNAEEAKKLVKEGGGLPGGQVKITYNADTGSHKQWVDAVCNSINNALDNDKACVGNPVGTFADFRNQITDRKMSGPFRSGWQMDYPLIQNFLQPLYYTNASSNDGEYSSQKFDDLIDKANGETDTAAAIKSFQQAEEVLRDDMGAIPLWYQNGSAGYSDRLSNVKLNPFSVPVYNEIKVG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00922 ABC transporter substrate-binding protein MTTQRTSGRRKQAMAAAAVVAALLTTAACGGGDSDSGGSKNGAAGFDAANNKIAQADQVKKGGELKFASTQDADSWDTTRGYYGFMWNFSRYYARQLVTNTPAPGEKGAGVSPDLAADVAKVSDDGKTYTYTLRDGVTWEDGKPITSKDVKYGIERGWAQDVLAGGPTYLKEVLDPDGKYEGPYKDKSADKLGLKSIETPDDKTIVFKLPEANSDFEEMLALTSASPVRQDKDTKSKYGLHPFSSGPYKFESYNPGKDLTLVRNTEWKQDSDPVRKAYPDKISIKFFTNANELDQRLIAGDYDIDLAQTGLSPQGRTSALKEHEGNVDNPVSGYIRYAVFPQSVKPFDNIHCRKAVLYGADHVSLQTARGGPQAGGDIGTnMLPPAVPGSEAQKYDPYEMAGANKNGNIEKAKEELKACGQPNGFKTTIAVRNNKPVEVATAESLQASLKKVGIEVGIDQYDGSQTAGIIGSPSNVKKKGYGIIIMGWGPDFPSVQGYGKPLWNSEFIQESGNNNYALIDDKEIDGLFDKYGTELEDSAKADIAKQINHKVMEGAYYLPFVFEKFINWRSSRVGNVYTSDGYSGMYDFVNIGLKSSSK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00927 ABC transporter substrate-binding protein MPVTPTRRSVIAAAVATGAGLLLPGCSSAGSGSSSPKKGGTLSAAFPGAGVKETMDPHAQRQFVDIARHKAVFDKLVELDSTLRPVPRLARSWSSDDEARVWRFELREARFHDGHALSADDVLYSLSRILDPSAADHLAKNSLSHIDLANCRKVGKRGVEIALDRPNAELPSQLAMTGTPIVRDGWDDPTKPVGTGPFRFVSFTAGRSFTGRRFDDHWNGAPHLDELRILSAESEARAAAVRSGEVHFAHEMTPTFARTVAHDSRVRVVATKRSGVQGFALKTDRAPFDDPDAAMAVKLLVDRKRLVEVVCSGRAETGNDLYGKGYTYYPDGLEQRERDVAEARRLLKRTGLYNKKVTFYTSTAADGFAQAAHLFTEQAGEAGLKVEVVNGPPESYFTDALAKGTVTNHRCGAMTIPTYISERLLTDAPQNQSAWKHDDFDDAFTAARAVVDDDERTARYRSVQTTLRDQGGLVLWGHPEWLNAVSSSVQGVKEAPPNTVDWARFDTVWLA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00932 ABC transporter substrate-binding protein MITHDQHRRGRTAPRPWRARLLAALGACALLLASGTVAPSASAENGDGDGGGGGDKVLTVAVAQSVDSLSPFLAVRLVSTSIHRLTYEYLTNYDAEDNHVIPGLATEWKSSPDKLTWTYTIRSDSRWSDGERATAEDAAWTFNTMMTDPAAATANGSFVGNFAKITAPSPTQLVIRLKKPQATMTALDVPIVPKHVWEKVDDFSEYNNDKDFPVVGNGPFVLTDYKPDSYVRLKANKDFWRGAPKFDELVFRYYKDQDAAVAALRKGEVSFVAGSPSLTPAQADSLKGEENIRVNDAPGRRFYALATNPGARAKDGTKFGNGDPSLLDRRVRNALFKAVDRKAIVDKVFQGHAVEGAGYIPPRFSSYFFEPSAGQELAYDPQQAAELLDEAGYRTGADGKRLGKDGKPLDYRVLCHATDPNDKAVGKYLQEWWGELGISVTLDCLDNVTDPWLAGEYDLAFDGWSVNPDPDFVLSIHTCDALPATPKDTGATDNFICDKEYDELYARQLAEYDAGKRAGIVKQLESRLYDTGYMNVMAYPNAVEAYRTDQIESITTMPAAAGNIYGQDGYWSWWSAVPADSGDSSGGSSSTGTVIGIAAGVVVLAGLVVLFAVRRRATADDRE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00937 ABC transporter substrate-binding protein MRSLRRPRLLAPFLLTPLIAGCFASGGGDSGDGGGKGGDGDRLRVALAFPPAENLSPYGADATLLSRLGVTEGLTALDANGSAAPALAESWRRDGEKTWEFTLRDATFQDGSDVTPDAVADSLGQAVRAKPAPAALAGVGLTAEAGGERVVRVTTAEPDPVLPLRLSSPSLAILSAKAYEEKGGKADPVGTATGPFRLTKVNGATSASLDRFDDYWGGRAQAAGIDARFVADGTARANALRTGELDIAEAVPVAQAASLDEGTRRDTATTRTTSLLFNASSGTFKDAGLRAAARGAVDTSVFAKDVYEGYGDPGAGIYGPAVTWAEGKRSAPVGRAGAGKPGGDDVIDLATYDNRPELPEAAQVVKQQLEKAGFTVKLTVREYSRLEADALDGKFDAFVLARNTLLDTGDPVAVLASDYTCDGGFNIAQLCDKDVDRAVADAERIADTAKRQDAAMAAEARILGSDAVVPLVHQRIITGVADSVQGVILDPYERTLVGTGTRR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00942 ABC transporter substrate-binding protein MRHPSRRTRRAAAALTVSLIVTAGAAACGPEDNDAKSGGADGDPQKGGTLTVLNAVPQTDFDPARLYTSGGGNVPSLVFRTLTTRNREDGAKGTEVVPDLATDTGRPNKDATVWTYTLKEGLKYEDGTKITSADVKYGIERSFAAELSGGAPYLRDWLIGGADYQGPYKDKGKGLDSIETPDERTIVFRLNKPEGEFPFLATQTQFAPVPKSADKGTKYEEHPVSSGPYKVVRNENDGERLVLERNEHWSEKTDAERKAYPDRIDVRSGLDSSVINQRLSASQGADAAAVTTDTNLGPAELAKVSGDKELAARVGTGHFGYTNYIAFNPKVKPFDDPKVRQAIAYAVDRTSVINAAGGSSLAEPATTYLPNQKSFGYTAHDHFPAGESGDPAKAKELLKEAGHADGLTVTLTHSNAKDFETSPEIATALQDALQKAGITVELEGLEDNDYRDTIHDAKSEPGFFLAHWGADWPSGGPFLAPIFDGRQIVRDGANFNTGFLDDKSVNDEIDAINKLTDLDEAAQRWGALDKKIGEKALTVPLFHPVYKRLYGKDVKNVVISDWTGVLDVSQVAVK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00947 ABC transporter substrate-binding protein MSRQFDRRAFLRRGAAGAAALAVGPGLLAACSTDAPGADREGAGSSPRSGGTLRAAFVGGGASETLDFFNGPSALDLVRARAWHGTLGNLDPEGPDGVRYGVLKGIDVSDDLSAYTLHVRPGVRFTDGSELTSADILHSLSVLAGRSTLPVYRLAAANFDLASAKADGDLKVVLPTLRPIADGRMILCQGNFLVVKDGTRAFRKGMPSCGPFRLTEFTAGQGSAFERYDDHYGHVPLLDGLELRSIADSTARAGALTGGEVDFAHDLSPVTARTLTDDAKVRLVPTGSPYLVGLSFQMnMAVEPFDDPRVREAFKLAVDRETMVKTVFYGNAETGNDLPAMGFPDYAGSLPRRTHDPERARKLLKEAGADGTEVRLTTGPETPGMVEMATLFVEDLKKVGVKASVRELPAGQLYADFAAYAALPLAGSYQMPIPALSTYQMSTAGGSPSAFGWKDAETDALVAKARAASDPAEAKELGTLAQRTRWEKGNQVLPVFKPNLNAQAEGVAGIREDLFEQFPGFSQASLA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00958 Acid phosphatase MPDRSKRPPARAAAGTRALRAAVAAVLAGALGLGALTTGGTAAAAPSAPASASGEASGGTDYTKLVDPFVSTAGDDGNDLPGAQAPHSLAKVNPMTVPDRNHSGYDYNEDHIAGFTATNLDGVGGSGGGGDLLVVPTSEQYDKRPATSTYAHPYSHDDESASPGSYRVGLGSDAGTIDAEMTATTRTALERYAFPDGARPQLVLDLANNFTSRTRSTLDATRLKDGTTAISGLVAGSFNGASYRLYYYATTNVPVTSLRSWGDDGALGGATARDGTDTGAVLGFDPADGDDVELRITLSPISAEQAATDQHNEVAGRGFEEVRAQTEAEWNSTLGTVAVEASRKADPDSTLTKQFYTHLYRMYALPVNATSTSGTYRGVDGAVHKANGFTYYDGWSTWDDFRKYSVTAYIDPAGYRDMVQSAVILFADARSTGKSLGSLTHSVPTVRWERLPVVIADALSKGYKDFDRLDEAYPALKSYAGYYTGTELRQGYVAGDPGTTVQRGYDQWALSLVADALGEDADAKKLREQATMATDNLVKPGAWTADDGTEVGLLTPRDGEGAWQGVDYEKFEEAKLYQGTLWQYHWYDAYDMGGLIEAMGGEKAGRAAIRHMFGEDSDADDGSAMLHSNANEIDLQAPYLFNYVGEPSLTQKWVRAIYTGETWNRYIATGSTGEAPSSGGEFRPPVKTKAYELAPDGFLPTMDNDAGTMSTMFVAAALGLFPVTAGSSQFQIGSPFFDSTTVHYAGGAEFTVEADGVSPDNYYVQGARLNGKRFSNTWLDYSQIVAGGTLKFDMGSAPSSWGARTEPAYSLNTDTGDGDDGSAPGRGTTVVSARPDSVDTAADGTVKGNIELRLSGKASFAAREGTSLTRSGAAGVTGLPDGVEADLRVTGRRTASLRLTGATQTDARLGLTFRDRAFAHGVPASTVTGAGVSVTDPLVVSAAVVHRGSLGALVEEASLVREGNYSDGSYGVFRTALERARTVLADADAATGTLMAAHDALKSAIDALTLDEGGYAVLQAEDPDSMEGPSLVKEAYHSDGDLGGVTEGAWEQYTNLDFGGVAPRGVSVRYANAQAPEAEPSSVDIHAGDAEGPVVATVSLPGTGGWQYYTTVRAAVTDPQALLEASTATFVFHAPSGQQWVSNFDWYQFSPAEPASSSPVTTLATLTTANATATGDGSLPLKLTNGVFENVTNGAWAEWRGTGLGDGADTVTVSYDKPRSRAASDSHIELRLGGRDGPAAVDVPLEYTGSGWGTVATTSVRLDPETFGGAQDVYAAFVSGTQTDAQPYVANVYSLTLTRETDAPVVFDATAFGASSGGGLKSEPATWDGAGSATSLGGTYDGAWLDYGDIDFGTEPKNTVTFTYVNNSARCGTGSAVEIHLDSFDADAPGTPDATVPLPVTGSSWSSGGTTSLTLPEAITGTHSVHLRLTTNADSSHPYVANLGRVAFDHVEAPAETDLSALRKAVEQYGGLAEHKDRYGTIDFGVFVRELAAARALLDAGDATQLEADLQTRGLTLAANQLVPLPRLKLENLVATASARADERYTDASWKAFTTALTAAKETVADDAASDATLTARYTSLDRAMSALRTKHRTVPAAPGAVSATASGTSVQVTWSAPEDDGGSPVTGYEVTLGGGRQVEIADPASRSTVFTRLADGTSHTARVRAVNALGDSAPSAPTRPVVTGDNRPQTPTVTGVVTDGKRVRVTWRPAGDGGFPVLGYTVALDDGTTAHVSGTTDSALLTTAGGAKAHTATVTARTLAGTSADPAPKAAATAGTGTATSTGTATGTGTAAASDPADYEPAPFPDDVLDAAYPSDEWPRTGDGGDYFTNLLSGFDDLGPGTLGANGELPEGSELGAENDEITVAVNNAATQKQVDRAEVDASNSATVTMADGLGSRLGPIYGEALKEGQLPKTSALFSRVAENLDTHDAAKNRWNYLRPYVRLGFAGDGGRIYESEDSSYDGLAKQGSYPSGHTYGGYEAGTILATLLPDLAPSILARTSEYGDNRLVLGFHYPLDVMGGRITAQATVAHRWADPAFGKLLQQAHTEIENVLLARCEEEGYGDTLTACAGDPYAGLGTAETVDLYTRRLSYGFSQVGEAGQALQAPSDAAALLITAFPDLTEEQRTQVVEQTATDSGLPLDLTGTGGPSWQRINLAAAMAADVTVGADGSVTVTNFPDATRAAVADASALTVEGVPLDGFDPGVGTYVVDWPEHGRIPAVGAVAAKSGARVKVTDGSRTVSSSRPGFTARTVTVTSADGEHSRTYTVGFQRTDHDHRPPWSGGPGGPGGHGDPWDRGGHDGPDGTGLWSPAREWEDARGR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00965 Acyl-CoA synthetase MTPGHGSTVDGVLRRSARRTPARVAVEYRDRTWTYGELDTAVSRAASVLLDEGLSPGDRVASYVHNSDAYLIAFLACARAGLVHVPVNQNLTGDDLAYILRQSGSGLVLTDPALAARLPGASRTLSLRDTDDSLLARLAAAPAYDGPEPAAEDLVQLLYTSGTTALPKGAMMTHRALVHEYLSAITALDLGAGDRPVHALPMYHSAQTHVFLLPYLAVGATNIVLDAPDGDRLLDLVEAGRVDCLFAPPTVWIGLANRADFATRDLTGLRKAYYGASIMPVPVLERLRARLPDLALYHCFGQSEIGPLAAVLGPDEHEGRMGSCGRPVLFVDARVVDEDGKDVPDGTPGEVVYRSPQLCDGYWDAPEETRAAFRDGWFHSGDLAVRDADGYFTIVDRVKDVINSGGVLVASRQVEDALYTHDAVAEAAVIGLPDERWIEAVTAVVVPRAEVTEDELIAHARAELAAFKAPKRVRFVDALPRNASGKILKRELRDRFTAS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp00970 Acyl-coenzyme A thioesterase THEM4 MSGTSPGLQPPADAVKPVRHPEAPAPGELLGAHYGQCFGCGGDQPHGLHLQARAGEGVSITAEFTVRPAHQGAPGLAHGGVLASALDETLGSLNWLLRTIAVTGRLETDFRRPVPVDTTLYLEAEVTAVAGRKIYSTVTGRIGGPDGPVAVRADALFVEVKVDHFVENGRDEEIRAAMDDPDQVRRARAFEVNP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00975 Acyltransferase papA3 MRMTDIQRCEIRPGRLVEWTLSPRTLDIAAGLPEDARPPAYIQESHIRTARSVREGGLFVPTWLGAAFDIPGAVDLDVLQEALRSWTLRHETLRSGFRWSGESGDTMRRFTLEPDAVSLHREDVGDFPDAADLAGHLQDRFDRVADALRWPNLIYTAVVRDDGVSVYMAFDHSNVDAYSIYRIPAEVGELYAAGIAGRTVPQPRVGSYVDFCEAERADADRIDADHDIVARWREFIRRCDGRLPSFPVDLGLRPGGALPEQRLLREPLVDAADAAAFEAYCRPYGGSLVGVLAATALIVHEIGGESVYRTVVPFHTRSRSQWSESVGWYVGGAPIEVPVDRAHDFPAALRTVRAELQANRRMSRMPIDRVLRLLGTDFRPGSPDLYSIVSYVDARDVPGAGDWAEQTAYAMLRVSYGDQVCAWVTRLPEGLWFASRYPDTDIAHKNLRLYVERLRDVITGIGQKPTD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00985 Adenosyl-hopene transferase HpnH MAMPLRQSIKVATYLAEQKIRRRDKFPLIVELEPLFACNLACEGCGKIQHPAGVLKQRMPVAQAVGAVLESGAPMVSIAGGEPLMHPQIDEIVRQLVAKRKYVFLCTNAMLMRKKMDKFKPSPYFAFAVHIDGLRERHDESVAKEGVFDEAVEAIKEAKRRGFRVTTNSTFFNTDTPQTIVEVLNFLNDDLKVDEMMISPAYAYEKAPDQEHFLGVEQTRELFKKAFSGGNRARWRLNHSPLFLDFLEGKVDFPCTAWAIPNYSLFGWQRPCYLMSDGYVPTYRELIEKTDWDKYGRGKDPRCDNCMAHCGYEPTAVLATMGSLKESLRAMRETVSSNRE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp00994 Allantoate amidohydrolase MSFHSMWAELLPVGRSSASGGYRRYAWTGADSDCRTWFREQAQARGLAYETDRNGNQWAWLGDPAAGNAVVTGSHLDSVPDGGAFDGPLGVVSAFAALDELRGRGARFTRPLGIVNFGDEEGARFGLACVGSRLTSGALTAEQAHRLTDADGITLPQAMEAAGHDPDTLGPDPERLARIGAFVELHVEQGRALDLSGDRVGIASAIWPHGRWRFDFRGEANHAGTTRLTDRHDPMLPYAEAVLAARREAQLAGAVATFGKVAVEPNGVNAVPSLVRGWLDSRAADQEDLDAVVAGVEKAAREYAAAHGVDLGVECESFTPVVDFDHALRDELARILGKEADLRVPVLGTGAGHDAGILSGRVPTAMLFVRNPTGVSHSPAEHAAEDDCAAGVHALADVLEGLART Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01011 Amidohydrolase MSESTTPPPTVLLRRGEVHSPADPFATAMVVERGQVAWVGSEGAADAFADGVDEVVDLDGALVTPAFTDAHVHTTATGLALTGLDLSGASDREAALALVRDFAAARPGDRVLLGHGWDAARWPEGLPPTRAELDDATGGRPLYLSRIDVHSAVVSTALLDLVPDGAARADGPLTGDAHHAVRAAALGAVTPAQREEAQRAALAHAASLGIGTVHECAGPEISAEDDLTGLLRLSAGEPGPRVVGYWAERDVDKARELGAVGAAGDLFVDGSLGSHTACLHQPYADAGHTGTAHLDAADVAAHVVACTEAGLQAGFHAIGDAAVAAVVEGVRTAADKVGLARVRAARHRVEHAEMLTPETVAAFAELGLTASVQPGFDALWGGEDGMYAQRLGVERARTLNPYAALLRAGVPLAFGSDSPVTPLDPWGTVRAAAFHRTPEHRVSVRAAFTAHTRGGWRAIGRDDAGVLVPGAPADYAVWRTGELVVQAPDDRVARWSTDPRSGTPGLPDLTPGRELPVCLRTVVGGRTVHVRPGE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01016 Amidohydrolase MTDRAVLHVKGRVLVGPEEVRDEVWVIDGRISYDRPAGAADVRTVEGWALPGLVDAHCHVGLDRHGAVPADTAEKQALSDREAGTLLLRDAGSPSDTRWIDDRDDLPKIIRAGRHIARTRRYIRNYAWEVEPDDLVAYVAQEARRGDGWVKLVGDWIDRDLGDLSACWPRGAVEAAITEAHRLGARVTAHCFAEDSLRDLVEAGIDCVEHATGLTDDTIPLFAERGVAIVPTLVNIATFPALADGGESRFPRWSAHMRRLHERRYDTVRNAYDAGIPVFVGTDAGGALAHGLAGAEVAELVTAGIPPVEALSATTWAARRWLGRPGLEEGAPADLVVFDRDPRADVRVLTDPRRVVLNGRVVG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01021 Amidohydrolase MTPTPHEKPKPGAARGEPADLVVTGCTVLVHDERERIGFEQDAAVVVREGAVDSVTTAAAGAAVPAAERIDARGQVALPGLINCHTHAPMAALRGLAEDLPTEEWFNDVVWPVESNLTARDVVLGTRLACAEMIRAGVTTFADSYFHMDAVAAVVDRCGMRAQLGQAYFSSQGPAGLEASVEFALRLRDGSGGRITTALAPHAPYTVTDADLAETARLARAHGLPVHLHAAENLDQTHTSLARHGATPIGVLERTGILDTDVLIAHGTGITDADLPLLARAGGRTAVATAPRGYLKFAWPTTTPVRALRDIGIPVGLATDGAASNNSLDVWESMALTSLIQKSTEGDPRWLTSRQALHHATVQSAHAVGLGDAVGRIAPGRRADLILVDLTGPHTQPVHDLAATLVHSARSADVRTTIVDGRVLMRDRELLTVDVPGTVRELGERLPALTDRGHGRRIQEYDT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01026 Amidohydrolase MLTIHAAERVRRTWDSASLEGGAVAVEGGRVAAVGPLAELAERFPGARVRRWPGVLGPARVHEGPLPDAPTPREQVHAVLKLGAVAVLAEYAGSRELRAAAERNDVAVLERARPAALVDLGRADLAVLDDGGACIATVCAGRLVHRRR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01031 Amidohydrolase MHLDALYTNGRFTTLDASRPTAHTVGVFAGRVVGLDDEVAGCTADRVHDLRGAPAVPGFNDAHQHLSMRGRRLLQLDLHTGTVPTLDALYAAVRERAARLGPDEWLFGAGYDQNKIGAHPTAAALDEAAQGRPVWLEHVSCHMGVANTAAFARAGFTDRTGVPDVAGGHVERDTGGRAAGLLQETAQHLVTRAFRPTPVDSIVAAIAAGNDKGVTEGITSVTEPGIAAADHVGHGPADLHAFHRAVEEGVLSIRTTVMPYMTVLHDAGPAGGGDTWFGLDTGLRSGFGDDRLKIGATKIATDGSLIGRSAHMCCGYHDEPDNSGFLLFDEDRLHHMINEAHRCGWQVAAHAIGDAAIDVVLDAFEAAQAAHPRPDARHRIEHFAVASDEQVRRLVAGGVVPVPQGRFVSEIGDGMITALGPERATRCYRMRSLLDAGAVLPGSSDAPVAHGSPLLGIHDMVNRRTAGGAPLAPAEAVTAEQALYAYTVGSAYAEHAEDRKGRLAPGMLADFAVLSDDLLAVDPGRIGALSVGATVIGGRVVHDAGALD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01036 Amidohydrolase MNAAGNSSGLGTGRPGTPVVFRNGTVLTMDDRRTLHRGADVLVVGERIEAVGPLPAVPEGTREIDATGGIVMPGMIDTHRHMWQTAMRGYGADWTLTQYFVWYYLEHGTHFRPEDVYAGNLLAAVEALDSGVTTTVDWSHGLQTVEHADAALDALDEVPGRFVLAYGNIRAAPWEWTAAPEFRAFVDRRFGGDRTGLQLAFDVTGDPDFPEKAAFEAARELGVPVTTHAGVWGATNDDGIRLMHEHGFMGPDTVYVHAATLGADSYHRIAATGGSVSVSTESEQSCGQGYPPTWALRAHGIPVSLSTDTSVWWSGDLFSAMRATLGADRAREHLEAHAGGETVTHSHLRAEQVVDWATRGGAKALGLDDRVGSLEAGKRADVVLVKNDHSPVMFPLLNPYGHVALQAQRGDVHTVMAGGRLVKHEHRLIGVDLAKVRRTVDSTVEHLRSRLGAEAWEQGMNPDVPETKMLDNPYTYTGYRTAATHGG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01041 Amidohydrolase family protein MSRCRCVAMSPCRRDVAVSLCRDPGWVRACRGMAWTCRKPGPWGGRDAVVRRMPSVGSLLTGHRADSGGnMSRFAVANTRVFTGTHVADASVVVVEDGTIAEVGHEAPEGVEKIDGVGGTLLPGLIDAHTHTDEDGLRTALSFGVTTELDMMSVPDAMEPLRKKARAEFDVADVRTASWGLAHPDGHPHQLRRGLGDPVWPTATVPGEAAAFVDGRLSEGADYIKIMVEDGDVFGTSLPLVPYDVVVAVVEAAHERGVMALVHALGAAATRVAVEAGADGVTHLHHDEVISDDLVVRMREQGMFVISTLAVTASGASDGAGPRLGADLRVASRLDAEWRDNLGREFGWNAHLPTALRSAGLLHAAGVEILAGTDAAHLGAPGIAHGASLHDELRLLEAAGLSPVEALTAATRRTADRFGLTDRGRIEPGASADLVLVDGDPTSRLSSTLNTRAVWRRGHRLALGGATAERAA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01046 Amino acid adenylation domain-containing protein MNHTARGMMRTPALSTGLARAVHERAGLTPHAPAVSDGGRTLDYAALDAEAAGAAAALRALRVGPGDAVAVALPRSWQLVCVMLGVLRLGARVVPVDLQSPAERRDHVLADSGAVVHVHTGDAPHGLPPGVAAVPVDGLLRDGRDAVDRPSPPDTAPPVSFVFYTSGTTGRPKGVEVRDAGILRLARPGYLRLEETERFACLANPAFDALSFEVWVPLLTGGCCVVLADDDVQSPERLAEVLLRERVDTAFVTAALFNAVVATVPDCFAGLGQLLIGGEQLNARAVRSWYRHNAGSGTRLYNGYGPTECSTFALCHPIPRDLDTPVVPIGRTLPETGATLVVPGTTREAAPGEVAELLLSGAGLAAGYRNLPEESARRFVPLSRPDGPPVVHYRTGDLVRRDARGDIEYIGRADRQVKVRGFRIEPGELEQRILAHPAVRQAHVCTRRAGGDGPNELLAYLVVDSALTWAEFDRHLAAHLPAYMRPHHLYRIDAVPRTANGKADQAALLARTDPPWRPDGDAAEVTDPVQRELLEMAGRVLGLPDLRPGDTWIACGGDSLTALRLRFEIRRRWNRDLPQSLVLRGDLAALAEAVRAAPDTDAPGYPSASAAGAGSAPATSEQQRLWLIQQQSPHSRAYDVRLAFAVEGDVDVPALRRASSRLVARHPALRTAFEAAPEGLLQVVGEPYDPWVPAERPYASPGVVAGGVPDPGAPQGAFFAEPFDLSRPRMLRMGLLPAESGSGSVLLLHLHHIAVDGWSVNVLLRDLSDGYAAALAGGEDAPDRAAPAPTPLDFAVWQEQWRAEPAYDALRTGLLAHYADRTEPGRAVPQPAPHLADRPGAALLHTQLDVVRRAALDRLCGAAGLTRFQVLLAVYAWALYGVTGDARPRVAAPVAGRPVREFEDSVGMFANTVLLPLDVSPRRELRQELLRLGRDTQEVLERQDVALADVVQGQGPLRRAGSPFDFLFVLENTDFDSLELPGCETSPRWPVPAGAKCPVTLSVIERPDGLACQWEYAPEHFTPERAAALAELFRRGVDALAEEHSATGTVADLVAGHRGSLPEPGRGESRAWAWTTVAEGFALQVARTPSDPALMTAEGPVDYRTLDAWAAALAADLRATAGARDAEGPCHVALFLEPSVEHVVALLALARLNLTAVPVDPSYPPALLRQILEQTDPLCVLLPPGDQSAFDAVDPRGRLGLPRRTVTLSAAPDPALPDPPHRGERPLYTLFTSGSTGTPKGVRVYDRTLCNLLQWQAASGGLGGAAATQQFSMLSFDVSFQEIFGTLCSGGCLHLVRPGLRQDVPALLDRLEAAGIERLFLPFVALQMLAEHAVHLGRYPSRLREVVTAGEQLVCTDAVRRWFAGMPGSRLFNQYGPTETHVVSSLCLDGDPSRWPERPAIGGPVANAVLHVVDEAGLPVPPGCPGDLLLGGVIDAPCYLGDGRLNEERFTELPGQGLFYRSGDRARFDSDGLLHFLGRADDQVKLSGHRLEPGQVEAALLRHPAVVGAVVAVDGGELVACLRCGDAAPSPAELREHLAGLLPAHVRVARYRLLAELPRTPSGKLDREAALRAPSRELPGAHRAADGPSSGREAALAAAFEEATGSAIGPDQTYFEAGASSLDLMRFHLRCTTVLGLPLTVADLFEHVTVRRLARFLDTDAGAGTGGGAGAGMSTGTATSTSVGAGTGDHAGAAAGAGAGDLTGAAAGAEGIAVVGMAVRAPGAPDLAAFWELIASGAGGIEYFDAPEGIVGARSQMDGLLAFDPERFGISRQEARLMDPQQRHLLMACVEALAHAGLADTGAARVGLVAGAGENTYFQAMLREADPAHLPDGFQLALHHDKDFLATKAAYHLGLTGPVLAAQTACSSSLVAVHLAAGMLRQGDADVMLAGGVLVDTSLSQGYRYRPQHILSADGHCRPFSDDADGTVGGSGTGVLVLKPLSRARADGDTVYAVITGSAVNNDGSAKLGYSAPSLAGQRAAVRTALRRSGRPGSDVAYVEAHGTGTRLGDPVEAEALRQALGTTEPDHCALTSVKSQIGHLGAAAGAVGLIRAVLSVHHGVIPPTRGFRALNPEIGPDPTPFYVPTEALPWPARRDRVAAVSSFGIGGTNAHVVLEGGSAAGPPDAADSGAADQEVVPLVVLSAAGAVRLRSDASRIADYLERRPEAYGQVLRHLQAGRPQERLRAAAVCPTPLSAVDWLRAAAASSAEPGAGERPAAPPRDPVAAAECRSVSELADAWLAGRTVAWPEGSAQAPWDFPPPSFDLADFHFGRASAAHSAPAPSGAPAAAPSGALAAARTPERLPEAQWLHQPQWVRLRRAATVPRGDRARTLVVVAEGPADAALVDAFAAGHRRVVWVRASADRARTGADRFEADPADPAHLRYVLDAVTEDGPPGVDWVHMLPLSVDGPVHATSVDRAAWACLDTPAALLRAVSGRPYAALLRPWWVSRGARPVHGDVSRPETALLAGVTEVGPQEGAPRGHWVDLPGTGPWAAQLAALFAEPETAGLPRQLALRQGCWWEQVLLPVAAAPDHEGEPLPASEGDHLILGGTGGLGTGIAAWLLAHTPGRVLLLSRRPRLPEVLAPWAERVELVDADLAVEPTAEVAVRIASRTTGLASVVHAAGVAAGGLVARRDAEDMRKALAPKLRGALLVEQLIEEHRPALAVYCSSMSAHLGGVGQFDYAAANALLDAFARYGGPGGGTTARSALAWDVWRETGMAVRTLHSDARHRAHLGVGLTVDEGQRVFARAVGLGLPHLLVSTTDVEESRVFYEGAGHDASDVPAARLPGAPAGDRAPAPDSARELLAEQLCILLGVDRLDPDASLYDLGADSLTLLSVIEAVDRSFGVELDLGSLSHRVSLDEIVARLDEARGEADRTQDSQDHLNPEEGKDEDGDEVTLTVWQQGAGRDVVCLVHPVGGDVQAYRFLAAALDPGATVALIADPGLRGRELPRWTIAERAHHYLAALRARFPETTWRWHLAGWSFGAWVAAGMAAEAESAGRPARSLHLLDPPPPGSGSVFQEYDERQLKTVFAAELGLGGEETGPGRQADTYADRLTRCCLANVHSMAAHRLPRITVTATRLWLARDPVEGLPSLGTPGEQRARWRAHLPEPTAAEVLDTTHYGVVRPPHAAAVAHAVNEAVHEAVAEGSTGGSAAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01051 Amino acid adenylation domain-containing protein MRRSSLAPARGPATVFAGKRTRGPVPAGRRSPSRTNCVDVRATSGGEPAEPRFSRRCDCNSGPPSQWPGPFTPRRTAPAGRAITSTTRRTCGSRSRGRPTRAAAPAPSPPLGRTGTPSARHSGRPDSAACRAAGRSARRNRVLTASVPRRGGELASVVAFANRRAGNTRRSPLTWSSAPPNDWLRLPHPRAGVAEYARSHPWQPFQHGRRPHLTATHTPHASSPGSQDDGFPPPLSFGQERLWTLAQTAGAVAAYNEPMAFRIRGPLDRALLGRALDVVVSRHETLRTRFVDVDGEVRQVVGPPESGLPLRVEDLSGAPDAEARLADHQREECETPFDLRRGPLVRGRLITLAPSDHALLLTLHHAVSDGRSGQVLTRELGVLYGALLRGEEQPLPPLPEQFAAHCRRQRAWVNGPEAAGQAGFWREYLDGAPPLLALPTDRPRPPRQSHEGDRVHVRFDADLTAALRAAARKEKCTLFAAVLAGWHILLSRLSGQPDGVVGIPVEGRRGSAASGLIGFYVNSLAHRVDLSGNPTGAEALRDVRASLRSVLRHQDLPFAHVVEAVNPRRSLSHGPLFQTMLTWGASRKDFLELAGTRVEPLAIDFAPAKFDYTLYLHEEDGGLVGYLDYARALFDRGTVERHLRYLTRVLRQLADDPGRRVADLVLLDDREHGELLAKGHGPVAPSPAADLVELFEEQVRGRPHGPAVVAGGTRLDYAALDRRANRLAHSLLARGVRPQQVVGLHCGRTAELLVGIWGILKAGAAYLPLDPGQPAARLRTIVEEATPALVLSDLGDPPGPWLPLGQVAAEGERDDPPGVAIGPSHLAYVIYTSGSTGRPKGVAVTHGNVVNLIGNWLDQYGAIPGEPSSAWASIGFDASVHELFLPLTTGAVLHVVPEDLRGDPEALLDWMREREIVHAYLPASYITWIDEDPGGRLRGLALRQVTTGAEPLPEMALHRMREVLPGLRVCYVYGPTETTVYSITYNQPQALGRRCPIGRPVRNTLVHLLDQGRRPVPPGVTGEVYIGGAGVARGYLNRPDLTDERFLPDPFVPGGRVYRTGDLARLLPDGDYEFVGRVDDQVKLRGFRIEPGEVAAALREVPGVTEAAVLADRDEAGETRLVAGVARAGGGSPLLPHEWRAALSERLPDYMVPSLFAEFERLPLNRSGKLDRQALLAHARSALSAAQVNTHAPRDRVEMSLYRIWRQVLVHPGMGITDDFFAVGGTSLSAIKVAHLVREEFGHDLPIREVLEHPTIERLAARVREGVPAKGDDSLIEFRAGGGAGRVVCVHPAGGTAFCYLPLATALPEGIGVQGVQALGLNPGEEPLASVESMAEHYLRLVRPEPGEALVLCGLSYGGLVAHEMGRRLAEAGHDRSAVVLLDTHGTDDPAERAAFAPVGADDFRARLVRFNGMYPGIDDAQIDRYFRIYNHNRAAARDHTPRSTAAPLLLVQADAEAPSPAEAAAVEERQRRFWGERALAGLVVERVEGGHWDVLEGERVSRIAALITDELARLDGRSV Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01056 Amino acid adenylation domain-containing protein MTDSPSAAHRDKVAIIGIGCRLPGHAGDHRSFWRNLIEGRDCLVPTPADRYDTTTLGSRDRAKPGRLTGGRGGYIDGFDEFDPHFFGISPREAEHMDPQQRKLLEVSWEALEDGGQRPAELAGRDVGVFIGAFTLDYKILQFADLGFETLAAHTATGTMMTMVSNRISHCLDFRGPSVSIDTACSSSLVAVHLACQSLQRGESELALAGGTLLHLAPQYTIAETKGGFLSPDGRSRAFDASADGYVRAEGVGVVVLKRLSDALRDGDPVHAVVIGSGVNQDGRTNGITVPSADAQATLIERVCAEAGVTPGSLQYVEAHGTSTPVGDPIEARALGRVLAQGRAPGARCYVGSVKTNIGHTEAAAGVAGLIKTALALRHRRIPPHLNLEQPNPAIDFAALPFEIPTAPVDWPEHQGPARAGVNSFGFGGTNAHVLLEEAPPRPPEEPRATARTPSLSVLPLSARHASGPAELAAGVRRELAAGVSLADLGHTLAHRRQHFEERLAVVHSPLGPPGSLDEVLAACERGEQHPRAVRGRLREPGAPRLVWVFTGMGPQWWGMGRELLDAEPVFREAVERCDREVRRQAGWSLLDELTRPEAESRMAETWLAQPANFAVQAGLAALWEHHGVRPDAVVGHSTGEIAAFHQAGVYGLEDAVRIALARSALQHRLAGTGVMLAANLSEEEAERLVRPYRDHVSVAAVNSPASVTLSGDRDTLRELAGRLEREQVFARFLDVEVPYHSVRMDPIEAELREALTGIAPRAAGLPLYPTAREGRARGPELDAVYWWENVRRPVRFRAAVDRLVDDGYTLFLEIGPHPVLGHSIRECLEGRAVEGVTLPSIRRREDEPERFARSLAELYTLGVDVDWSVLQPVGRPVPLPGYPWQRERYWVEPAPVEQIRLGRLDHPLLGRRASALQPTWESRLDTERLPYLADHRIEDSTVFPAAGYLEMAAQAVRALTGGDTATLADVEFSRALFLPDGEATTVQLAFAPEEAGFTIASLAGSGTGTPDRTVHASGVVRTGQPRRLAQPLDTGAVRARAGRRLDREACYGELAALGYHYGPAFRAIDEVWTGPGEALSLIRPTPGMGDGAADCHVHPVLLDACFQTMLTAMTPDDGRSAGIRLPAGIAELRLDAVGDRAALWAHATVTAESDEELVGDLALYAEDGTPLGRIGGFRAAAVDRGASSVKLGTIDGWLAEVVWEEAPTEAETPTEAPEDVGTAEGSGAGPGGSPAPGLVVFADEGGLGARMAEAVVARGGRCRLVRPGSRYRSGARHVTVRPDSAADLRRLFAELGPGFGAVVHLWNLDLPPLDTVGAADLDGIGTLGGYSLVLLAQVLPEAFPQGRLHIVTRGAQAVVPGEPVEPFGAPAWGIGRVLWQQELTGHSGKLIDLDPAGGPGEPEVLLRALTTDDGEGEIALRSGRRHLSRLRPPAGLTRPLPLRLRADGAYLVTGAFGALGRLLCRTLVRRGARRLVLLGRTGVPARGAWRGLDPGGPEGRRVAFLRELEALGAEVLVAAVDVTDAAAMEGWLAGRRAAGLPPVRGVFHLAGQVRDVLLPSLDREAFDAGYGPKAHGGYLLHRLLRDEPVEHFVLFASVASLLTTAGQVNYAAGNAFLDALAHHRRALGLPALSLDWGPWATGMIEELGLVAHYRDARGMSSLAPEAGMAVLERVIGQDRAQLLVAAVVDWPVFLSWYPTPPPLVSALAAAAAREVPAGQGGSLLAAFRAADEAARTALVAERFAALAAGVLRVRPEQVDADARLGSLGLDSLLAMELRARTHTELGVSLPVVALLSNGPVSELTERLHAGLTELAAAGGPVAETAVELFTDEACYPLTHNQQALWFLRQLNPDGFAYNIGGAVEVRAELDPELLFDAFRTLIARHPSLRVNITTEDGRPVQRVRPEAVADTGLLDVSGLPWDEVRARLVAEYRRPYDLERDPLVRLRLFRRAPDRWVLMKAVHHIVSDAISTFVFIEELFEVYHGLRTGRPAELAPVRARYLDFLNRRNRFLAGPEARRMLEYWREHLPREVPALELPTDRPRPPVQTDNGASEFFQLDDELSARVQTLAREHNVTVFTVLLTAYYLLLHRWSGQDEIVVGSPVTGRTEEELASVYGYFVNPLPLHVSLAGEPSVAELLGRVRDTVLGGLDHQEYPFVLLVEELGLQHDPSRSAVFQAMFILLTHKVGVERFGYTLEYIELPEEEGQFDVTLSAYEDRSDGRFHCVLKYNTDLFDAATVRRMAAHYQNLLDGLTRAEGERPAGRLPMLGAGERERIVTGFGGVGRRIDHDVPVHELIGKIAAQFPEAVAVSVPGGRRLGYRELDQRSRRVAASLRERGVGAGTVVAVRLAKSPELVIALLAVWRAGGAYLPLDPDHPAERLAELMENAGATLVLTDGRRGGAARLPGRPVTLDELDRPGTEERPEPAVDLDQTAYVIHTSGSTGRPKAVRVSHRNLASVFVAWQQEYRLDTDVRVHLQMAGLSFDVFTGDLVRALSSGGTLVLVDRDLLFDTARLYRTMRAEGVDCGEFVPSVARGLLAHCEREGLGLEFMRLVIVGSDAWRADEHHRLVALCGPGTRVVNSYGLTEATIDSAYYEGPAEGLEPGRMVPVGRPLPNSELYVLDRHGEPVPPGVAGELWIGGAGVADRCLGDPERTAERFVTLEPGGEPVRLYRTGDLGHWDAEGVLHLLGRRDGQVKVRGHRVETGEIEARLAARPELAQVCVTVRRDETGENVLCAYCVPAPGAAADARELRRHLAEQLPTYLIPAHFTELSALPLTANGKVDLDALPKPRAEAGPERYEPPVTLYETRMAAHWRSLLGLERPGLRDDFFEAGGSSIKLIQLIHHLRTEFNASVPVGRLFKTSTLHGMARTLEDVVTGRLPGAEPYLWFNPGADPAATVFCLPPAGGHGLVYRQLAARLPEHRFAAFNYLSGPDKAARYADLAEELHPGGPYTLFGYSLGGNLAFEIAGELERRGRAVDLVLIMDSYRMAEAVALGEEHLAEFEAELTEHLRRHTGSEIVARETVEQAREYLAHCAAHPSLGVLDAPIAVISDQDKLLRFAVDEPGGWHGGTAAGCTVREGHGRHAEMLDGSFLDGNAELVRALLTGGAANGRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01061 Amino acid adenylation domain-containing protein MRVDGGLLPKPCTTRGPGSDHGPHPGHRRPGRLLAARGISPRIGAAKVTVTVGEVLALVADRLVLPAEQLDPERSFVAAGADSLSLMALARAVQSEFGVRVSVRELFTGVDTPQKLAEAVAGRAMNRSAPAVPAASAAPAQVPTTALATEPVGHAPVAQPPAPTGDALESALALFTDQLQLAGKMMTRFSELTSEQLRVLRGLHPGPAVGASPALPAAQPAPETDLTDDVATAEPLPATGTTRRPPAGAPRTGTPDPAPAGTTARTSPDFSLYFFGDYPAPDSAVAYQHLLQAAEYADELGFHALWLPERHFHSFGALFPNPSVLAASLATRTSRIRLHAGSVVLPLHNPIRVAEEWAVVDNLSGGRVGLGFASGWHSTDFVLAPENYGRQRDIMYEHLETFRSLWSGRSVAMTSGDGRPTEVSLHPRPVQGDDVPLFAAVLSNPESYERAARAGLGVVTNLMTQSVEDLATNIARYRAARAAHGHDPATGRVVVLVHTYLEPDAERARQEARKPFCDYLRSSIDLFDNAANSLGIDVDLLATHQDDLDYVLDLAYERYCETRALIGNAAEVRPVLDSLTAAGADEIGCFIDFGVPPERMLGGLPELDRLRAASTEPRAEAAPVPAAAPRTAAVTALQRQLWLLDRMTPGSHTYYEPKALFIEGPLDTEALRGALRRVVARHPQLRAVFRERADRLEQVVLDAVAVDCPVTELPGHDDTAALLRLRDLEDETDFDLATGPLIRARIGRLDGERHLLYLVAHHAVLDALSTRILCRDLAAYYRAWPGEPTDLPELPPWPATVQESSTADGLAYWQRDLADASPLTLATDRPRTAGHEVRGATLVHEIDGELRGGIRSLARAEGCTPFMALLGAVSATLGRFAAQDDIVIGTAVTNRPEDAADVVGMFVETVALRLDLSGGIGFRELLHRVKARTTAAMDHRGVPFDQIVEVVNPDRSSGANPLFQAAVEYEEELGSVFEDTGLTAEFREVPRKHAPFGLTFYFSDRAAGIRCTVEYDAGLFDESTVRRIAEYIEKLLRRSVDAPDAALCELLALTARDEWSLAGFQGERTETEPATLHGLFEEQAALTPDALAVAGVGDPLTYAQLDAAANRLARRLADRGLAEGEVAAVSVSRGPGLATAVLAVLKCGAAYVPVDLALPAERRAFMLSDSGARLVVADGTLDGDTADTLPCPVQWLEDVAPSDTDEPLGRTVDDEATAYLFYTSGSSGRPKPVAVPHRGPVNLIRWQLRTLGALRTAQWASAGFDVSVQEIFSTLASGQALITVDDETRYDPAAVAAQLRHFEVERMSVPFTPLKYLARELKAVPSLRQLLISGEKLTLTPELRELAAHCPELSLYNQYGPTETSVVVTSHRVNPATETVVPIGRPVDNVTLAVVDDSGRPVPVGVPGELVIGGVAVSHGYHGNPDATARGFFRTPDSGERRYRTGDLVRWRDDGVLEYIGRIDEQVKIRGYRVEPEEAQWALGRLDGVREAVVLARPGESGDTELAAFVVLSPAHAPDGDWSAPLRAQLATVLPHYLVPQSWVRLDRIPYGATGKLARGELLTLRAEPALAATDVELSDLEPTVHKLWAVELGVDTIAPDTSFFDIGGNSLSAVRLLERVLTEFGQRIPVADFFAAPTIRGVAHRLTVLQGEER Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01066 Amino acid adenylation domain-containing protein MVPGAARPGHALREPPRGRSHPLRRLPVLHRPGRDRGVRGGTGRPVRRLRRRTARFRDGRRGQQVSRTARKIEDILPLAPLQEGLLFHSVYDEGELDPYVVQMSFDIDGALDTAALRTAAEKLLARHANLRVAFRQRKSGDWAQLVMREVPLPWTERDLSALPETDRAEAAAGLIAAERATRFDVTRPPLLRFTLLRLGADRHRLVLTNHHLLLDGWSLPVLMGDLFALYDAGGDDSALPRVRPYRDYLTWLEDQDRDAARDAWRDTFADLVEPTLVAPGADRAAVAGAEVRAELPREETAALTELARGRGLTLSTVVQSAWAIALSKHLGRDDIVFGTTVSGRPPEIDGVERMVGLFINTLPSRVRLRAAEPLAGLVARVQREQAALTPHQHLGLAEIQRTVGHGELFDTSMVFQNYPVNRSGTAGTGIGAAISLAPGKNREATHYPLLLIAAARDSMTFRLNHRPDLFDAATAQQILDRFVRVLRALVTDPEQPVGRLDLLTDRERDSVLREWNDTAHDVPDATVLGLFRAQADRTPQAPAVTSAGRTLTYAELDARSSRLAHLLAEHGAAPERFVAIALPRDCDTVVALLAVLKTGAAYLPVDPDYPAERIAFMLADTEPALLLTTRELAPGIPDSGAPRLLLDDPAHTGDLAARPDTAPTVPIPPGLPAYVIYTSGSTGRPKGVVIEHRSLGAYLQWARDAYPAMTGTSLLHSPISFDLTVTALYTTLVSGGLVRVADLDERAAEGPGATFLKGTPSVLALLEALPAEASPSELIMLGGELLLGEVADRWRARRPDADLLNVYGATEATVNSVQYRIPAGAPAPTGPVPVGRPFWNTQVYVLDSGLRPVPPGVPGEAYIAGTGLARGYWRRAALTSERFVANPYGPAGSRMYRTGDVLRWNHDGRLEFVGRGDGQVKLRGYRIELGEIEAVLAGHEGVTQAAVLLRQDQPGDKRLVAYAATAGASVPADALRALAADRLPDYMVPSAFVVLDAFPLTPNGKLDRRALPAPDYGPQAGGGRAPRSPREDILCTLFAEVLGVGSVTIDDDFFALGGHSLLATKLVSRIRSALGAEMAIRQLFETPTVAGLSGALDTGNGAARTPVTAVLPRPERLPLSHAQRRLWFLHRFEGPSAAYNSPVALRLSGALDRAALEHALADLTARHETLRTVLAEDAEGPHQVVLDEARPSLAVVSSDATRLAADLSEAAGHAFDLASEPPLRATLFEVGGDEHVLLLLTHHVATDAWSRAPLARDLTAAYAARMRGAAPQWAPLPVQYADYSLWQRDVLGTEDDPDSEAGRQLDYWGKTLAGLPQELSLPFDRPRPAVASHRGDVVTFELPPELHDRLARVARDSRTSLFMVLQASLATLLSRLGAGTDIPLGTPIAGRTDDALDDLVGFFVNTLVLRTDVSGDPTFAELLERVRTADLAAYAHQDMPFERLVEAVNPERSLSRHPLFQTMLNLNNAGPVEALDEIAKLPGLTVHHEPVETHRVKFDLGFSFAESHSTTGTPGGLRGALQYSTDVFDRSTAEALVQRMVKVLEWVVASGNGSRVSEVEVLEEAEREQILSGWQGASRPVRGASLPQLIAEQAERTPDAVAVECGDRALTYGELDAWAGRVAGWLQGQGVGRGTFVAVKLPRSVELVVALLAVTKAGAAYVPVDPEYPQERVAHILSDATPALVIDDTAMLEQETDGPFDTVRIDPHDPVYVIYTSGSTGRPKGVVVEHASVGAYLERAREVYPDASGTALLHSSVAFDLTVTALYTPLVSGGRVVLTDLDEHAATTGQPTFMKVTPSHLGMLEALPEEVSPSGTLITGGEALVGEALAAWRAAHPDVTVINAYGPTEATVNCTDFRIEPSDVMGSGPVPIGRPFWNTRAYVLDDHLRPVPPGVTGELYVAGIVLARGYHNRPDLTAERFTADPYGPPGTRMYRTGDTARWTHTGQLTYTGRTDDQIKLRGFRIELGEIQAVLMTHPHITQATVIVREDQPGDQRLTAYTVNTAGTDTTTDDLAAHTAAHLPAYMIPSHFITLDQLPLTPNGKLDRNALPTPQYGPQNENGRAPRTPHEQALCTLFADILGTDTVTIDDDFFHLGGHSLLATKLVSRIRTDIGAELPIRQLFETPTVAGISAALADKARAARRGVVAVDPRPARIPLSYAQQRLWFLNRFEGPSATYNAPVALRLTGALDQEALRQALADVVTRHESLRTVFAEDAEGAHQIVRGPADARPEFTIVETDEARLRDDLAWAAGHPFDLAAEIPFRASLFALSEEEHVLLLLTHHIVSDAWSRAPLARDLTAAYAARVRNAAAPEWAPLPVQYADYSLWQRDILGTEDDPTSEITRQLDYWTHTLTGLPDQLELPYDRPRPAVATYRGDRIPFDIPAELYERVGEVARRVQASPFMVLQAALAALLTRLGAGTDIPLGTPIAGRTDEALDDLVGVFLNTLVLRTDTSGNPTFAELVDRVRERNLGAYAHQDLPFERLVEAVNPERSLARHPLFQVLLTLNNTDYQGALDSLGDLPGLRAEREPIESSVAKFDLAFGYTERRDPHGRVTSLHGVLEFSTDLFDRRTAGALVDRLLRFLDHAVTTPDVKVGDIEILAGAERGRLLELWNDTAREVPERSVVELFEERVASNPLAEAVVAGEEALSYEELDARAERLARVLVERGAGAERFVAVALPRSVDLVVALLAVWKTGAAYLPLDTEYPAERLAYMLDDANPVLLLTTSDLTPVLPEEPAVPRLLLDTPETTEALSRPAGDRSLTRPALANPAYVIYTSGSTGRPKGVVVPQGALVNFLTAMRDRFELGAGDRLVAVTTVGFDIAGLELFVPLLSGASITLAERDVVRDPAALCRLVRSAGASVMQATPSLWRAMLAEDASALAGVRVLVGGEALPADLAEALVQRAMSVINLYGPTETTIWSTEWPVTAEGARRPRIGRPIANTRVYVLDGTLRPVPAGVPGELYIAGDGVVRGYHGRPGLTSERFVADPHGPSGTRMYRTGDLVRWTVDGELEYLSRVDDQVKLRGFRIELGEIEAVLAGHERVAQAAVLVREDRPGDRRLVAYLVPAAEAVETAEVRAHLAAHLPDYMVPSAFVTLDSFPLTPNGKLDRRALPAPDYDQGTSEGRAPRTPREDILCTLFAEVLGAGSVTIDDDFFALGGHSLLATKLVSRIRTVLDTEIAVRRLFEAPTVAELAAVLDNATGTRKPLRAPVSRPDRVPLSYAQRRLWFLHRFEGPSATYNLPVALRMTGTLDQEALRLALADVVDRHESLRTVFAEDAEGPYQIVQDTAEVSLTVTATDEEHLPEDVDRASRAPFELSEEPPLRAFLFELGEDEYVLLAVVHHIAGDAWSMGPLAQDLTSAYAARVRGAAPEWAPLPVQYADYSLWQRDVLGSEDDPDSEAGRQLEYWKNSLSDLPAELSLPFDRPRPATASYVGDRVTFELPEDVYGGLVRVARAGRSSLFMVLQTALATLLSRLGAGTDIPLGTPIAGRTDDALDKLVGFFVNTLVLRTDVSGDPTFAELLERVRTADLAAYAHQDLPFERLVEAVNPERSLSRHPLFQTMLTLNNTDQGAASAVASLPGLEVSSRPVGIGAAKFDLSFRLAERRPTSESESATLGGALDYSTDLFDRETAQSITERFVRVLTALAQDPDRRVSEVEVLEEAEREQILSGWQGASRPVRGASLPQLIAEQAERTPDAVAVECGDRALTYGELDAWAGRAAGWLQGQGVGRGTFVAVKLPRSVELIVALLAVTKTGAAYVPVDPEYPQERVAHILSDATPALVIDDTAMLKQKTGKPFDGVRIDPHDPVYVIYTSGSTGRPKGVVVEHASVGAYLERAREVYPDASGTALLHSSVAFDLTVTALYTPLVSGGRVILTDLDEHAATTGQPTFMKVTPSHLGLLEALPDEISPSGTLITGGEALLGEALASWRATHPDVTVINAYGPTEATVNCTDFHIQPGEPVPSGPVPIGRPFWNTRAYVLDDHLRPVPPGVTGELYVAGIVLARGYHNRPDLTAERFTADPYGPPGTRMYRTGDTARWTHTGQLTYTGRTDDQIKLRGFRIELGEIQAVLMTHPHITQAAVIVREDQPGDQRLTAYTVGTDTTTADLAAHTAAHLPAYMIPSHFITLDQLPLTPNGKLDRNALPTPDYNQHTSEGRAPRTPHEEALCTLFADVLGTDTVTIDDDFFHLGGHSLLVTKLVSRIRTSLGAELPIRQLFETPTVAALSAVLGNDTAPSRPTVTAVDPRPARIPLSYAQQRLWFLNRFEGPSATYNIPVALRLTGALDQEALRQALADVVTRHESLRTVFAEDADGAYQIVREPADARPDLHVIETGPEEVEERLRDAARRGFDLSAASGELPFRVTLFEVGDGEHVLLLLLHHIVSDAWSRAPLARDLTAAYAARVRNAAAPEWAPLPVQYADYSLWQRNILGTEDDPTSEITRQLDYWTHTLTGLPDQLELPYDRPRPAVATYRGDRIPFDIPAELYDGVAALARDTQASPFMVLQAALAALLTRLGAGEDIPIGTPVAGRTDEALDDLIGVFINTLVLRTDTSGRPSALTLIERVRNQTLEAYAHQDLPFEQLVEAVNPERSLARHPLFQVLLAFNNTDTAAVEDAVAKLPGLSVSRATADTGVGKFDLSFAFAEQAGSGTGLQGVLEYSKDVFDRETVETLGLRYLRLLRAMVDAPQKPVDEAVLLDEAESRTLLSGWNDTACEVPGRSTVELFEERAASDPAAEAVVAGTHSLSYGELNDRADRLARVLAAHGAGAERFVAVALPRSTDLVVTLLAVWKTGAAYLPLDTEYPAERLAYMLDDANPVLLVTTSDLSPLLPASTQVPRVLLDEPGLQEELAAPAGPGPLRGIHDPSASAYVIYTSGSTGRPKGVVVPHGPLVNFLTAMQRQFPLGANDRLLAVTTVGFDIAGLELFLPLLTGASAVIAERDTVRDPGALCTLIRTSGATTMQATPSLWRAVLAEDPTVLTSRHVLVGGEALPADLATALTRHAASVTNLYGPTETTIWSTHWPATSDTAHHPRIGHPIANTQIYLLDHTLQPVPTGTPGELYIAGHGVVRGYHNRPGLTAERFTANPHGPAGTRMYRTGDLARWTPDGTLEYLARVDDQVKLRGFRIELGEIETALTAHPHVAQAAVLVREDRPGDPRLVAYLTPTAHQPIPTTDLRQHLATHLPDYMLPTAYITLDAFPLTPNGKLDRRALPAPDYATHTEGGRAPRTPREELLCTLFAEVLGTDTVTIDDDFFTLGGHSLLATKLVSRIRTVLDTELAIRQLFEAPTVARLAGVLDSSAAARGRLVAAPRPARVPLSHAQQRLWFLQHLEGPSDAYNVPISLDLTGELDQEALRLALADVVDRHESLRTVVVEDGSGAAHQVVLGREQTRVPLAVERVASDAEVDARMRRAAGYVFDLASEIPLRATLFAVGEEGVTDRWALLLLTHHIASDAWSRGILIRDLVAAYAARTTTGRAPDLAPLPVQYADYSLWQRDVLGSEDDPGSEARRQLDHWKRALSGLPEELSLPFDRPRPAVASYRGDRVAFDLPQDVYERLVRVGREQGASLFMVLQAGLAALLTRLGAGTDIPLGTPIAGRTDDALDDLVGFFVNTLVLRTDTSGDPTYAELVDRVRAESLAAYAHQDLPFERLVEAVNPERSLSRHPLFQTMLSFDNAGRAATHADLAGLAVSGRTLGAPAAKFDLSFELAERPAGPDRAADLSCALDYSTDLFDRGTAQDVADRFVRVLTALADDPGRRIGETEILGRDERRRMLVEWNETAVQHADRTPVHVLFEERAAAEPEALAVVSGEERLSYGELNARANRLAHRLLGRGVGRESRVAVFQERSAELIVATLAVLKAGGVYVPIDPQQPASRSEFILRDTGAVALLTDRDPGDLPFAVDVPVLDVGPGTDLSGEADTDPGVPTDAEQLVYVMYTSGSTGTPKGVANTHHNVVHLAADRYWRGGRHERVLMHSPYAFDASTFEIWTPLLTGGTVVVAPAGRLDAADLAAAISGHGVTGLFVSAGLFRVLAEERPECFRGVREIWAGGDVVSPTAVRRVLETCPGTVVANEYGPTETTVFSAVNPLRDPAEVPEAVVPIGRPLWNTRLYALDERLRPVPVGVPGELYIAGSGVARGYLGRAALTAQRFVADPFAGAGERMYRTGDVVRWLADGRLEFLGRVDDQVKLRGFRIEPGEVEAVLAGRPEVSQAAVVLREDRPGDKRLVAYVVAGAAAEPEALRAHVAGTLPEYMVPSAVVLLDGLPLTLNGKLDRRALPAPDYGADTERRGPRTEREKVLCGLFADVLGLAEVGVDDGLFDLGGDSIMSIQLVSRARRAGLELSVRAVFEHRTVAALAEVVTETDTTVTEEPGAGIGDVPLTPIMRWFLERGGPVDGFNQSRLVQVPASLRLPDLTAALGALLEHHDALRARLTDGSERRLEIRGPGAVDAGSVVRRVDAAGLDDDTLQDLVRGETVAARERLDLGAGRVVQSVWFDRGDSRPGLLLLIVHHLVVDGVSWRILVPDLAEAHRAVVAGRPVELQPVGTSLRRWAQRLTEVAGDPARTAEADWWRSVLRPADPLLGRRPLDTARDTYASARHLTLTLPVAVTERLLTRVPAVFRAEVNDVLLAAFALAWARRGGGRGAGVLLDLEGHGREEELVGGADLSRTVGWFTSLHPVRVDAGPADLADAFAGGPAAGAVVKRVKEQLREVPEKGIGYGLVRHLNPRTAPGFAGLPTPQVAFNYLGRFTTAGVENAGSEAVPDWTVLATASGVGGTDPRVALAHPLELNARTNDGPRGPELSATWSWAGGILDEDEVRELAELWFRALEALADHAENPEAGGLTVSDVSLSLLDQSEIELLEDEWRNL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01071 Amino acid adenylation domain-containing protein MPTPDRRSAPPPEHRPLLAAQEGIWAGQQLDTESPAYNTAEYLRIAGPVDTAVFDRALHRVVAETEALNATFDIDDTGRPRQATTPAGDWRTHIADLTAEPDPHAAALAWMDRDTARAVDLTRGPVFGHALLRTGPQEHLWYHRVHHIALDGFGLSLVARRVAEVYSGLMAGDPVPESGFGTLDSVREEEAAYLASARHTQDRAYWTDRYADHPPVATPADRSALPARTFHRHVTDLGPAAAHRLRTGARELSVTWSEVLLAVTAAHLHRLTGAPEIVLSLPATGRLGSVSLRVPATVRNILPLRVPVAPDDGLRDLAPRVSRELRAGLPHQRYRYERLRRDLKLVGGGRRLSGPGVNIMPFEYDLRFAGHPSTVHNVSAGPVDDLAVNVYDRGDGTGLRVAVDANPDLYTEAETAAFQEGLLALLEQALTDPGRPLGGPRAHRTVAVLDGGPLPAPARPVLSLIADHATRGGGAVAVEHAGERLTYARLLGAARDVARRVTALGVAGGDVVAVALPRGTDAVTAVLGVLMSGAAYCPLDPKAPAERTARLLADTAPALVLTTADRAADFADHTVLPLHEPDPAPAGAHTPSAKGDSAGAGSTARRRSELGPLDGNESQEPGPRHFAAPAVEDPAYVLHTSGSTGRPKGVQVSHGALAHFVAAATHRYGLRREDRVLQFAPLHFDASVEEIFLTLCAGATLVIRPDDMTESVPGFLDACARLRVTVLDLPTAYWHEVAHTVSTGAAALPRAVRTVVVGGEPALPERVERWRKAVGTSVALLNTYGPTEATVVATVADLHDPGLGTGDVPVGLPLPGTRAAVLDGELYLLGPALADGYRPEVPDSARFAPLTALPDGPRAYRTGDLVRIGEDGQLRHLGRADDEFKISGQRVQPAEVESALLFHPGVREAAVAGQVLPDGTRRLVARLVPEGPAPSAADVREHLRARLPAAMVPSAVEFVGRLPRTGSGKIDRAALAAPPARRAPTTGSPLEQTVTGVWCRILGIDAVAVDDDVFDLGAQSLQAIQAANRLGTELGRDVKVAWLFQHPTAGGLARFLAQGPQPRAAGPAGLPPALLADARLDPDIRPGTRSAPRDAPRRILLTGATGFVGAHLLAQLLSDTGAEIVCTVRAADVPEATGRVHAALARHGITLDERTSARLTALPADLAHPGLGLPPDTLAGLAASCDAVFHNAATVSIMRDYANLRAANVESTRRLVRLAAVHATPLHYVSTLSVAPPASRAPEVPEAFLPPHEGLRHGYQQSKWAAERLLQQAAERGLPVTVHRLGRVIGRAGTGGVNERDFLWSVLRAGIPEGIVPELFEDEIWTPVDFVARALVHLSLTPDTAATGPVFHHATLPRVRLADVYDWVRAYGYPVRALPLARWRERLPRSADVAATTLAFFDAAELDAAGPDSTELGFSEPDSTGPDFTGRDSHDRTTATDLRLGHVRADRVRAGLVGSGITCPPVDRALFFRHLDHCVTAGVLPAPAGRPVSRSGPAAK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01076 Amino acid adenylation domain-containing protein MMEPTARLVLLSPKHLTDLRRRTGDHSDAALATACAIGLSYWATGQSPAGLDLTAATLFGDVLGWADNGGAAPEGWGVAADGRTITLPEGVVPDDAQLALDDLADFPGRPLGTIGPAGPTARLENLARWNDTDADRERPTLMEMFLEQARARPGAVAVVDERRTLTYRELSDRSAQLAHRLRERGLSDEDVVGISLERSADMVVGLLGVLRAGCAFVPLDPHWPAERRAVVAADARVAVQLNASGEPAPHEPEAVPVDLADWRHGDRPTEGPDPTVRGDALAYVIFTSGSTGRPKGAMIRHEAISERLLWQVHEILDFGHDDASLFKAPLSFDISINEIFLPLVCGARLVVLRPGGERDPHHLLGVIAEQRVTFTYLVSSMLDVLLEMAGDTGRLDSLRHVWCGGEVLTPELYERFRTQLDIPLYHGYGPAETTIGVSHVVYRGAAERLSTSIGRANPNTRLYVLDDELRPVPVGVGGELYAGGLLLGRGYVNAPGLTASRFVANPFADDGSRLYRTGDLARFAPDGSLDFLGRADNQIKIRGMRLEIEDVEAGLAEHPGVRHTCVVPKKNTAGGTYLVGYVIPAAGHGSLRPDEVKAWAAEHMVEYMVPTHVVVTDAFPLTANGKLDRQALPEPTVAASAARPPGTENERAVCTAVAAVLQLDEVGTDQDFFRLGGDSILAISLLSALRDAGLYVTARQIFTHSTVGALAAVASREDTAAVDHRDTPTGTVVGPPVVQWLGETTGAIDGFVQSVVLNTPAALTADALDEILTALVRRHPMLRARLVRGDRWGFDIPDEVPAGALWQESDRPLDSCTALATEALDPAGGAMLRAVWRRSARQLVLVAHHMVIDGVSWRVLMEDLATAWRQYASGAPVELPVEGTSFRRWTGLLERAASDADGQYFRRPLPAADEPVGRRALTEDDTVARERIRTVETGAETTAAVLGTVPAAFHAGVGDVLVTALAVALARRRRDLGQDQTFAHLELEGHGREAAFVAPSAGFEPELSRTVGWFTTLFPVVVDPGTAPDLTAPEYLATALKAVKEDLSRVPDNGISYGALRYLNRVAFDAPAPQVLFNYLGRFDAGAPGDWQLAGSTGQLGEKRDPAMRLPRALEFNAVAEPGPDGEYRLVTTVSWPEGLFTDQDIDALAGHFQDALTGLAALERGGHSPADFRPLRLTQADVDDLDGPALRDILPLTPLQEGLYFHSVYDDETAGSYVEQQLLTLDGDVDADRLATAATRLLTLHPGLAARFTALADGRVVSVLESGHHAPFTTLDRPGITDEEIRDLAERDRRAGFDLATGPLMRYTLIRAGAGRHVLVQTVHHIVADGWSVPPMLRTLLAEYHRPGSAHPLGGFPEHVRRLAALDDRESDRVWREQLAGLPGPSLIAEGHTPSDRFADTATTPGIDVDAAARAAGVPLSVAVHSAWALTLGGILHSEDVVFGSTVSGRDADVPGIQnMVGLLINTVPVRARWSADTTAAELLAQVRAHQSAVLPHQHVSLARTARHTGTGPLFDTLVVFDVATDVGALREPGDTLVVTDIVNEGAPHYPLTLVVERTPDGTPRFNAVHDAALLRESQVQDILHTFTRTLTTLLTSPDTPVAAPVPHTARRAPAVAPATLGDLLDAAARRDPAATAVTQCSLDGATRSLTYGELTEAKDGLAAVLRAAGAGPGRLVAVAVPPSVEQVVALTAVTGAGGAYVPLDAAHPDERLEYILADAAPQVVLVDREQRERFTRLLERAGVPARVLVQGDEPAPADDGPASPAGWHDPAYVIYTSGSTGRPKGVVVPHSGVVTLLAHTQADMGFGPDDVWVQFHSFSFDFAVWELWGALAHGGELLVPEYALTRSPVDFHRLVREHRVTVLNQTPSAFHRFIEADRHAGEPLPALRRIVFGGEALDLGRLRDWVDRHGTATPELVnMYGITETTVHVTHRVLTDADFGPGDAPSPIGTPLPGLVVHLLDDRLRPVPPGRVGAVYVAGDQVSLGYLGRPGLTAGRFVADPFTGDGSRMYHTGDLARRTLDGELHFAGRADDQVQLKGFRVEPGEVEAALRDLDGVSDAAVTVADGGDHLVAHVVGRAPGDLTALLAARLPAHMIPGRVLSVDALPLTVNGKLDRKALAERAANAPLPDGALHRTDSGSAAPDGPAVLDTVVRVFAETLPGSTPDADTDFFAAGGDSIVAITLINRARAAGLSVTPRDVFLLKTPRALAEHLTASTPPPATPEPVRREDGPLPPTPIILRQRELGGSLARFAQARTLLAPEGTAFADVERAARAVVAAHPALRLRLRVDHGVWSLRTEADREVTVVRADGTDPTAAADEAASRLDPESGDVAAFSWLAANRTLVVTVHHLAVDAVSWLILLDDLAGALRGTPVPAPTTSYAEYAEALTHRAAHAAPGLGHWTTALQAPTPLPPPEALRETTAVLAPGISDRLTRTAPTALGLGLTELLCGALRTALTRIQPSPTDLAVDLERHGRVPALEHHDYTRTVGWFTAVAPVRLTPHTDPVAAAREVTERRPDEREHVAYGLLRYLNAQTAPLLTARPQVLFNYLGRGAESEAPRLAGGDRGSPYAVEVNAWTDAATGSLHAVFTLAEGIPDTLTAHWLAALEQLADSAATAERTAPVTPLQRGLYFQSQLTGPTGHYVAQSWFTLERRLDTDALADAMAHVIARHPVVGAGFTTDDDGNPVQVLGAGRRVPVRTVEAATDAEAEALRLADRDTGFDPAEPPLVRLTVVRLPGDRDGLLLSYHLLLWDGWSRETVLRDLFDAYEDILAGTPLDTAPATPRFEDHARALAARDPAPAERFWSEHLAPLSGPTLLAGPAPSLSDDLPHALVHTLTAAESERLRETARTHGVTLNSVLTGAFGLLLGAHTGRADAVFGVTVSGREGEGASGVVGVLLNTVPMWTRARPHDTVRAYLTAVQASRVAAMEHEHLGLGEIQRAAGHDTLFDNLFVLQNFLDLDAFAEMNARHGITSVQADDSTHYPFTWVVTPGDRLTVKLEHRDHDAGRARRLLDDYLRVLADLAASDGPLGALPGPAPAPAPGARTDIGTDTVVDRFDRAADRNPRRVALVAHGSTLTFAELRDRSRAVAGVLVRRGIGPETTVGIAVPRSLDSIVALFAVLRTGAAYVPLELDHPDERIAAIVADARPDVILTVGTVAPRLTGDLIELDRPLPEAEPYVTFAPDDPHRLRHPAYIIHTSGSTGKPKGVVTEYAGLTnMLVNHRRRIFEPVLAEHGHRTFRIAHTVSFAFDMSWEELLWLADGHEVHVCDEELRRDAPRLVEYCAEHAVDVVNVTPTYAQQLVAEGLLDDPARRPALVLLGGEAVTPALWRRLAETEGTVGYNLYGPTEYTINTLGVGTFECPDPVVGVAIDNTDVHVLDPWLRPLPDGVPGELYVSGIGIARGYLGQTAQTAHRFVACPFGAPGERMYRTGDLVTRRPDGNLTYLGRTDQQVKIRGHRVELGEVEAVFTAHPAVRFAAAVAQPDPQVDGAHRLAAYLVLDGADLATVAAEVGAGLPDFLRPTHYARVDGIPLTVNGKADTRALPEAKPLGALTTAGERPPATETETTVCEFFAEALDLDDDEVSAVSDFVSLGGHSMLAVRLTGLLRREYGPVITIRDLFTLRTPEAIARHLDDH Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp01081 Amino acid adenylation domain-containing protein MQETAPDPVAGRQPAPAAGPEDAVAALAHACAAALASDPASVRLAARLKVASVLLGRASPAPDASWRDLVRHVGTDDGRSEAEEAWANASAAAGATAERLGRYELRALRLMRDDPDLPHTRHGLLTPEETEAVVARGAGPLRPLPGRRFHELFEERVRRHPDAVAVVHGTTTRTYRELNDDANRIAGALLREGLAPEDVVAVVTGRHPLWPAAVLAVFKAGGCYLPLEPEFPASRIARTLTRSECRWVLSDPDVASLDEALNGRDTIRRMTVGDLARGDGPTRDPGVAVAGDQLAYVYFTSGSTGEPKGAMCEHDGFLNHLYAKIEDLGVQEGDTVGQTAPQCFDISLWQLVSPFLVGGRVLLVEQEAVLDVARFVDLVNRHRVQVLQLVPTYLELVLAEAARGRAALPHLRVMAVTGEALKKELVRRWFEQFPGVPLVNCYGLTEVSDDSHHGVMHTVPDHRSVPLGDTIRNCRVYVMDEQLHLVPDGAPGEIVIAGVCVGRGYVNDPDRTAAVYHQDPLRPAERLYRSGDFGRRLPSGELEYLGRRDAQVKISGFRIEIGEIEDRLLQVPGVRDGAVVVAGTDDAPQLVAYYTGEDAPDGAGTAHALGTALPHYMVPHRLHRVRELPLSGNGKIDKKALTARARDNAHARGSAGTGAPRLDTPAERRVAAVWARLLRVPEDRIGRDSRFTDLGGTSLTAIRLAIELDRRVTVAELRDTPTVADVAALLDGKSAPARATAPAGPAPATTPARPAEGPAPLPLLDCRAADPEPDPAARATAHRAPALAALAASGAVMLRGVGARTPADVARVAAALGIEPLTEREGFAPRTALAPGVYSGSHWPAEDPMCMHHELSHAATVPGTLLFACLTAPDSGGRTTVADSQQVLAALPSGLTARFAEHGWLLRRAYHDVGLSWPEAFGSTDRASVDAYCAEAAVEPTWLADGSLLTRQRRAAVVPHPRTGAPCWFNQIAFLNGLTLEPAIREYLTDVYGPGGLPFDTAAGDGGPVTAGTVEEINAVYDRFTVGEPWQQGDVLLVDNIRTAHAREPYEGAREIAVVLGDPVRLPGHVLPLSDGGPS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01086 Amino acid adenylation domain-containing protein MSEARLLRRPVSAAQSGIWVAQHLHADSPLYNCGGYYEIAGPVDAEIFAEAVRRGVQETEALRSRFAQEERDTDSGPEVTLHQLVEPAEPHPLRFVDLRAASDPEAAAHRWMNARMARPFDLTRGPVSEQALLTLADDLHWYFHGYHHAVLDGFGQSVYATRVAALYSALLAGEEPSPTGFATLDRVVADEAAYAGSRRHTRDRAHWREVFTDLPEPVSLGRASGSTHSLRRHVRTLPTPLAERLPGAAARLGVQWPALALAATAAFFHRMTGGTDFTFSIPLAGRSGRTSLTTPSAMVNVLPLRVRLTSDIRFTELAAQVSRSLADVVRHQRFRGEELIHELGLSGAGQARLGPTVNIMAFAGEPLFGTTPAVTHPLSTGPVNDLKINFYGTADSRTGIRVELDGHHELYGADELAAHCDRLVRVLEWVADSDDESRVSEVEVLEEAEREQILSGWQGASRPVRGASLPQLIAEQAERTPDAVAVECGDRVLTYGELDAWSARTAGWLQGQGVGRGTFVAVKLPRSVELIVALLAVTKTGAAYVPVDPEYPAERVAHILSDATPALVIDDTAMLKQETGKPFDGVRIDPHDPVYVIYTSGSTGRPKGVVVEHASVGAYLERAREVYPDASGTALLHSSVAFDLTVTALYTPLVSGGRVILTDLDEHAATTGQPTFMKVTPSHLGLLEALPDEISPSGTLITGGEALLGEALASWRATHPDVTVINAYGPTEATVNCTDFHIQPGEPVPSGPVPIGRPFWNTRAYVLDHRLRPVPPGVTGELYVAGIVLARGYHNRPDLTAERFTADPYGPPGTRMYRTGDTARWTHTGQLTYTGRTDDQIKLRGFRIELGEIQAVLMTHPHITQAAVIVREDQPGDQRLTAYTVNTVGTDTTTDDLAAHTAAHLPAYMIPSHFITLDQLPLTPNGKLDRNALPTPEYNQHTSEGRAPRTPHEQALCTLFADVLGTDTVTIDDDFFHLGGHSLLATTLISRIRTTIGAELPIRQLFETPTVAGISATLDQQPARAAVRRPGVTAGPRPGRIPVSYAQQRLRFLSLLEDGSTAYNAPGALRLTGALDQEALRQALADVVTRHESLRTVFAEDESGFTQVILEPYEVALGLDVVAVDEERLAARLAEAARYSFDLAAEPPLRATLFEVGDDEYVLLLLLHHIAGDGSSMRPLARDLAAAYAARVRGATPEWAPLPVQYADYSLWQRDILGTEDDPTSEITRQLDYWTHTLTGLPDQLELPYDRPRSEVVTQHGGQVSLRIPAELHGQLHELARTTRSSLFMVFQAGLAALLTRLGAGTDIPLGSPIAGRTDAAVEELVGFFANTLVLRTDTSGDPTFAELVERVRARSLEAYQHQDLPFERLVEAVNPERSLTRHPLFQVCLTLHNTDPRATVAEEARLPGLAVELERLPIEDTKFDLNWELTEHVDGLGRPAGVTVDLEFSAELFDRGTARSVADRFVRLLSATARDVEVPIGEIDVLAPGERTEILDEWSDATRPPVAAALSGSSLPRTADDTRAYVLDDTLVPVPPGVVGQLYVTGSGPAGDAAEQERWLPCPYGRAGWMYRTGTSARWSADGELRLVEVPGRTPVGPADVWPARSRGPRSPREQILCTVFAELLGVASVGIDDDFFDRGGHSLSAVRLLSRIRAVLGVELSIRRLFENPTVAGVVEALDEASGARRPVTAVARPARIPLSYAQQRLWFLNHLEGPSATYNIPVALGLKGALDRAALRLALTDVVARHESLRTLFAEDSEGARQIVLPAAHATPELIEVDVAPGELPGRIRAAASHPFDLATELPVRAWLFSAHDGERVLVLVVHHIAGDGWSMGPLARDLSLAYTARARGDAPAWTPLPVQYADYTLWQREVLGSEDDPDSEISRQLAHWKTALADLPEELELPVDRPRPARQSHRGGRVPFEVSAGLHARLAAFARETGTSLFMVAQAALAALLTRLGAGTDIPIGSPVAGRTDAAVEDLVGFFVNTLVLRTDTSNDPTFAELVGRVRETNLGAYGHQDVPFERLVEVLSPVRSLARHPLFQVLLGFDNNQEALEILRLPGLTVDVHAPETGRAKFDLAFFFDERYGPHGEPEGLGGAVEYNSDLFDRSTAQEFAERLLRVLEGAVADPERPIGRLEVMSPAERDRVVDEWNRTAHDVPPLPVPTLFERQVAAEPRATAVLGEDVTLSYAELNSRANRLARLLAASGVGAEDVVAIALPRSADLVVALVAALKTGAAYLTLDVSAPEQRLRAVLTDCGPRVVVTDLATRPLLGDGIALDVVLDAPETVRELAAGADADLTDADRVRPLDLRHPAYVVYTSGSTGTPKGVVMPMSSLVNLLAWHTGTYCGGVGTLTAQFLAVSFDFAVQEILQALVVGKTLVIPEEHVRRDAYELAQWIARYSINELFAPTLVIDAVLAAAADTGERLDSLTDLFQGGEQFRLSHELREFCASGWRRMAHNIYGPAETHAATTATLPGDIDEWPTAASIGQPLWNASVYVLDAGLRPVPPGVRGELYIGGAQLARGYLGRPDRTAERFVASPFGRPGARLYRTGDVVRWNHCGELEFLGRADHQVKIGGFRVEPGEVEAVLADHPSVETAVVVTREESAGPTRLVAYVVPEGQDADPALGRTLRAHLEQQLPHYMVPSFVVPLDELPLTANGKLDRRALPAPGSDTVAAEPRTEREKVLCGLVADVLGLAEVGVDDGFFDLGGDSIMSIQLVSRARRAGLQLSVRDVFEHRTVAALAEIVTETDTTVTEEPGAGIGDVPLTPIKRWLLARTDDLDAFnMSAVLRVPADVDADALTGAVQALLDHHDALRARLTPAPQRRLEVREPGSVDAGALVRRVDASGADGADLHALVREAGAAARDRLHLGEGRVVQAVWFDRGRDSAGMLLLIIHHLVVDGVSWRILIPDLAEAYEAVSAGRKPALQPVGTSLRRWSQRLTEEAVKPAWVADAAWWQDVLRSAGPPPGRRPLDPARDRQATAGRLTVTLPTEVTEAVLTRVPAAFHAEVNDVLLTAFALAWARWRPGGPELLLDLEGHGREEHLVEGADLSRTVGWFTNLYPVRLDTGGVDLARAFAGGSAAGSAAKRIKEQLRSVPDKGMGYGLVRHLNPATAAGFDGHAAPHVAFNYLGRFTAADCDRAADWTPVTGFDAVAGDPPQLPLAHPLELNSRTEDGPEGSELVAFWTWAEEILDEDEVRELAELWFQALRALVTHSENPHAGGLTPSDVSLSSIGQDEIEAFEEELDDLFDDFDDEPHDFETEEEASK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01091 Amino acid adenylation domain-containing protein MPGRVVEMINAQVRRHPRAPALVAPDGSLDYAELDRRSAYLAGHLTRQGVRPGDVVLIQASRGVALGVALLAVLRSGGAFCVVDPQYPADRIQHMWRRSHARFALIESGLRAPDVPDGPAVLPLRQWATPGSAHRAPAPHRAEPGSEDPAYLVFTSGSTGGPKAVLMPHRCLDNLIEWTLASTSSEPLRTLLFAPLGFDVFVQEVFTAWCSGGCLYTPSDAERVDLQCVWELCREREIQRVFLPPVALRRLADLTVEFGILPGALREVAVAGEALHITPAIRELFGRLPAARLHNHYGPAETHVAVAHTLTGPPRSWPDLPPIGRPLPGMTAQVVPRAEGGELWLTGVGLAHGYVHDPRQTQERFRSILVEGRTVRAYRTGDLVRERTDGALEYLGRADGQLKIRGYRVEPGDIEAALLRHPAVRECAVVAWTSLGSEERRLVAHVAAVPGGAPDAAELRAHVAGLLPDYMVPHHVVLATELPLSPNGKIDRRRLPPPGDADDSAGTLPEPEPGDVRSAVADIWSTVLGVADIPPDRHFMDLGGTSLSAALVVTRLHQRFQVQVSVQEFLYDPRVDAIAALITERAAA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01096 Amino acid adenylation domain-containing protein MSGHRTQQTYTRIPRWTMPGSDEQGAAEHREALPAPLTRALEERAADTGAELPAVLLAAHARVLATVVAEPDLLIGLVPAAGRAESPLGLTVTDSSWADLVGLASTAPAAAPRAEGRPEVVFDLSGLTPTDTAPAGRADPDGTAVGLGEGVVLRVAVVAGSAGLSLRLVYDRAHLDESYARRLAGYHLRALELLAADTSAPHHGRSLLSEEEIDTHLYGLAGPRVDLTDRTFVDHFEDRVREVPDAVAAVHGPVRWTYRELDGRANRVAHALLDAGVRTEDVVAVVMDRTLDWIAAALGVFKAGGVYLPVRPDFPADRVAAQFSRSECAFVLTEPGSATLARKAGELTGRAPTVLSVPEIQASGVSDAAPRVPIAPGQAAYIYFTSGSTGAPKGAMCEHAGMVNHLHMKLDDMEMTNGTAEVVTQTASQCFDISLWQFAAPLMVGGSVRVVDTDALLDVAGFLDEIVTGGVTVVQIVPSYLEVLLTHLEQHPRPLGALRTVSVTGEALKYELVQRWFALYPEIKLVNAYGATEVSDDTMHEVLDRVPDRDFVTVGRSLRNVNTYVLDQDLALVPLGSPGEIAFSGVCVGRGYINDEERTREAFVPDPFRDGTRMYRTGDFGRWLPEGRIEYLGRRDEQVKIRGFRIEIGEIENKLLALTGVREAAVVIDGTDDGQRNLVAFFSGGDGGARPDAEPTTERARDFLAGLLPEYMVPTYFHRLDRLPLTENGKVDKKALIRLAGTLGHGGAAYAAPSTPAEQRLAMLWAQVLGVPLERIGRDDNFFELGGTSLAAVRLLVQLDRALSLKDLVAHPVLADLGRALDERVRGGERAAAENLLQPLANATDPHRILVCFPYAGGNAVNFRSLAAELERDGIAVLGVELPGHDFAGGDDPMADVPEIARRVRDEIAARVTTPVLLWGHCAGAAPALETARLLQEAGRPAERVFVGALLLEDVGALRAEMAEAAEADNKSLLSRLRADNAYVELDELKPERADVVGRAYRHDVLTANSHLIRIREDAGSHRIDAPVDVVVARDDASTARFAADHGDWKAVSDRVTLHELDQGGHYFIGTRAADTAALVRACCPKPTHRD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01103 Aminoacyl-tRNA hydrolase MDGMSGPHVIRGSVLLPEAELVWRFSRSSGPGGQHVNTTDTAVELRFDLARTGALPEVWKRQALERLAGRLTDGIVTVRASEHRSQWRNREAAAVRLAALLAEATAPPPRPRRPTRIPRGINERRLREKKQRSQTKRGRSPKDWD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp01108 Aminopeptidase N MSCMSVLTRDEAQTRSRLLDVHHYAIALDLTRGDETFDSRTAIRFTVRGDTDATDTFVEVKPAELRSVTLDGQPLDPAALDGNRLPLRGLAPGEHELRVDAAMRYSRTGEGMHRFTDPADGETYLYTQMFLDDVQRVFAAFDQPDLKAVFDLAVTAPEGWTVLANGTTEHTGDGHWKAATTPLISTYLVAVAAGPWHSVRTEHRGLPFGIHCRRSLAPHLDTDADELFEITRACFDRYHEKFTEPYPFDSYDQAFVPEFNAGAMENPGLVTFRDEFVFRSAVTDTQRQTRAMVIAHEMAHMWFGDLVTLRWWDDIWLNESFAEYMGYQTTAEATRFADTWTDFGVSRKAWGYDADQRPSTHPVAPEHVEDTASALLNFDGISYAKGASALRQLVHWLGEKDFLAGINIHFERHKYANASLADFIDSLAAATDRDVHAWADAWLRTTGVDTLTPRVTGDNGGRALEVGRKGERPHRVAVGLYDRDLNDEGRLTLRERLDLDLPQDDPRPIGKLPALVVLNDGDLSYAKVRFDAESFRTIREGLSGLPDPLTRAVVWNALRDAVRDGELPARAYLDIARAHLPRETDLALVDGVLAFAAGQVADRYVAPEQRPAALTTLAELCRDLIRRTEDGDHPGLRLIAVRHRIATAAHPDTIAAWLADGTVPGGPELDPELRWRILTRLAVLGATDEAAIAAELERDPSATGQEGAARCRAALPDAEAKSRAWEAMFATDDLSNYLFTAMAQGFWQPEQADLVREYVPRYYAEAVAVAARRGPAIADAAGRWAFPGHAVDADTLRLGEQCLADAEPLPALRRKLTDQLDDLARALRVREAGAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01113 Aminopeptidase N MPGTNLTREEARQRATLLTVDSYEIDLDLTGAQEGGTYRSVTTVRFEVAETGGESFIDLVAPAVHEVTLNGDALDPGEVFQDSRIALAELLPGRNILRVVADCAYTNTGEGLHRFVDPVDDQAYLYTQFEVPDARRVFASFEQPDLKATFQFTVKAPEGWTVISNSPTPEPRENVWVFEPTPRISSYVTALIVGPYHSVHSVYEKNGQSVPLGIYCRPSLAEHLDSDAIFAVTRQGFDWFQEKFDYAYPFKKYDQLFVPEFNAGAMENAGAVTIRDQYVFRSKVTDAAYEVRAATILHELAHMWFGDLVTMEWWNDLWLNESFATYAEAACQAAAPGSKWPHSWTTFANQMKTWAYRQDQLPSTHPIMADISDLDDVLVNFDGITYAKGASVLKQLVAYVGEDAFFQGVQAYFKRHAFGNTRLSDLLGALEETSGRDLKTWSKAWLETAGINVLRPEIETDADGVITSFAIRQEAPALPAGAKGEPTLRPHRIAIGGYDLDADGKLVRGDRVELDVDGELTAVPQLVGKVRPAVLLLNDDDLSYAKVRLDEQSLAVVTEHLGDFAESLPRALCWASAWDMTRDAELATRDYLSLVLSGIGKESDIGVVQSLHRQVKLAVDQYAAPTSREALLTRWTEATLAHLRAAEAGSDHQLAWARAFAATARTPEQLDLLDALLDGTQTIEGLAVDTELRWTFVQRLAAVGRFGGSEIAAEYERDRTAAGERHAATARAARPTEAAKAEAWESVVDSDKLPNAVQEAVIAGFVQTDQRELLAGYTERYFEALKGVWESRSHEMAQQIAVGLYPALQVSRETLDRTDAWLASAGPTAALRRLVSESRAGIERALQAQAADEAAGA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01118 Aminopeptidase N MRTPRLLASAAALTALAACGGDGAVGGGPGGPGAGDPYFPEAGNGGYDVGHYDLKLDYDPGTGRLAGLATITARATRDLSAFNLDLKGLNVEKVAVGGRDARSHRAGQELTVRPADALDAGETFRVTVRYSGRPVTVTDPDASEEGWLRTADGAVGLGQPTGSMAWFPGSHHPSDKAAYDLAVTVPEGLGAVSVGELRGERTRAGRTTFTWHAAEPVSSHVVTVAVGRWETDRSRTGDGLPVYTAVDPQQADASREVLARIPEIMDWARKNFGPYPFSSTGAIVDRAGDAGYALETQNRPYFPGAPDTVLLVHELTHQWFGNSVSPKTWRDMWLNEGFATYAEWLWQEDHGGDSAQQTFDALYDGTYYPDEAANDAVWSFPPADPPDAAHISASPVYQRGAMVLHQIRRAVGDDAFRALLRGWAAAHRHGNADTADFTAYVEKSAPDEDFTEIWRTWLHGEGRPRRS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01123 Aminopeptidase N MLHTPHLPAPRPRAHSRRRLRAAALLASAVSVCLVAASAPPTPLGVGDRLYPHLGNPGYDVAAYDLAFTYSGSNSEPLEAVTTIDARATADLDRINLDFAHGKVDSVEVDGEPADFAPAGADLVVTPQDALDEGERMRITVRHSSDPVYAEDRPGGWVRTTDGLAMANQADVAHLVFPCNDHPSDKARFTFHVTAPDGLTAVANGLPTGVERAGGSTTWTYRTQHPMATELAQVSIGRSTVLHRTGPHGLPVRDVVPTEHRAALEPWLEKTPEQIAWMEKKAGRYPFETYGLLMADATTGFELETQTLTLFERELFTEPAYPKWYVESIMVHELAHQWFGNSVTPATWSDLWLNEGHATWYEALYAEETADRPMAERMKAAYGASDRWREAGGPPAAPKPPKSGSKTGIFRANVYDGSALVLYALRQEIGRTAFEGLERAWTATHRDGTATTADFVRLASETAGRDLGGFFQAWLYGEKTPPMPGHPDWKPVAEKEPVKASRKPQGE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01128 Aminopeptidase N MPLRLGAFVHRRFIVPGALGAATLMLAIPASAAAHSPGAPGIGDPYYPAYGNGGYDVSHYDLRLKYQPDTDRLEGTATILARTTEDLSRFDLDFLLDVGEVRVNGAKASFTTSGEQELEITPAKPLDKDTPLTVVVRYSGVPSSKQAFGFTSWHRTPDGGIAANEPEAAAWWFPSNDHPLDKATYDVSVQVPDGTQAISNGTLQSTSSRLGWTRWNWRSAQPQATYLATLAIGRFDLTTGTTEGGIPVVNAYSEDLGPNGGAARASVERTGEVADWLSGYFGPYPYDALGGYVPNTDTGFALETQTRPFYSPRQFANGSNVSVVVHELAHQWYGDLVSLRGWKDIWINEGFARYAQWLWSEHEGEGTAQELADYTYASYPADDPFWTVKPGDPGPENQFDTAVYDRGALAVQALRNEIGDDAFFTVLKGWPAKYAHGNASVADFQRYAEEVSGKPLAALFDTWLFQPSKPDAAAARAQSLAKPAGTPAQPRSWRKIAATNDVHDHDHGHRH Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01133 Aminopeptidase N MSRDEARERAALLSVDGYEVSLDVRSALGEARGEAPDEAQGGGPRTFRSVTTIRFRCNEPGASSFADLIAPSVTAVSLNGRDLDPSEVFDGSRIALEDLAAENELIVDAQCAYSRTGEGLHRFVDPEDGEVYLYTQYEPADSRRVFANFEQPDLKAPFRFEVRAPEEWTVWSNGAGERADGVWRFAETKPISTYITCVVAGPYHYVTDTYERTFEDGTRLEIPLGALCRKGLAPHFDAGDVFLITKQGLDFFHDRFDYPYPFGKYDQAFVPEYNLGAMENPGLVTFREEYIFRGKVTRASYEGRANTILHEMAHMWFGDLVTMEWWDDLWLKESFADFMGAFANVGATRFKDAWITFANRRKAWAYRADQLPSTHPITADIRDLEDAKLNFDGITYAKGASVLKQLVAYAGQDAFLEGARRYFKRHAYGNTRLGDLLSVLEETSGRDMTAWARSWLQTAGVNSLTPQVLLSTAGTVDELAVVQEAVESHPELRPHRVAVGLYRRTAEGALERYARAEVDVEGPRTVVAELAGAEAPELVLVNDDDLTYCKTRFDATSLATLREHLGALTDPLARALCWSALWnMTRDALLPARDFAALVLRFAGRESDIGVLQMLHAWAGSALVHYAAPDWRETGGRLLGEGAVRELRDAAPGGEQQLAWARFLASVASGEEELSLLRGLLDGTEKIDGLAVDQELRWAFLAPLAAHGAADEGVLAAELARDDTASGKRHQVRCLASRPSAEVKARAWAQVVESDALSNALVEATIAGFAQASQRELLAPYAERYFAVIERVWAERSIQIGMDVVRGLFPSLRDSPETLDATDAWLSAHEDAAPALRRLVLEARDDLARALRGQACDAAAAAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01138 AMP-ligase MADLHARLEQLASDRPHDTALVLGRRDGSGRAITFARLVAGCREAADAFERAGVRRGHKAVTMTGDPYHLFTTVHGLLAVGAVPVLVDPGLPRADLRQCLDEVAPEVFVGQPLAHLGRTALGWARGHVRTAVVTGAAVPGLRRRLPVPGARRGWAPAGPPPVRDPLPPTPDDGLALIAFTSGSTGVPKGAEYHHSTLLGQAETLARLVGTDGTLFAGFLPVVLLGPVLGHTTVAPAVNHRAPARTPSARLVRPLLENRTEVVVGSPAVLGLLAEHCARRRLVLSCVDRVISFGAPLRAGLADALHAVLRPDAEVLSAYGATECLPVSAVSTTDACAPGAGTCVGRPLGGVAARILDAGPDGVGEIAVTGANVSPAYHARPEITAATKTATDRGVQHRTGDMGLIDGEGRIWFHGRRSHRVIGTDYVLTTEDVEAAADTLPGVRRTALVGVGAPGRQRAVLCVELTARGPGRGAAVTAVRELLDRRPEGRHVAAVLVHPGFPTDIRHNSKINRDRLADWATRRLRRPR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp01146 Ansalvamide A NA Marine fungus, Wilt of banana Apoptosis inducing Not specified HCT-116 Colon cancer IC50 : 9.8 µg/mL
dbacp01184 Apo E LRVRLASHLRKLRKRLLRDADDLQKRLAVY Apoprotein E Cell membrane disintegration MTT/MTS assay COLO-201 Colon cancer 65 % Cytotoxity at 40 µg/ml
dbacp01202 ATP-binding cassette domain-containing protein MPESATTATPGPAAEGPREDTPLLEVRGVTKAFGSGRRRLTALDGVDIEVGRGTTLGLVGESGCGKSTLARVLLGLERPDAGTVRFDGTDPFALRGKELLAWRRRVQMVFQDPFASLNARMSAADLIGEPWRTHRDVVPGAGAREKRIRELLDLVGLRAGDAHRYPNEFSGGQRQRIGIARALALDPDLVVCDEPVSALDLSVQAQVLNVLSDLRTRLGVTYVFISHDLSVVRHISDRVTVMYLGKVVEHGATDEVFETPRHPYTAALMSAAPALHPGGGSRREEIQLRGEVPSPFDIPSGCRFRTRCPRAEERCASEAPPVAARGTADGGEPHTALCHFPLAAGSSWA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp01207 ATP-binding cassette domain-containing protein MVPVLAADGAAVELADTTLLAPTTFEVGPGERWCVTGGNGTGKTTLLRAFAGTRSLTAGSVSVRGEPVAMTDPRHRRLMASLVEPVPVARDMTLREQVALVAASWYGNSTAAAEGTGRVVERLGLSALGERFPHQVSSGQSQLFSLALTLVRPADVVLLDEPERHLDRHRVDLVAGLLAERAEAGTAFLVATHDPALVAACDGRVELG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp01221 ATP-binding protein MGVVVLAMLGSLAVLAVAGPLWWGHAADRPDPSAVLQGPTGRHPLGTDHLGRDLLARLLASTWPSLLPAVAATLLGAAAGITLGALTAVVGGRVRRLLGAFVNLLLAFPALLIAMFFAALFGAGARGAVFALAVACAPGFARLTQTLAAGVAGTDFMAAARVLGLRRHRLLLRHVLPHVAEPLLLNVTVAVGSALVALSGLSFLGLGAQSPSYDWGLLLSQGLERVYTEPLPAVAPGIAIVYAGVAFQLLGEVLAKTATRHAVPRHAEEPAPPPAPAGRRPASPDHVLEVEDLRVALPAGDRTIRPVRGVSLALRRGEMVGLVGESGSGKSLTALALADLLPDGARATWNAHWFLGADVGSLTRGERHRQLATGMAMVFQNPASAFNPALRIETQLTEAVRAHHGTPRDQAVEQALVQLRRVALPGERRLLRSRPFQLSGGQRQRVAIAAASMLRPDLVIADEPTTALDVTVQRQIMDLLRRLRRDDATAILFISHDIALVADTCDRVLVMYGGTIVESLPARRLADGARHPYTRMLVASVLDLTADRDGTPPTVEGPPPDAAGTDPGCPFLDRCPQRLDRCAVEGPVPTLLAPGHEVACWRPLPLAAPPGQPETEEAET Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01229 ATP-grasp ribosomal peptide maturase MTVLILTSEEDVTADMVVVHLNASSVPVVRLDPADLTESVALSGEFVHGSFRGHLSAGERLVSIGGLRSVWLRRPGGPAARAAEPSAWLTEESGQALYGMLRGSGARWMNQPDAAHRARYKPWQLRLAQQCGLPVPATLITTFPRAAREFAERYPDLVVKPVSGAHPQDPPLAVPTSRVPPEADFSAVAHGPTLLQRRVAKRADIRLTAVGDELLAARKATAHPDPDEVDVRFAASAEPWRPVEVPPRVAESVRSYLRAAELAYGALDFAEDGDGTWWFLECNQSGQFGFVEVDTGQPIARTIAEWLARPGPGDPMPSGPPGATAVG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01234 ATP-grasp ribosomal peptide maturase MDDPTTDLVIDELHGRGVPVVRFDSGDFPATLSIAATLTSNGIGGTLTTPTRTADLSRVRSLYYRRPSGFAFPHLDDQTARFAVTQARYGIGGVLASLPGCRYVNHPHRIGDAEFKPSGLAVAAACGFRLPPTVITSDPDTARAFVKAHGPVLYKPLSTPLYRIDGVSCTVEVREATADEIDDSVTGTVHLFQQRIDKTGDVRVTVMGDHVFCVRIDSDLLDWRTDYARLRYGVVQPPPGVLESLHAYLDHFRLVFGAFDFAVDRRGRWWFLECNPSGQWAWLEPETGLPMVAAMADLLERKTT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp01254 Aurein 3.1 GLFDIVKKIAGHIAGSI Southern bell frog, Australia Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10 µM
dbacp01263 Aurein 3.1 GLFDIVKKIAGHIAGSI Southern bell frog, Australia Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10 µM
dbacp01273 Aurein 3.2 GLFDIVKKIAGHIASSI Southern bell frog, Australia Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10-100 µM
dbacp01283 Aurein 3.3 GLFDIVKKIAGHIVSSI Southern bell frog, Australia Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10 µM
dbacp01294 Aurein-1.3 GLFDIIKKIAESF Southern bell frog Cell membrane disintegration One-dose and five-dose assay HCT-15 Colon cancer IC50 : 4-5 μM
dbacp01313 Aurein-2.5 MAFLKKSLFLVLFLGLVSLSICEKEKRQNEEDEDENEAANHEEGSEEKRGLFDIVKKVVGAFGSLGKRNDLE Green and golden bell frog Not specified Not specified Not found Colon cancer Not found
dbacp01322 Aurein-2.5 GLFDIVKKVVGAFGSL Green and golden bell frog Not specified Not specified Not found Colon cancer Not found
dbacp01331 Aurein-2.5 GLFDIVKKVVGAFGSL Green and golden bell frog Cell membrane disintegration One-dose and five-dose assay HCT-116 Colon cancer IC50 : 4-5 μM
dbacp01340 Aurein-2.5 MAFLKKSLFLVLFLGLVSLSICEKEKRQNEEDEDENEAANHEEGSEEKRGLFDIVKKVVGAFGSLGKRNDLE Green and golden bell frog Membrane disruption Not specified Human tumour cell lines Colon cancer LC50 : 10-5 - 10-4 M
dbacp01349 Aurein-2.7 GLFDIAKKVIGVIGSL Southern bell frog Cell membrane disintegration One-dose and five-dose assay HT29 Colon cancer IC50 : 4-5 μM
dbacp01360 Aurein-3.1 [Cleaved into: Aurein-3.1.1; Aurein-3.1.2] GLFDIVKKIAGHIAGSI Southern bell frog Cell membrane disintegration One-dose and five-dose assay COLO 205 Colon cancer IC50 : 4-5 μM
dbacp01373 Aurein-3.2 GLFDIVKKIAGHIASSI Southern bell frog Cell membrane disintegration One-dose and five-dose assay HCC-2998 Colon cancer IC50 : 4-5 μM
dbacp01385 Aurein-3.3 [Cleaved into: Aurein-3.3.1] GLFDIVKKIAGHIVSSI Southern bell frog Cell membrane disintegration One-dose and five-dose assay KM12 Colon cancer IC50 : 4 - 5 μM
dbacp01408 Aurein1.2 GLFDIIKKIAESF Southern bell frog Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10 µM
dbacp01417 Aurein2.5 GLFDIVKKVVGAFGSL Southern bell frog Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10-100 µM
dbacp01426 Aurein2.6 GLFDIAKKVIGVIGSL Southern bell frog Cell membrane disruption Not specified Colon tumor cell line Colon cancer LC50 : 10-100 µM
dbacp01596 BF-30 KFFRKLKKSVKKRAKEFFKKPRVIGVSIPF Banded krait Cytoplasmic membrane permeabilization and DNAspecified-binding Lactate dehydrogenase release assay, DNA retardation assay, Real-time PCR, Western blot, wound healing assay, and chick embryo chorioallantoic membrane assay B16F10 Human Colon cancer IC50 : 7.3 μM
dbacp02039 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay COLO-205 Colon cancer IC50 : 11.2 µg/ml
dbacp02040 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay HCT-116 Colon cancer IC50 : 14.6 µg/ml
dbacp02041 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay HCT-15 Colon cancer IC50 : 13.2 µg/ml
dbacp02042 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay HT-29 Colon cancer IC50 : 17.6 µg/ml
dbacp02043 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay KM12 Colon cancer IC50 : 12 µg/ml
dbacp02044 Buforin IIb RAGLQFPVGRLLRRLLRRLLR Histone H2A Inducing mitochondria-dependent apoptosis MTT/MTS assay SW-620 Colon cancer IC50 : 12.7 µg/ml
dbacp02300 Carrier domain-containing protein MTRPGPAVRDGRPAPDAAGPATAPATYAQERAWLASRLAHDPPTYCAVDEFPLHAAVTANDLVHALYVLMDRHEPLRTVLRTVDGRLRQEVHPRPEPRIELTDLRAHDHAAQAEERRSLRARLARTPFDPHRAPQWRAAVLNLGEGAWSVVFAAHHTVYDTASGFNVHAELTELCAAAEEGREARLPRLPLGYGAYARRERERARTGGADAAAAHWRTRLRGLPPVHTVPLDRPRPPARTFRGAEVRAALPVGVTAALTGAARHHGTRPVMLFLAAWTALLHHHSGAADLAVGLPVAGRDDPATRAMVGTFVnMRVLRADLSGDPDGTELVRRTTAAVRAGEKFDIPFQSLVELLAAPRLPGVPPLYQLAFNHTPADGLGPPVSSCEEDLLLDVAGSGLRLVYDAALFDRSTADLLLADYLRLLAALLDAPGTRLSALLTGPAPRGTPRPAPTAPRARTAPRDAAEERVAAVWRTLLGTDGGTVDVHEDFFTAGGHSLQALRLLARLAPARGSGPTLRTFFADPTVAGLATALKSTPDGRTAWR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02305 Caseinphosphopeptides PPPEE Bovine milk Regulation of immune response; Apoptosis inducing MTT/MTS assay AZ-97 Colon cancer Inhibition at 24-28g/l
dbacp02359 Cecropin B KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL Silkmoth Pore formation at the cytoplasmic membrane MTT/MTS assay HRT-18 Colon cancer IC50 : 25.5 µM
dbacp02360 Cecropin B KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL Silkmoth Pore formation at the cytoplasmic membrane MTT/MTS assay DLD-1 Colon cancer IC50 : >100 µM
dbacp02363 Cecropin B KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL Silkmoth Pore formation at the cytoplasmic membrane MTT/MTS assay HCLO Colon cancer IC50 : 33.5 µM
dbacp02365 Cecropin B KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL Silkmoth Pore formation at the cytoplasmic membrane MTT/MTS assay MAC15A Colon cancer IC50 : 37 µM
dbacp02367 Cecropin B KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL Silkmoth Pore formation at the cytoplasmic membrane MTT/MTS assay HT-29 Colon cancer IC50 : >100 µM
dbacp02373 Cecropin P1 SWLSKTAKKLENSAKKRISEGIAIAIQGGPR Small Intestine of Pig Pore formation at the cytoplasmic membrane MTT/MTS assay HRT-18 Colon cancer IC50 : >100 µM
dbacp02374 Cecropin P1 SWLSKTAKKLENSAKKRISEGIAIAIQGGPR Small Intestine of Pig Pore formation at the cytoplasmic membrane MTT/MTS assay DLD-1 Colon cancer IC50 : >100 µM
dbacp02444 Chaperone protein DnaJ MATDYYAVLGVRRDASQDEIKKAFRRLARELHPDVNPDPKTQERFKEINAAYEVLSDPQKKQVYDLGGDPLSQAAGGGAGGFGAGGFGNFSDIMDAFFGTASQRGPRSRTRRGQDAMIRIEVELDEAAFGTTKDIQVDTAVVCNTCNGEGAAPGTSAQTCDMCRGRGEVSQVTRSFLGQVMTSRPCPQCQGFGTVVPTPCPECAGDGRIRSRRTLTVKIPAGVDNGTRIQLAGEGEVGPGGGPAGDLYVEIHELPHSTFQRRGDDLHCTVTIPMTAAALGTKVPLETLDGLEEVDIRPGTQSGQSIPKPGRGITHLRGGGRGDLIVHVEVTTPTKLDPEQERLLRELAQQRGEERPTGQFQPGQQGLFSRLKDAFNGR Beras-beras Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02449 Chaperone protein DnaJ MSTKDFIEKDYYKVLGVPKDATEAEIKKAYRKLARENHPDANKGNARAEERFKEISEANDILGDPKKRKEYDEARSLFGNGGFRPGPGAGGGGGTFNFDLGDLFGGGPQGGGGQGGAGGFGGGLGDVFGGLFNRTGGPGTGTGPRTQPRRGQDIESEVTLSFTEAIEGATVPLRMSSQAPCKACSGTGDKNGTPRVCPTCVGTGQVARGSGGGFSLTDPCPDCKGRGLIAEDPCDVCKGSGRAKSSRTMQVRIPAGVSDGQRIRLRGKGTPGERGGPAGDLYVVVHVKDHPVFGRRGDNLTVTVPVTYTEAALGGEIRVPTLGGPPVTLKLPAGTPNGRTLRARGKGAVRKDGTRGDLLVTVEVSVPKDLTGKARDALEAYREATADEDPRAELFQAAKGA Beras-beras Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02454 Chaperone protein DnaK MARAVGIDLGTTNSVVSVLEGGEPTVITNAEGARTTPSVVAFAKNGEVLVGEVAKRQAVTNVDRTIRSVKRHMGTDWSVNLDGKDFNPQQISAFVLQKLKRDAESYLGEKVADAVITVPAYFNDAERQATKEAGEIAGLNVLRIVNEPTAAALAYGLDKDEQVILVFDLGGGTFDVSLLEIGDGVVEVKATNGDNNLGGDDWDQRVVDYLVKQFQSGHGVDLGKDKMALQRLREAAEKAKIELSSSTETNINLPYITASAEGPLHLDEKLTRAQFQQLTADLLERCKTPFHNVIKDAGIQLSEIDHVVLVGGSTRMPAVAELVKDLTGGKDANKGVNPDEVVAIGAALQAGVLKGEVKDVLLLDVTPLSLGIETKGGIMTKLIERNTTIPTKRSEIFTTAEDNQPSVQIQVYQGEREIAAYNKKLGMFELTGLPPAPRGVPQIEVAFDIDANGIMHVTAKDLGTGKEQKMTVTGGSSLPKDEVDRMRQEAEKYAEEDHARREAAESRNQGEQLVYQTEKFLKDNEDKVPGEIKTEVEESVAELKEKLKGEDTAEIRTATEKVAAVSQKLGQAMYADAQAAGGEAPGAGAGAGAAAGDKADDDVVDAEIVDDERKDGAA Beras-beras Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02490 Citropin 1.1 GLFDVIKKVASVIGGL Amphibian skin secretions Penetration and disruption of the membranes Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp02501 Citropin 1.1D glfdvikkvasviggl Amphibian skin secretions Penetration and disruption of the membranes Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : 5 M
dbacp02537 CoA ligase MEPAPQAPTQPVIDARRPEAGPRWETIGELIKDAALLHGDKEFLRCGDKTLSFSETDTRTDRLAQALIAQGVKPGDRVAVMMDNVADWPLSWFAAIKAGAITVPVNTRFGATDLAHVLKDSQAVLVLASPGCVPLARDVSGSIGNPCAVRTLRELEAGFGDRPVDGPGLSAHADDTVNFQYTSGTTGFPKACMLSHDYWLRTAWMIAVHSGLRPDDVVLTAQAFSYMDPQWKAVMCLMGGVPLVVLPRFSASGFWHSVRQHRATLTYVLGSMPMLLYKQPPHSGDRDHAMRLVLCSGIPRDLHHAFEDRWGAAWREVYGSTESGLDLIMPPGEEATVGSGAMGYPPSGKEVLVADERQRPVQPGQIGEILVRGRPMMKGYWNNPDSTERAFRGGWYHTGDLGRAEAAGSVVHAGRLKDMIRRGGENIAAAEVESVLEAHPAVLAAALAGIPDELFGELPKAFLQLRPGYRPTTATARSVLAHTRRHLAKFKVPAYVEFVDSFPMTPSARIQKRQLLRPGDDQRTGAFDAAADAWA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp02568 Creatininase family protein MKTKGRAGMDASLVPADTSADVRERGSGVSRQVAVLPVGSYEQHGDHLPLATDTLVACAVAREIAAGYPVHLLPPVTIGCSHEHADWPGTVSISAVTLHAVVRDIAESLRRSGVGALVVVNGHGGNYVLGNVVQEASARGERMALFPAGEDWEAARQRAGVRTSLLTDMHAGEIETSILLHAHPASVRPGYETADFVADDRRHLLSLGMSAYTDSGVIGRPSLASAEKGKELLASLADSFGTYFSFLTAADGAEGTSAQGARGRS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02596 Cyclic [W(RW)4 ]-Dox WRWRWRWRW Not found Inhibition of the cell proliferation MTT/MTS assay HCT-116 Colon cancer 50-67% inhibition of cell proliferation at 1 µM
dbacp02603 Cysteine hydrolase MGKTALIVIDMINTYDHEDADSLIPSVESVLPRATGLLERARRRGVPVIYVNDNFGEWRSHHGEILDKALSGPHSRLVEPLRPDDSSLFVVKARHSVFFETPLTYLLHQQGIDRLVLCGQVTEQCVLYSALDAHIRHLQVIVPRDAVAHIHADLADAALRMMERnMGARVCDSGELWT Not found Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02614 D-aminoacylase MEELVIRDADVVDGSGADSYRADVVVDGGRIVSIVKEAAAAGCQRPKARRELDAEGLVLAPGFIDMHAHSDLALLRDPDHSAKAAQGVTLEVVGQDGLSYAPVDDRTLGEVRRAIAGWNGPGDDVDFDWRSVGEYLDRLDRGIAVNAAYLIPQGTVRALAVGWDDREATPAELERMRRLVAEGMEQGAVGMSSGLTYTPGMYAKDAELTELCRVVAEYGGYYCPHHRSYGAGALEAYEEMVELTREAGCPLHLAHATMNFGVNRGRAPELLTLLDEALDGGADITLDTYPYTPGCTTLAALLPSWASEGGPEQILKRLADDDTAERIRHHMEELGSDGSHGVPMEWETIEISGTGDPALGEYVGRTVQESARLRGESPWTVVRQLLLADRLAPTILQHVGHEENVRAIMRHRVHTGGSDGILQGAKPHPRAYGTFPHYLGHYVRELGVLPLEECVAHLTSRPAARLRLPDRGLVREGYRADLVLFDRATVAAGSTYEEPRRLPTGIPYVLVDGRFVMEEGRRTDVLAGRSVRRGSR Not found Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02746 DI LTFEHYWAQLTS E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.29 µM
dbacp02747 DI LTFEHYWAQLTS E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 1.6 µM
dbacp02753 Diacylglycerol O-acyltransferase MHAPHLGTDGGPPTPVPMGTADLAYHLAMRGEPLPAGFLFAFSGPVPTLASVRARVAERAHRIPALRYRIDREGRAFSRVEGIDVERHVHEAWLPGDDDGSGAGRLMLSHPPGGDDRPPWDVWLVHGPGGEHSLCYRTDHTLQDGIGAAHTARALLDDDPVGGPPGYHGGRPTARGLASAAGALAASFRHSDKPAFDVPLSGRTGLCQTVVPVARLRAVGRAHGATVNDVFLAALAHAVGTWHRKNTGAAHPPLPVAVPMSVRAPGEECVPGNRIVVARVLLPCDAPSPRHALSRVVARSDGMRTGRLRESLRLMQTAGPRGIGARVGTRVVNGRAVAGPVSSVNFGTALVHRGNAAHRSVVWSGLGAGIRCLVTLTSQHDTACLAVIHDEALTTADELPDLWLASLLDLEQP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02762 Dipeptide ABC transporter ATP-binding protein MSDNTKTTTAVADTFPQQRDGDTAPLLKVSGLSKYFPIKGGFPIKRTVGHVKAVDGVDFEVFPGESLGLVGESGCGKSTTGRLLTRLYEPTQGTIEYRGKDITRANRRELAPIRSEIQMIFQDPYASLNPRQTVGTIISGPMEINGINPPGGREKRVRELLEIVGLNPEHYNRFPHEFSGGQRQRIGVARAVALQPKLIVADEPVSALDVSIQAQVVNLLQEVQREMGIAFVFIAHDLAIVRHFSQRVAVMYLGKVVEIADRDSLYNRPRHPYTHALLSAVPEADLDAEKRERIRLEGDVPSPISPPSGCRFRTRCWKAQDKCATEEPPLVQISGNREGHLTACHFPEEGTTEARAEDVVMDPGLKALEANTDA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02767 Dipeptide ABC transporter ATP-binding protein MPETTEPLLEVRGLVKHYPLTSGILFKKQVGAVKAVDGVDFELARGETLGIVGESGCGKSTVAKMLVNLERPTAGEIRYRGEDITRLSGRALKSVRRNIQMVFQDPYTSLNPRMTVGDIIGEAYDIHPEVAPKGDRRGRVQDLLDVVGLNPEYINRYPHQFSGGQRQRIGIARGLALRPEIIVADEPVSALDVSVQAQVINLLARLQSEFDLSYIFIAHDLSIVRHISDRVGVMYLGRIVETGRDAEIYDHPTHPYTQALLSAVPVPDPQAREHRERIILAGDVPSPTNIPSGCRFRTRCWKARERCALEVPALAVPAEFRSVSGPAAHDSACHFAEEKQVVPPEEPGEGPHRPSGDRFGK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02772 Dipeptide ABC transporter ATP-binding protein MASGIPAQSDGTQEKSGGTATLTKDAAPGETLLKVTGLQKHFPIKKGLLQRQVGAVRAVDGIDFEVRSGETLGVVGESGCGKSTMGRLITRLLEPTAGTVEFQGKDITHLGVGGMRPMRRDVQMIFQDPYSSLNPRHTIGTIVSAPFKLQGVEPEGGVKKEVQRLLSVVGLNPEHYNRYPHEFSGGQRQRIGIARALALSPKLVVADEPVSALDVSIQAQVVNLLDDLQQELGLTYVIIAHDLSVVRHVSDRIAVMYLGKIMELADRDLLYKSPMHPYTKALMSAVPIPDPARRGAKSERILLKGDVPSPIAPPSGCRFHTRCWKATQVCTTTEPPLKELRPGQQVACHHPENFEDQAPQDVVLLSAAKEAAELVSEDALAQSAATSAAVAAEVAETDADADSGAGADADSGAGADVDSGAGTEEPPAQEK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02832 Elongation factor P MASTNDLKNGLVLKLEGGQLWSVVEFQHVKPGKGPAFVRTKLKNVLSGKTVDKTFNAGVKVETATVDKRDMQFSYMDGDYFVFMDMQTYDQLHIERKVVGDAAHFLIEGFEATVAQHEGEVLFVELPAAVELTIKETEPGVQGDRSTGGTKPAILETGHQISVPLFITTGEKIKVDTRTSDYLGRVNS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp02962 FK-16 FKRIVQRIKDFLRNLV Not found Inducing apoptosis MTT assay LoVo, HCT116 Colon cancer Not found
dbacp02964 Folate-binding protein MKSPLLSLPGAVPAEGVDEGVAAHYGDLFREQRALADGTGFVDLSHRGVVAVTGDDRLSWLHLLLTQHVSDLPAGEATEALVLSANGHIEHALYLVDDGTTVWAHVEPGTQEELIAYLESMKFFYRVEVADRTADTAVVHLPAGSITGVPEGVAVRETPYGRDVFLPREELEAFAAGAGPAAGLLAHEALRVEQHRPRLGFETDHRTIPHELGWIGTAVHLQKGCYRGQETVARVHNLGKPPRRLVFLHLDGSEVHLPPNGAEIRLADDGPDGRKIGFVTTSVRHHELGPVALALVKRNVPVDARLMAEDTAAAQETVVEP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp02974 GA-K3 FLGWLFKWAKK Undecapeptide analogues derived from Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 27.00 µM
dbacp02981 GA-K3 FLGWLFKWAKK Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 27.00 µM
dbacp02988 GA-K4 FLKWLFKWAKK Undecapeptide analogues derived from Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 14.80 µM
dbacp02995 GA-K4 FLKWLFKWAKK Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 14.8 µM
dbacp03002 GA-W3 FLGWLFKWAWK Undecapeptide analogues derived from Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 24.63 µM
dbacp03009 GA-W3 FLGWLFKWAWK Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 24.63 µM
dbacp03016 GA-W4 FLWWLFKWAWK Undecapeptide analogues derived from Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 14.80 µM
dbacp03023 GA-W4 FLWWLFKWAWK Brevinin-1EMa Cell membrane disruption MTT/MTS assay HCT-116 Colon cancer IC50 : 14.80 µM
dbacp03029 Gageostatin A ELLVDLL Bacillus subtilis Perturbation of the cell membrane Sulforhodamine B (SBR) assay HCT15 Colon cancer GI50 : 4.6–19.6 μg/mL
dbacp03047 Gamma-glutamyl-hercynylcysteine sulfoxide hydrolase MCRHLAYVGPAEPLGGLLVAPPHALYRQSWAPRHQRHGTVNADGFGVGWYAEGDPVPARYRRAGPIWADQSFADLARVVRAGALLAAVRDATLAGADAEAAAAPFAAGAWLFSHNGAVGGWPGSLAPVAAALPPEELLSLEARNDSALVWALVLSRLRAGDDEGRALAETVLEVAAAAPASRLNLLLSNGTTVTATTWGDTLWYLTRPGAGGTVVASEPYDDDPGWQQVPDRTLLTATRTDVLLTPLKDPGEPAPADAVATEKEPRT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03063 GlcNAc-PI de-N-acetylase MTDRPLTLMAVHAHPDDEATSTGGVLARYAAEGIRTVLVTCTDGGCGDGPGGVKPGDPGHDPAAVTAMRRQELEASCGALKISDLEMLDYADSGMMGWPSNEAPGAFWQTPVADAAARLAELMRHYRPDVVVTYDENGFYGHPDHIQAHRVTMAALELTDLSPKVYWTTMPHSGVRRFGEIMSEFQEGAPEPDPAEAAATAELGLPDDEVTTWVDATGFSGQKFDALAAHASQGENIFFLKMGREAFGELMGTETFLRVRDTTGAPLPENDLFAGLR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03069 Glutathione hydrolase proenzyme MRRPVARNLTVLAVSAAVVVSLGAAAPPTHPSGPAGPDRPAAPKAPVAVGYGGAVSSVDQDASAAGIEVLRKGGNAVDAAVATAAALGVTEPYSAGVGGGGYFVYYDARSRTVRTIDGRETAPLTAGEDLFTEDGEPLAFADAVSSGLAVGTPGTPATWQRALDRWGSRRLSSVLEPAERLARHGFTVDETFRSQTADNEERFRYFPDTAELFLPGGELPAVGSTFKNPDLARTYRELAREGVGALYHGALGKDIVDTVNAPPVDPDSGWNARPGDLSAKDLAAYEAKVQAPTRTSYRGLNVYSIAPSSSGGTTVGEALNILERTDLSEASKARYLHRFIEASRIAFADRGRWVGDPAFEDVPADELLSQRYADSRECLISDDAALTGPLAPGDPRHPAACAAGGTAAPTTYEGENTTHLTVADKWGNVVAYTLTIEQTGGSGITVPGRGFLLNNELTDFSFAPANPAVHDPNLPGPGKRPRSSIAPTIVLDRHHKPVVAVGSPGGATIITTVLQTLTGFVDRGLPLVDAIAAPRASQRNAAQTELEPGLYDSALRAELEALGHSFKENPEIGAATGVQRLPGGKWLAAAEKERRGGGSAMVVEPVRQR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03086 Glycoside hydrolase family 92 protein MQYRVRHRWGPAVVMTTAFALAVGSQGAAVALPNAPAKTDREFTSSFEDGDPAPDWVSTVDTGADGGKRSSGVDGGFSTGIPGNVTEHVTRVRASAENTNGGEVKENLADNEPGTKWLTFAPTGWVEFDLDAPTKIVKYALTSANDHSERDPRDWTLKGSADGESWQTLDTRSGETFGEPFTTKTYDLAEAAEFQHFRLEFTKNNGAGDALQLGDVQFSTGDAETPAPEDMLAFVDEGPTSSPTAKANAGFTGTHALRYAGRHTADGRAYSYNKVFDVDVKVDRRTELSYKIFPAMADRDLDYDATNVSVDLAFTDGTYLSDLEATDQHGFPLTPRGQGDAKILYVNQWNSVESGIGSVAAGKTVDRILVAYDSPKGPAKFRGWLDDVEIKRAEPERPEAHLSDYALTTRGTNSSGSFSRGNNFPATAVPHGFNFWTPVTNAGTTSWLYDYASGNNDDNLPTLQAFGASHEPSPWMGDRQTFQVMPSAASGTPDTSRDARELAFRHENETARPYYYGVRFENGLKAEMAPTDHAAMMRFTYPGDDASVIFDNVEDKGGLTLDKENGTFSGYSDVKSGGSAGATRLFVYGEFDSKVTGGEDTGGVKGHLRFDAGRDRAVTMRIATSLLGVDQAKDNLRQELPKRASFEKVKRDAQKQWDTILGKVEVEGATRDQLTTLYSSLYRLYLYPNSGHEKVDGKYKYASPFSKAVKENTPTETGAKVVDGKVYVNNGFWDTYRTTWPAYSFLTPSKAGELVDGFVQHYKDGGWTSRWSSPGYADLMTGTSSDVAFADAYVKGVDFDAKAAYDAALKNATVVPPSSGVGRKGMETSPFLGYTGTETHEGLSWALEGYLNDYGIAKMGEKLYKETGEKRYKDESAYFLNRAQDYVNLFDSKAGFFQGKDTKGNWRVDSEKYDPRVWGYDYTETNGWGYAFTAPQDSRGLANLYGGRDGLGDKLDEYLSTPETASPDLKGSYGGVIHEMTEARDVRMGMYGHSNQVAHHALYMYDAAGQPYKTQKNIREVLQRLYTGSEIGQGYHGDEDNGEQSAWFLFSSLGFYPLVMGSGEYAVGSPLFTKATVHLENGRKLVVKAPKNSTKNVYVQGLKVNGKRWTSTSLPHSLISKGGVLEFDMGAKPSSWGTGENAAPPSITKDDEVPTPRADAITGEGALFDNTSATDATVTSVDLPVADKGAKALQYTLTSSADHTGAPAGWKLQGSADGKTWRTLDRRSGESFAWDRQTRAFSVKSPGTYAKYRLVLDGEHTLSEVELLS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03091 Glycoside hydrolase family 92 protein MRAPRRLRLCVAGVVAASALLTAPAAQAVPTTDQHLTDLVNPFIGTENEGNTYPGAAVPFGMVQFSPDTGHSTGYDHSDTHIRGFSLVHLSGVGCGLGGDLPVLPTTGDVTETDYTKYAAPFSHDDEEASPGYYRVGLGSGVDAELTATERTGVQRYTFPSTDKANVLLNAGQSLHKNVSTKVEVLDSRTVRTAITGSGFCQDTKPYTVYTVTRFDRPFASYGTWDDGTVTAGAKSGGDGAYVRFDTTEDRTVEATTALSYVDARGAARNLRAEGGHSFDSVRRGAERTWEKRLDDVKVRGGDDTLRRTFYSSLYRSFLAPNVGSDVDGRYTGWDRKVHRAKGFTYYQNWSLWDTYRTQSQLLALLAPREARDMAVSVIKIDEESGWLPKWGYGTVETNIMTGDPVTPFLTNAYQQGLLHGWEERAYRALKKNADGVPPTDSPAVGREANREYLADGFAPYVKGRPHAKPGDSDYDHGASATLEYALSDAMLSRMARDLGHDRDAKRYAERAQSYRNVFDASTGFFRARDAEGAFTGPADPAQSEGFHEGTSWQYQWMVPQDLPGMIDLIGGTDAANERLDSFFAYDQLLADPAKTAREVWVNGPYDYYNADKYNPQNEPDLIAPYTYLSTGQPWKTTDVVHAALTLFTDTPTGMTGNDDLGTMSAWNVLSSIGIFPIQPGYDTWGLSTPVFDRVDLALDRRYYPRGALTITAPGTSDTDRYVQSARTDGAEYARTWLTTDALRSVRSLAFTVGPQPSGWGTSAEAVPPPLT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03096 Glycosyltransferase MASRTRRHGAARSARGGFRRRLPLRLLLPLLVLVALAAMLMLRGYVHSEILADHRVQPPAATDKVPEKILEGGPVIDVRGGRTEGLSVPDHRLVLTFDDGPDPTWTPRVLDVLKKHDAHAVFFVTGTMASRYPDLVKRMVDEGHEVGLHTFNHPDLSFQSTKRIDWELSQNQLAITGAAGVRTSLFRPPYSSFADAMDNKSWPVTEYIGSRGYITVVNNTDSEDWKKPGVREIIRRATPHGGKGAIVLMHDSGGDRHQTVQALDEFLPGLKEKGYEFDNLTEALEMPSAMSPVTGAELWKGKAWVFLVQASEKITDVLVVGLAVIGTLVIGRFGLMLLLSGVHARRVRRKRFSWGRTVTEPVTVLVPAYNEAKCIENTVRSLVASDHPVEVIVIDDGSTDGTARIVEGLGLPGVRVIRQLNAGKPAALNRGLANARHDIIVMMDGDTVFEPSTVRELVQPFGDPKVGAVAGNAKVGNKDSLIGAWQHIEYVMGFNLDRRMYDVLGCMPTIPGAVGAFRRSALEPIGGMSDDTLAEDTDVTMALHRAGWRVVYAENARAWTEAPETVQQLWSQRYRWSYGTMQAIWKHRRAVIEKGHSGRFGRVGLPFVSLFMVLAPLLAPLIDVFLLYGIVFGPTEKTVVAWLGVLAIQAVCAAYAFRLDRERMTHLISLPLQQILYRQLMYVVLLQSWITALTGGRLRWQKLRRTGVVEAPGGSVPRQRSRSSDDRRPVA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03101 Glycosyltransferase MTTPTTPTAPPSPPARGRRRGPSRIGRAASRAAALQRPRVLLALLLLLALTCVMLLDGYLRAEVGGDERVRTGASASDVPDDVLDGGPILTFPGGQATTVSVPDKTIVLTFDDGPDPTWTPQVLDILDEYDVPGTFFLVGSMISRHPGIVRDLVEQGNEVGVHTFTHVDLSYQSEARVTREIEQTQLALAGAAGITTTLFRAPYSSETNAIDDYSWPVYQNLGEDGYTSVFIDTDSDDWKRPGVSKIVEWATPEDDEGASVLFHDAGGERSQTIAALPKYIEKMKAKGYTFTTVSGAMADQQSPQQEADQQSQQQQQESQQPGGGRQPEQSGGGLQAAHHKATGATLYEGKALVAAVAVAEWTVPALSVGLVIVGVAVMGRFAMMLVLARRHHRQRNRRRFSWGPPVTGPVSVVVPAYNEKECIEATLRSLARSTHPVEIIVVDDGSTDGTAEIAESLGLPGVRVVRQANAGKPAALNNGVRHARYDIVVMMDGDTVFEPDTVRHLVQPFADPAVGAVAGNAKVGNRRTLIGAWQHIEYVMGFNLDRRMYDLLRCMPTIPGAIGAFRREAVLQAGGMSDDTLAEDTDITIALHRAGWRVVYEEHARAWTEAPGSLGQLWSQRYRWSYGTMQALWKHRRSLTDKGPSGRFGRVGMPLVVLFQVVTPVFAPLIDVFTVYSMVFVDFRAALLAWLAVLGVQLVCAAYAFRLDREKYRYLLMMPLQQLAYRQMMYLVLIHSCVTALTGGRLRWQKLKRTGEVGTPAGNG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03107 GNAT family N-acetyltransferase MVDVVLKLSVRDLVHADLASCGWAGSDHHLDGVAEQLVRARIGEVDYLAVCAATNIPVAKGGVDYQVKEGVGTLWQLAVHPALQSCGIGTFLVEAAELRIRRRGLRQAELGVEENNPRARALYERLGYVAYDRQPDAWDEQAPDGSLRRYETMCTLMRKELA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03112 GNAT family N-acetyltransferase MALADCERVSRIRVRGWQSAYAGLVPQPYLDAMDTAEDAERRRATFARAAEGVVNLVAEDDDGRVVGWAAHGPYRDGELRTADAELYALYVDTGRFGAGVGRALLGEAVRRCGAAGHPRMLLWVLRGNARARRFYERSGFLADGAEESFEVRGVAVPEVRYARPLPG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03117 GNAT family N-acetyltransferase MPGDLLLRSAGPADLDAVLAFWKAAAEGTSISDDREGVERLVARDPEALLLAEAGGDLVGTVIAGFDGWRCHLYRLAVHPDHRRRGIGSALLAAAEERFVRLGGRRGDAMVLRRNERAQHAWRAAGYAPEEQWRRWVKPLAE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03154 GPR15LG MRLLVLSSLLCILLLCFSIFSTEGKRRPAKAWSGRRTRLCCHRVPSPNSTNLKGHHVRLCKPCKLEPEPRLWVVPGALPQV Human Inducing G1 arrest Not specified Not found Colon cancer Not found
dbacp03190 HAL-1 GMWSKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 44 ± 8 µM
dbacp03193 HAL-1/10 GMWKKILGKLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 60 µM
dbacp03196 HAL-1/12 GKWSKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03199 HAL-1/15 GMWSKLLGHLLR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03202 HAL-1/17 KMWSKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03205 HAL-1/18 GMWSKILKHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 18 ± 2 µM
dbacp03208 HAL-1/19 GKWKKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03211 HAL-1/20 GKWSKILGKLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03214 HAL-1/21 GKWKKILGKLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03217 HAL-1/22 gmwskilghlir Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03220 HAL-1/29 GMWSKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp03223 HAL-1/4 GMWSKILGHLKR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp03226 HAL-1/5 GMWKKILGHLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 44 ± 5 µM
dbacp03229 HAL-1/6 GMWSKILGHLIK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03232 HAL-1/9 GMWSKILGKLIR Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 50 µM
dbacp03235 HAL-2 GKWMSLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 35 ± 3 µM
dbacp03238 HAL-2/1 GKWKSLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03241 HAL-2/11 GKWLSLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 40 µM
dbacp03244 HAL-2/13 GKWMTLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 60 µM
dbacp03247 HAL-2/18 GKWMSLLKHIWK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03250 HAL-2/19 GKWMSLLKHWLK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03253 HAL-2/2 GKWMKLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 35 ± 5 µM
dbacp03256 HAL-2/20 GKWMSLWKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03259 HAL-2/22 gkwmsllkhilk Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp03262 HAL-2/24 GKFMSLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03265 HAL-2/4 GKWMSLLKKILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 38 ± 6 µM
dbacp03268 HAL-2/6 GKWMSFLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03271 HAL-2/8 GKWMSLLKHILK Sweat bees and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp03345 Hydrolase MPDSQPQPPHSPSPSGPADPGSLLLCGARLTDGRTVDVRLCRGRIEAVGTAGSLSPPRAPGPGTRVDLAGYLLLPAPAEPHVHGDTALTADAPGPASYEPQDVEGRATEAALLQLGHGATALRAHVRVGDVAGLGALTAVLRARRTLRGLVEVTAVAMPRVLTGVAGADGLAVLRDAVKMGADVVGGCPDLDPDPAGYVEAVLEVAAEHGCPVDLHTDAGDPARLARLAAMAGGLRPGVALGPCDGLARLPAEMASRAAEQLSAAGVTVVCLPQGACGAVDHHDGMAPVRLLRAAGVRVAAGSGALRDVSNPVGRGDPLEAAYLLASRHGLRPEDAYAAVSSAARAALGLPEVRVEAGFPAELLAVRGDGLAGALSLAYSRVVVHRGRVVARTNAVREYGDATAGADLGLPRQGRGKRGRE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp03354 Hymenochirin-1B KLSPETKDNLKKVLKGAIKGAIVAKMV Zaire dwarf clawed frog Membrane disruption and cell lysis Cytotoxicity assay, Cell TiterGlo Luminescent Cell viability assay HT-29 Colon cancer LC50 : 9.7 ± 0.2 μM
dbacp03530 KW5 KAAKKAAKAAKKAAKAAKKAA Synthetic peptide Through interactions with the plasma membrane MTT/MTS assay HT-29 Colon cancer IC50 : 55 ± 14 µM
dbacp03535 L-amino oxidase (CP-LAAO) (LAO) (EC 1.4.3.2) MNVFFMFSLLFLAALGSCADDRNPLEECFRETDYEEFLEIARXXXXTSNPKHVVRVGAGMSGLSAAYVLAGAGHQVTVLEASERPGGRXXXXXXXXEGWYANLGPMRXXXXXXXXXXXXXKFGLNLNEFSQENDNAWYFIKXXXXXXXXXXDPGLLKYPVKPSEAGKSAGQLYEESLGKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXFDEIVDGMDKLPTSMYQAIXXXXXXXXXXXXXXXXXXKVTVTYQTPAKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXIFLTCTKKFWEDDGIHGGKSTTDLPSRXXXXXXXXXXXXXXVIIAYGIGDDANFFQALDFKDCADIVFNDLSLIHQLPKEEIPSFCYPSMIQKXXXXXXXXXXITTFFTPYQFQHFSEAXXXXXXXIYFAGEYTAQAHGWIDSTIK Mangrove pit viper Cytotoxic; Anti-proliferative; Apoptosis Not specified SW480 Colon cancer EC50 : 29.43 ± 0.48
dbacp03536 L-amino oxidase (CP-LAAO) (LAO) (EC 1.4.3.2) MNVFFMFSLLFLAALGSCADDRNPLEECFRETDYEEFLEIARXXXXTSNPKHVVRVGAGMSGLSAAYVLAGAGHQVTVLEASERPGGRXXXXXXXXEGWYANLGPMRXXXXXXXXXXXXXKFGLNLNEFSQENDNAWYFIKXXXXXXXXXXDPGLLKYPVKPSEAGKSAGQLYEESLGKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXFDEIVDGMDKLPTSMYQAIXXXXXXXXXXXXXXXXXXKVTVTYQTPAKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXIFLTCTKKFWEDDGIHGGKSTTDLPSRXXXXXXXXXXXXXXVIIAYGIGDDANFFQALDFKDCADIVFNDLSLIHQLPKEEIPSFCYPSMIQKXXXXXXXXXXITTFFTPYQFQHFSEAXXXXXXXIYFAGEYTAQAHGWIDSTIK Mangrove pit viper Cytotoxic; Anti-proliferative; Apoptosis Not specified SW620 Colon cancer EC50 : 23.19 ± 1.57
dbacp03537 L-amino oxidase (CP-LAAO) (LAO) (EC 1.4.3.2) MNVFFMFSLLFLAALGSCADDRNPLEECFRETDYEEFLEIARXXXXTSNPKHVVRVGAGMSGLSAAYVLAGAGHQVTVLEASERPGGRXXXXXXXXEGWYANLGPMRXXXXXXXXXXXXXKFGLNLNEFSQENDNAWYFIKXXXXXXXXXXDPGLLKYPVKPSEAGKSAGQLYEESLGKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXFDEIVDGMDKLPTSMYQAIXXXXXXXXXXXXXXXXXXKVTVTYQTPAKXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXIFLTCTKKFWEDDGIHGGKSTTDLPSRXXXXXXXXXXXXXXVIIAYGIGDDANFFQALDFKDCADIVFNDLSLIHQLPKEEIPSFCYPSMIQKXXXXXXXXXXITTFFTPYQFQHFSEAXXXXXXXIYFAGEYTAQAHGWIDSTIK Mangrove pit viper Cytotoxic; Anti-proliferative; Apoptosis Not specified CCD-18co Colon cancer EC50 : 15.99 ± 1.20
dbacp03551 L1 PEWFKCRRWQWRMKKLGA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : > 404 µM
dbacp03554 L10 PAARKAFRWAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 35 µM
dbacp03557 L11 PAARKAARWAWRMLKKGA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 248 µM
dbacp03560 L12 PAWRKAFRWAKRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 25 µM
dbacp03563 L13 PAWRKAFRKAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 29 µM
dbacp03566 L14 PAWRKARRWAWRMKKLAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 423 µM
dbacp03569 L15 PAWRKARRWARRMKKLAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 178 µM
dbacp03588 L2 PAWFKARRWAWRMKKLAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : >440 µM
dbacp03599 L3 PAWRKAFRWAWRMKKLAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 141 µM
dbacp03606 L4 PAWFKARRWAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 57 µM
dbacp03609 L5 PAWRKAFRWAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 14 µM
dbacp03612 L6 PAWRKAFRWAARMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 15 µM
dbacp03631 L7 PAWRKAFRAAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 16 µM
dbacp03634 L8 PAWAKAFRAAARMKLKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 180 µM
dbacp03637 L9 PAWRKAARWAWRMLKKAA Lactoferrin Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 52 µM
dbacp03648 Lan-7 fA*YwKA*T Analogue of TT-232 Tubulin depolymerization Sulforhodamine B assay HCT-116 Colon cancer IC50 : 29.97 ± 1.19 µM
dbacp03659 Lanthionine synthetase C family protein MTAPEATHVAVGEVEDVAADGLRWLLGAARETPGGGLAWPAGPSDDALHPMLYSGTAGTVPVLLEAWRHFGDDSYADAALRAARELAARVDDLDDDSLYFGRTGLALVLRTLQEELGDTAAGAAADRALALVRSRFDGTRWGSLFELMGGNAGIGLGALLTGDPELAVLALEPYLRTAERTANGVHWAHRPDTDARMHHLSHGTLGIAVALARVGAATGRTDLLDLGLTAVRDVVARDEAGPEGFLVRHSTPQFRPDVIDPVSYGWCHGPAGDAQVFRALRYVTSDPAWTALADRCWHTVTHSGLPRRLRPGFWDNNGRCCGTAGVLALACDRIAEQGDDQDTRDFAGVLVTDLVARAVRDADGARWSNFDHRSTPGDLEPQTGWAMGGAGIVRELLRFVRVARGGSPRYAFTWPDQPPVPA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp03671 Large ribosomal subunit protein uL2 MGIRKYKPTTPGRRGSSVADFVEVTRSTPEKSLVRPLHSKGGRNNAGRVTVRHQGGGHKRAYRVIDFRRHDKDGVPAKVAHIEYDPNRTARIALLHYADGEKRYILAPRNLQQGDRVENGPGADIKPGNNLALRNIPVGTTIHAIELRPGGGAKFARSAGASVQLLAKEGSMAHLRMPSGEIRLVDQRCRATVGEVGNAEQSNINWGKAGRKRWLGVRPTVRGVVMNPVDHPHGGGEGRTSGGRHPVSPWGQKEGRTRSPKKASNKYIVRRRKTNKKR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp03691 Lasso peptide biosynthesis B2 protein MRLESADPPPWPLRPPAVLAAAVARVLTRLPPARLRRVLTFASRGAGPASAAQALRARNAVVHVSLACAGPRCLQRSVAAALLCRLGGTWPQWCTGVVTEPFGAHAWVAVDGEPVGEADAHARAFHVIMSVPPRR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03696 Lasso peptide biosynthesis PqqD family chaperone MSFALKPGVSLADTEHGTVLLDERSGRYWMLNRTGAVVLRSLLDGESPQEAARTLLRRYPDAADGAGGHVESLLDALRTAKVIVP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03701 Lasso RiPP family leader peptide-containing protein MAKEDVYEVPALIEVGDFAELTQLTSQGYWIDSPWGAWWL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp03721 LFB GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC The Fujian Large Headed Frog Cell Apoptosis MTT assay H460 Colon cancer IC50 : 3.47 μM
dbacp03725 LFB GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC The Fujian Large Headed Frog, China, Asia Cell Apoptosis MTT assay H460 Colon cancer IC50 : 3.47 μM
dbacp03729 LfcinB FKCRRWQWRMKK Bovine milk Regulation of immune response; Apoptosis MTT/MTS assay AZ-97 Colon cancer Inhibition at 0.1g/l
dbacp03730 LfcinB FKCRRWQWRMKK Bovine lactoferrin (Lf-B) Cell membrane disintegration; Regulation of immune response; Apoptosis MTT/MTS assay HT-29 Colon cancer IC50 : > 160 µM
dbacp03734 LfcinB FKCRRWQWRMKK Bovine lactoferrin (Lf-B) Cell membrane disintegration; Regulation of immune response; Apoptosis MTT/MTS assay HT-29 Colon cancer IC50 : 148 ± 8 µM
dbacp04105 linear (RW)4-Dox RWRWRWRW Doxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPP Inhibition of the cell proliferation MTT/MTS assay HCT-116 Colon cancer 21-61% anti-proliferative activity at 1 µM
dbacp04108 Lipid II isoglutaminyl synthase MSDNQLRIVWIYPDLLSTYGDQGNALVVERRARQRGLDVARLDVRSDQPIPTSGDIYLIGGGEDRPQRLAAERLRRDGGLNRAVENGAIVFSVCAGYQILGHEFINDLGQREPGLGLLDVVSTRGEGDRCVGDVLGDIDPRLGLPPLTGFENHQGVTHVGPHARALAQVRFGNGNGTGDGTEGAYNDTVFGTYMHGPVLARNPQIADLLLKLALDVNALPPTDDRWYEALRSERIAAAQQPA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04113 Lipid II isoglutaminyl synthase MAGNSDPLTPRAKIAVTAGKAVARASRAAGRGSGSVIGGRVALKLDPDLLARLAGHLDVTLVSATNGKTTTTRLIAEALKAAGPVVSNALGAnMPAGITSALASGAEARYGVIEVDEKYLVGVAQATDPKCIALLNLSRDQLDRAAETRMLAENWREGLAGSKAVIVANADDPLVVWAASSSPNVIWVAAGQMWKDDAWSCPSCGGVMQRPGDDWFCGECGFRRPTPSWALSGDHVLDPHGSAWPIHLQLPGRANKANAASSAAVTAVFGVPPQVALERMYQVQAVAGRYDVVQFQGRDLRLLLAKNPAGWLETFSLIDPPPAPVILSVNARGADGTDTSWLWDVDYTRLTGHPICVVGDRKLDLAVRLEVANQQFQVCEDLDQAVQLCPPGRIEVIANYTAFQDLRRRVGN Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04118 Lipoprotein MHRRRRSALLLTAAIATAAPLLTACGNDAHPGAAAVVGDQRITVSQLENRVDEVREAQRAAVPDDGQYQQVVARSGALTRDTLHGMVLDRVLHSAAAEAHVSVSRKEVQAMRGDLEDQAGGAEQLETVWLQQYGVAPGRLDDNLRVQLEAQKLAESLGTDTSRPEFWQALSKASDKLDIDLNPRYGAWDVQKAGRVDSETPWVREVAEAEPSQQTA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04124 Lipoprotein signal peptidase MAEAERIIGTPDTPDAAGDGQELPDAEQEQAPERPRGRRRVAVLFVVAVFAYLLDLVSKMIVVAKLEHHEPIEIIGDWLRFAAIRNAGAAFGFGEAFTIIFTVIAAAVIVVIARLARKLYSVPWAIALGLLLGGALGNLTDRIFRAPGVFEGAVVDFIAPKHFAVFNLADSAIVCGGILIVLLSFRGLDPDGTVHKD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp04181 LL-III VNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 18 ±4 µM
dbacp04184 LL-III/1 VNWKKILAKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 12 ± 3 µM
dbacp04187 LL-III/10 KNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04190 LL-III/11 VNWKKIILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 48 µM
dbacp04193 LL-III/12 vnwkkilgkiikvvk Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 20 µM
dbacp04196 LL-III/15 VNFKKLLGKLLKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 42 µM
dbacp04199 LL-III/16 VN-NAl-KKLLGKLLKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04202 LL-III/17 VNWRRILGRIIRVVR Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04205 LL-III/18 KNWKKILKKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04208 LL-III/19 VNWKK-Aib-LGK-Aib-IK-Aib-VK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 28 µM
dbacp04211 LL-III/2 NVWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 11 µM
dbacp04214 LL-III/22 KNWKK-Aib-LKK-Aib-IK-Aib-VK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp04217 LL-III/23 VNWKKLLGKLLKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 15 µM
dbacp04220 LL-III/24 VNWOOILGOIIOVVO Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 20 µM
dbacp04223 LL-III/25 vnwkkllgkllkvvk Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 20 µM
dbacp04226 LL-III/26 VYWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 30 µM
dbacp04229 LL-III/27 VNWKKVLGKVVKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp04232 LL-III/3 VNWKKILKKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp04235 LL-III/34 NKWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 37 µM
dbacp04238 LL-III/36 VNWKKILAKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04240 LL-III/37 VNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 5 ± 1 µM
dbacp04241 LL-III/37 VNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 13 µM
dbacp04244 LL-III/4 VNWKKILGKIKKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 40 µM
dbacp04247 LL-III/6 VNWKKILPKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04250 LL-III/8 VNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04253 LL-III/9 VNWKKILGKIIKVVK Lasioglossin III and its analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 25 ± 5 µM
dbacp04258 Lon protease MAAESAAFTPLTLPVLPLDDEVVLPGMVVPLDLSDAEVRAAVEAAQAAARSEPGKPRVLLVPRIDGNHAATGVLGTVEQVGRLADGDPGALIRGRGRVRIGAGTTGPGAALWVEGTRVDETLPEPLPGQVSELVTEYKALATAWLRKRGAWQVVDRVQAIDDVSALADNSGYSPFLTTEQKVELLETTDPVARLKLATQQLRDHLAEQDVAETIAKDVQEGVDKQQREFLLRRQLEAVRKELREINGEQEGEESDDYRARVEAADLPEKVREAALKEVDKLERSSDQSPEGSWIRTWLDTVLEMPWSERTEDAYDIQGAQGVLDAEHAGLQDVKERITEYLAVRKRRGDRGLGVVGGRRGGAVLALVGPPGVGKTSLGESVAHAMGRKFVRVALGGVRDEAEIRGHRRTYVGALPGRIVRAIKEAGSMNPVVLLDEIDKVGSDFRGDPAAALLEVLDPAQNHTFRDHYLEVELDLSDVVFLATANVLEAIPEALLDRMELVRLDGYTEDEKVVIARDHLLPRQLERAGLDAGEVTVDESALRKLAGEYTREAGVRTLERSIARLLRKVAAQHELGERELPFTVTDADLRALIGRPHHVPESAQDPAERRTSVPGVATGLAVTGAGGDVLYVEASLADPETGAAGLTLTGQLGDVMKESAQIALSFLRSHGAELELPVGDLKDRGAHIHFPAGAVPKDGPSAGVTMTTALASLLSGRLVRTDVAMTGEVSLTGRVLPIGGVKQKLLAAHRAGITTVIIPKRNEPDLDDVPAEVLDRLDVHAVNDVRQVLELALAPATSGAQPEVPVAA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04263 Long-chain fatty acid--CoA ligase MTGPRYADKPWLDLLTDAQKAPLHPDDSLVHALRRAAAEAPDRALIAYFDGRLTYREVDRLSDSVAGHLTARGLERGDRVAVLLQNSPHFVLAVLGAWKAGAVVVPVNPMYKSGEVGHVLRDGEVAALVCSDRAWESYLRETAARSPVRIVLTACELDFQTRRDTRVLAFERLPRAAGTDDLAEVARAGHRAPEGRDPGPDDTALISYTSGTSGTPKGATNTHRNIMYNAERQRTGLLLPDAPVYFALAPLFHITGMVCEFGACLNSAGTLVLAYRFEAGVVLDAFAEHRPHYTVGPSTAFMALAAHPSVTREHFASFANISSGGAPLPPALVEKFRAGLGPYVRNGYGLTECTAPCASVPPHLEAPVDPASGTLAVGVPGPETVVRIVDDQGAEVPFGEQGEIVVSGPQVVPGYWRRPDATAETFPGGELRTGDIGFMDTQGWLYVVDRKKDMINASGFKVWPREVEDVLYTHPAVREAAVVGVPDGYRGETVKAYISLRPGADTDPDALAAYCGERLAAYKYPRQVEILPDLPKTASGKILRRELRSRTHQDTAVNGQ Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04268 Long-chain fatty acid--CoA ligase MATLSVAAVLAENARRRPDKEALVEGDLRLTFGEVWRRARAQAGALVGLGVRPGDRVALMAPNTADFPQAYYAIAAAGAVVVPVHLLLSAAEVEHVLRDSGATLLLCHPAQARTGAAAAREAGVRTLTLGEEFGGLAADAEPLTSYVTRDADDPAVVFYTSGTTGVPKGAVLSHFNLVMNATVNAFDANDIRPDDVALGALPLFHAFGQTVSLNSTWRAGATLVLLPRFDAGRAIELMVREKVNTFHGVPTMFVALAAAAADAGALPGLRVCVSGGASLPVAVLERFEEAFGARIYEGYGLSETSPAAAVNQPAFGARPGTIGHPLWGVDVEIARSETEDAVELLPPGELGEVVVRGHNVFSGYLGRPEATAEALVDGWFRTGDLGTKDGDGFLRIVDRKKDVIIRGGYNVYPREVEEVLARHPGIAQVAVIGLPDDLHGEEVCAVVVPAQGSAPDAREVTEWSKEHLGRHKYPRRVEFADALPLGPSMKVLKRELRARYADRPVTVTG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04273 Long-chain fatty acid--CoA ligase MTVALHDLLPATLRRTWAVEGTCPDLDLYSLYRARQIADPHRTAVLDGKGKLCYTALDRKARCLAAGLSGLGIHAGDVVGVQLPNGRDAVVADLALAALGAVALPFPVGRGGREAASLLRRSEAVAVIATAEHRGNHHAADLLALTGELPALRTVVAAGPAGAAPQGAVPLSALTRTDPKTFAPARPDPDTAARILVSSGSESEPKMVAYSHNALAGGRGNFLGSLIPDGRPPRCLFLVPLASAFGSNGTPVTLARHGGTLVLLDHFTPEAALEALAEHEPTHVLGVPTMIRMMLDRIAEGGHRTFTPPTAMVVGGSPLDEATATEARLAFGCPVVNLYGSADGVNCHTGLTHGSPDGDGRPGIAAGQPDPRVADIRIAVPGTRELREVSGGTVGEIVARGPMTPLCYVAAPELDTRYRTEDGWVRTGDLGLIDDDGTLRVVGRLKDVVIRGGANISPAEVEVELAAHPAVRDVVCVGVPDPLMGERLAACVVPRDEATPTLEELCAHLDTRGLERRKHPERLLVLSELPLTPAGKPDRAVLRERCTPQAERQQQPLASAG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04278 Long-chain-fatty-acid--CoA ligase MKTSTALRPQSARVHHPEPGTLVHTARFHAARQPEATAVICEGRTVTYADLHRESNRMAHALRAAGLGEGDRVAYLGKESEHYYEALFACAKTGTVLVPVNWRLTAPEVSHILQDSGTRLLFLEDEFAPIVEGMPTEPPETVVPVNSIHSWRAQHPDDETEFEATPDTPVAQLYTSGTTGLPKGVVLAHRSFFAIRDGLASEGLDWIDWRAGDLALIGIPGFHVGGLWWATQNFNAGTTVVAMRAFAARQAVDLIRDLGITTACVVPAMLRMMLNEPGVSAQDFSTLRKTVYGGSPISEALLEESLTVLDCEFAQIYGLTETGNTAVCLPPAAHVPGGPLMQAAGRPYPGVRAKVIDHRGRELPPGAVGEVCLHTPARMVEYWGLPEKTAETLVDGWVHTGDAGYVDREGYVFIRDRIKDAILVAGENVYPAEIENVLEHHPGVGEAVVVGVPDARWGEKVHAFVVPAAGERPSPRDLHTFLVPRLAAFKLPASYEFTDRIPRNPSGKILRRELRDRFWNDSARKVN Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04296 LTX-302 WKKW-Dip-KKWK Synthetic peptide Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 75 ± 5 µM
dbacp04299 LTX-315 KKWWKKW-Dip-K Synthetic peptide Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 38 ± 3 µM
dbacp04305 LTX-318 OOW-Dip-OOWWO Synthetic peptide Cell membrane disintegration MTT/MTS assay HT-29 Colon cancer IC50 : 248 ± 5 µM
dbacp04367 M1 family peptidase MTNRPDRPLRPSRRRTRRGRAALGAGLALAGTAYGMGTALGQPVPGPATAPADDGVRAYDVAGYDVRVTYDPEASRLEGDAEVAVRATADLARFDLDLALTARSVDIDGKPARSFSRSGDGSVTVVPEEAIEEGRTFTVRVRYDGDPGRSNPSWARGEDGGVITVLAPVGTWFPGNGDPDDTADFRLAATVPDGWTVVSGGRDRPVRRHGGRSTFDWRSTKPLPAKDALFGVGKWDVERTRLADGTPLTTVYAAGRKAEFEKYADQQRGIMSFLSSEFGPYPNDTLVSYFLDSVSEEVPNLAVQGGVIFPNAENEAYFDATVVAHELTHQWYGSLVREKEQRNLCLSECFASYAQWMWPEFSAGEDLDAKYRQEIEEHRTDDGFWQQRLSEGRGVYDKGPVMLHALRRQIGEAAFAEVLREWPARYGGTAPEWAELEKLVQEVSGQNLKGFFDAWVRGDRAPDDAYLRSRS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04372 M28 family peptidase MPRSPLSGRALTAGAVAVATLMAGGSAAGAASAAEWPAAVADAPDIPVANVKAHLTQLQSIATANGGNRAHGRPGYQASLDYVRAELDAAGFTTSLQEFTASGSTGYNLIADWPGGDADQVVMSGAHLDSVTSGPGINDNGSGSSAVLETALAVARSGYQPTKHLRFAWWGAEELGLVGSSHYVDSLGSADREKISGYLNFDMIGSPNPGYFVYDDDPTIEKTFKDYFAGLGITTEIETEGDGRSDHAPFKNAGVPVGGLFSGADYRKTSAQAAEWGGTVGEPFDPCYHSSCDTTANVDDTALDRNSDAIAYAVWELSQ Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04377 MAC1 GFGMALKLLKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 23 ± 4 µM
dbacp04380 MAC1/1 gfgmalkllkkvl Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 19 ± 2 µM
dbacp04383 MAC1/10 GFKMALKLLKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer Not found
dbacp04386 MAC1/16 GFGMALKLLKKVL-NH2 Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp04389 MAC1/19 GFGMALKLLKKVL-NH2 Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 68 ± 2 µM
dbacp04392 MAC1/2 AFGMALKLLKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 16 µM
dbacp04395 MAC1/20 GFGMALOLLOOVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 35 ± 4 µM
dbacp04398 MAC1/21 GFGMALRLLRRVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 17 ± 2 µM
dbacp04401 MAC1/24 GFGMALKL-(AC6C)-KKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 16 ± 1 µM
dbacp04404 MAC1/25 GFGMALK-(AC6C)-LKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 14 ± 1 µM
dbacp04407 MAC1/26 GFGMA-(AC6C)-KLLKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 18 ± 1 µM
dbacp04410 MAC1/3 LFGMALKLLKKVL Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 11 ± 1 µM
dbacp04413 MAC1/4 GFGMALKLLKKVL-NH2 Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 49 ± 9 µM
dbacp04416 MAC1/6 GFGMALKLLKKVL-NH2 Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 29 ± 3 µM
dbacp04419 MAC1/9 GFKMALKLLKKVL-NH2 Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : 13 ± 3 µM
dbacp04422 MAC2 GTGLPMSERRKIMLMMR Wallabies and their analogs Cell membrane damage MTT/MTS assay SW Colon cancer IC50 : > 100 µM
dbacp04446 Maculatin 1.3 GLLGLLGSVVSHVVPAIVGHF Fringed Tree Frog, Australia Disruption of cancer membrane integrity Not specified Not specified Colon cancer MIC : 1 – 100 µg/ml
dbacp04456 Maculatin 1.4 GLLGLLGSVVSHVLPAITQHL Fringed Tree Frog, Australia Disruption of cancer cell membrane integrity Not specified Not specified Colon cancer MIC : 1 – 100 µg/ml
dbacp04465 Maculatin 1.4 GLLGLLGSVVSHVLPAITQHL Fringed Tree Frog, Australia Disruption of cancer cell membrane integrity Not specified Not specified Colon cancer IC50 : 10−5 - 10−6 M
dbacp04490 Magainin 2 GIGKFLHSAKKFGKAFVGEIMNS African clawed frog Dissipate ion gradients; Induce osmotic lysis; Membrane damage Trypan blue assay Daudi Colon cancer IC50 : >150 µg/ml
dbacp04667 MFS transporter MASSLTKDSVSPGTPGSEKTFFGHPRGLATLFMTEMWERFSYYGMRALLPLYLVAPGGLGLSAGTATAIYSVYLSLVYLLTMPGGWFGDRVWGPRKTVAVAGGVIMLGHLTLALPYAGTFYAGLGLVAIGSGLLKANISTMVGQLYDGPDDPRRDGGFTVFYMGINLGAFFAPLTIGTIGESVNWHLGFALAALGMGLGVVQFLLGSRHLAPHSSTVPKPLSAEEKTSTLRKAAFWAALAVVFYAIVGFSGHYTLNWILVPLTLLGVIIPVLVLTSIKRDKSLDRAEQSKMSAYIWFFVAAAVFWMIYDQGGSTLSLFADSSAKNSVFGWGFPVSWYQSVNPVLIMALAPVFATLWLALARRGREPSTIVKFAFGLVLVGASFFLFLAPLGIAEGGHKAAALWLVAIYFVQTCGELLLSPVGLSVTTKMAPVKYASQMMGVWFLAVTAGDATTGLLSLAGVDLNKTGIVAAEATLAVVAGLAIWMYRRRVKELMGDVR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04672 MFS transporter MKNAQPDGPPPSGDDAAFFGQPRGLLTLSGLEVWERFSFLGMQAILVLYFADTVANGGLGMAAGTAASVSAAYGTLVYLVSVAGGWLADRILGSYRAVLWGGILIACGHYAMAVPAGATTWIGLGLISAGTGLLKPNAATMVGKLYRTDDERRDAGFAVYYMAINIGAFAGPLVTGWLSDHQGWHWGFSAAAVGMTLGLAQYVLGRRHLAGRRHAAEFALAPDAMRRAVRLIASGVVAAAVVATVLALAGWLTMSRFVDLLTLISVLAPVAYFAVMFASPRVTSQERGRLKPYVVIFLASTVFNYILFQAYSTMMLLASTDAETTLLGFDFPASWYASALGAFEVALAPVVAALWVRMGRRQPHASNKIAIGVVLGGLSFLLMVLPTSGDSGGHLMSAWWIVGSYLLLGLGDIVLETSGMSATTKLAPTAFSSQTMSLWFLSLALANGIQAQTVKLYDHVSQPAYFGVNGAIAVAAGLAVMAAAPYLRRTMHPVH Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04685 MIP PRFWEYWLRLME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.01 µM
dbacp04686 MIP PRFWEYWLRLME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.12 µM
dbacp04687 MIP(F3A) PRAWEYWLRLME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.57 µM
dbacp04688 MIP(L10A) PRFWEYWLRAME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 1.14 µM
dbacp04689 MIP(M11A) PRFWEYWLRLAE E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.4 µM
dbacp04690 MIP(R9A) PRFWEYWLALME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 0.02 µM
dbacp04691 MIP(W7A) PRFWEYALRLME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : >100 µM
dbacp04692 MIP(Y6A) PRFWEAWLRLME E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : >100 µM
dbacp04717 Multivalent DR5 binding peptides, TRAILmim/DR5 (1m) WDCLDNRIGRRQCVKL Not found Inducing apoptosis Not specified HCT 116 Colon cancer Kd (Binding constants of TRAIL mimics): 129 ± 3.68 nMol/L
dbacp04718 Multivalent DR5 binding peptides, TRAILmim/DR5 (2m) WDCLDNRIGKRQCVRL Not found Inducing apoptosis Not specified HCT 116 Colon cancer Kd (Binding constants of TRAIL mimics): 664 ± 18 nMol/L
dbacp04719 Multivalent DR5 binding peptides, TRAILmim/DR5 (3m) WDCLDNKIGRRQCVRL Not found Inducing apoptosis Not specified HCT 116 Colon cancer Kd (Binding constants of TRAIL mimics): 226 ± 5.64 nMol/L
dbacp04721 Mycothiol acetyltransferase MTSDDTVHPGRPRSIETLAELAPEQTEAVLALLAEAARNDGQYAVSEQGRLQLRGPAREGVAHLLLTADGGELVGYAQLEGVDPIEPPAAELVVHPSHRGRGHGRALGSALLAASGKRLRVWAHGGHSAARHLAQVLGLTLFRELRQMRRPLAGLDLPEPRLPEGVTVRAFAPGQDDAAWLAVNAAAFAHHPEQGSLTQRDLDDRKAEGWFDPAGFFLAERDGRLIGFHWTKVHAEEGLGEVYVLGIRPDAQGGGLGKALTTIGLRHLAGQGLPTAMLYVDADNEAAVAVYERLGFTVHETDLMYRTET Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04726 Mycothiol S-conjugate amidase MTDQLRLMAVHAHPDDESSKGAATMAKYVSEGVDVLVVTCTGGERGSILNPKLQGDPYIEEHIHEVRKKEMDEAREILGVRQEWLGFVDSGLPEGDPLPPLPEGCFALEDVDKAAGELVRKIRSFRPQVITTYDENGGYPHPDHIMTHKITMVAFEGAADTEKYPEAEYGAAYQPSKVYYNQGFNRPRTEALHHALLDRGLESPYADWLKRWAEFERKERTLTTHVPCADFFEIRDKALIAHATQIDPDGGWFRVPLELQKEVWPTEEYELAKSLVETSLPEDDLFAGVRDNA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04755 N-acetyltransferase MLSLALRDGVRLRALEVWHAQEFAAHLDRAREHIRPWVGAAFVTDDVAGARATLRRYGESGAADGARLYGIWRDGVLVGGVMYVHFSEALGSCEIGCWLEPSAEGQGLVTAACGALLDWAFTARGLHRAEWHCRADNARSSAVAERLGMSLEGVRREAWPYEGRRYDKQLWAVLAPEYAHPGG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04760 N-acetyltransferase MLHAGQFEQALTVTQVTERRMTSTFPNISINTERLVLRPLDEDDVPALAAMMNDEQVAAWTHVPQPFTEKDAGVWIGDHAPAERTAGRGLDLAVTEFLTQRLVGVVRLTRTDWHVRSTELSYIVAPWARGEGYASEAALATAQWLFGDQKFERVELRTAADNTASQQVAQKIGCISEGVLRGACIARARTDDGVWTDVRTDFIVWSLLPEDLEGTTGQPVGSDGFTAFTDWN Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04765 N-acetyltransferase MPSMPYLTRPVIAEGTLSRTPQPALPTGDGLLLRPWRADDAPAVHAAFQDPAMHQWHARAADSEDEVRGWITEWQRAWEGERGVQWAVADASDDRLLGRVALREVVLGDGVAEVAYWTTAAARGRGVAARATRALAHWALDGIGFQRLELLHAVANEASCRVAHKSGFALEGTKRSALLHPDGWHDMHLHARVRGD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04770 N-acetyltransferase MAPTPAHRTHATGVPDPSRAEPRGHGLHLRSWDADSDSDAEAWLRGFLDPEFQRWNTPLNLWTDVAGARESLRARARDAADGRSVSFRVTDGGSGTTLGHIGVNEISRQMKVARVGYWVLPAARGRGVAGRALLLASRWAFAELGLHRLELGHAMGHEASCRIAERCGYRAEGTLREAMFESGRHDAFRDVHLHARLATDTEPAPPDTR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04775 N-acetyltransferase MEPVTLTTDRLVLRTVGSQDTEAVYAAAQDPDIQRWTTIPSPYLLEHARNFAEQAVPDGWANDSMFTFGLFLPDGDLAGMLGVTMISLGVGEIGFWGTKEHRGHGYVTEAAVAVSRWAFTERAVDRLEWRAEVGNTASRAVARRAGYTMEGTLRSAINNNGVRRDCWIASLLPSDLTLPSTSPYLPAP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04780 N-acetyltransferase MNSPSWPAELRDGGIVLRPIRLRDQRAWREVNRRNRDWLRPWEATIPPPGPGGPITSRPTYRQMVRHLRSEAHAGRMLPFVIEYQGRLVGQLTVAGITWGSMCSGHVGYWVDEAVAGRGVMPTSVALAVDHCFRTVGLHRVEVCIRPENAPSRRVVEKLGFREEGLRPRYLHIDGAWRDHLVFALTADEVPEGLLRRWHRSRNRSTPNAGN Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04785 N-acetyltransferase MGGVTGGELGAEQVQAAVAGSVALLATAADRDWEAARAGRLEWSCRYTAEHVAGDLITYAGQLAGRATTAYVPFEITLDEGTGNGGVLRVIETTGALLAATLRTTPREVRAFHPYPYRSANREGFAAMGVAEVLLHTHDIAEGLGLSYEPPAGLCADVLTRLFPHVRPGGDAWRTLLWATGRGELPGRAPVTEWRWRNNLVVPAERLTLQGVTPAAATDLAAGGDGGFAWVDGGPLEGTRFSAGMVLKAYEAGTHRPEWGVFVLVRRADGRAVGGIGFHGAPDEDGRVEIGYDLAEAARGNGYATEGLRALSAWALDRDEVTSVFATTEPHNAASQAVIARAGFRRAAVVEEHGGESGQYAYELRR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04794 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer > 100% cell viability at 5 µM
dbacp04795 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 60% cell viability at 50 µM
dbacp04800 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer > 100% cell viability at 5 µM
dbacp04801 N29D PDEDAINDALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 60% cell viability at 50 µM
dbacp04806 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 100% cell viability at 5 µM
dbacp04807 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 40% cell viability at 50 µM
dbacp04812 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 100% cell viability at 5 µM
dbacp04813 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer 40% cell viability at 50 µM
dbacp04818 N29N PDEDAINNALNKVCSTGRRQRSICKQLLKK Synthetic peptide Apoptotic inducing Cell viability assay SW-480 Colon cancer MIC : 5 µM
dbacp04827 neo-N-methylSansalvamide A NA Marine fungus Apoptosis induction Not specified HCT15 Colon cancer 0.85 ± 0.63 nM/L
dbacp04833 Nickel ABC transporter permease MSAPRSRAGRLARPDARLRRLPVTSRIALGVLLVVVLGAVFAPLLTQDPLATGIPARAPGADHWFGTDRAGRDVFARVVHGARYSLVIGLGATLAALVLGSALGALAATSRRLADESVMRTLDVVMSFPPIALAAVLVAVFGPSVPVIIFTIAFVYSPSLARVVRANVLEQYGEDYVAAERVVGARRGHIVVRHVAINCAAPVLVFATVMVADSIIFEASLSFIGAGVQDPDPSWGSVLAYGRQILLSGGWWATLFPGLCVLVTVLALNVLSEGMTDAAASPDTSRTGGTDSDATAATAPAAERADGAEVDAALAELASRLRATEPAVPPLAADAADLLVVRDLSIRFPDRYGDTRVVDGISFTVREGETLGLVGESGCGKSVTSLAVMGLLARNAEAAGEIRYRGRDLLKLTPKERRALMGPEIAMVYQDAMSSLNPSVLIGTQLKWLTSRGGTRTPAELLELVGLSPERTLRGYPHELSGGQRQRVLIAMALSRGPRLLIADEPTTALDVTVQAQVVELLVRLRDELGFAMVLVSHDLALVGDLAHRVAVMYAGQVAETGETRALLTDPAHHYSRGLLGSVVSLESGAERLHQIRGVVPAPKAFGAGCRFASRCAAATELCATTPPPATDREAGLDHLFACHHPASALRPPSADRPAAGKTPASGDGPASGGPSATSLERAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp04838 Nickel-type superoxide dismutase maturation protease MMPEQLSQETERARGALPFGPAEVTGPSMVPTLHHGDVLLVHWGARVRPGDVVVLRHPFQQDLLVVKRAAERRRGGWWVLGDNAFAGGDSTDYGVVPEELVLGKVRLRYRPRAGQRSPFTVVRWALSALRPVLADRSASRRLRAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp04843 Nicotinamidase MRRALIVVDVQNDFCEGGSLAVSGGADVAAAITELIGQAPAGYRHVVATRDHHVAPGGHFADTPDYVHSWPAHCVAGTEGVGFHPNFAPAVASGAIDAVFDKGAYSAAYSGFEGADENGTPLAEWLRSREIDEVDVVGIATDHCVRATALDAAREGFRTQVLLDLTAGVAPETTERALEQLREAGVELSGKPVVQ Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp04890 Non-ribosomal peptide synthetase MPVSAAPQHHHYCPHRAATRSVDGPRGHDRRPSPHGGVHVIPASYAQRRLWLVDRLEGPSALYTVPLVLHLTGRPDVTALRAALHDVVARHEALRTRFPQVDGEPVQEIVPVGELDDLLTEDEVRADELEHEIGRTARHVFDLAAGIPFHARLLTVDDRTSALVVALHHIAADGWSAAPLWRDLSAAYAARLTGAEPDLAPLPVQYADYTLWQRELLGDADDPGSLLAEQLAHWRAALAGAPEELALPTDRPRPAASAHDGGVVRLDVPAGLHARLADLARDENATMFMVWHAALAVLLSKLGAGEDIPVGSPFAGRDEADLEDLVGFFVNTLVLRTDVSGDPAFTEVVRRVRGTAVDAMNHQDVPFERLVEDLAPARSLTRHPLFQVNLTLHNTPRLPVDLPGLTAVAEFAAPPLAKYDLDVQVQEHADAQGRPAGQRVELHYSADLFDRTTAEAIAGRLLRVLSQVAHTPELPLHAVDVLSPAEHQALTAAAGSAAAPPPGDTVPDLFAARAAAHPDAAAVTHGATTLTYAELDAESNRLARHLVARGAGPETRVAVSLERTPGLVTALLAVMKAGAAYLPADPAHPAARTGALLADAAPVLLLTTADTAAHAAAAPELRRVLLDDPQTRTAVAARDAGPLTQDERRTPLRPGHPAYVIHTSGSTGAPKGVVVGHAQVTALLRSAADRYGFGTDDVWTWFHSYAFDFSVWELWGALLTGGRLVVVDHDTSRSPDDFHDLLVREGVTVLSQTPSAFQQLDQADARRDAAALGARLRLLVFGGEALDPARLTDWHDRHGTDGPRPVnMYGITETTVHVTHLDLDPGTAAAPGTHGGSPVGRPLDHTRVHVLDDALRPVPPGVPGEMYVTGSGVARGYLNRPATTAARFVACPFEPGTRMYRTGDRARRAADGTLTYLGRTDDQVKLRGFRIEPGEVEAALLDHAPIGRAAVVLRTDTPGDRRLVGYVVPRDPAAATGEAGAELARRAREHAAALLPAHMVPSVCVPLARLPLTANGKLDRAALPAPDREGAAGGRGPATAREEILCTAFAEVLDLPSVGADDDFFALGGHSMLAVRLLDHLRTRGVRVDMRTLFTAPTPARLAAAAGPEPVRVPEGTVPPGATRLTPEMVPLAGLTEDELRTVTDALPDGAAGVADVYPLGPLQEGLFFHHRLNAGTGTAGGSGDGDPYVVRYVLGFDTPRLLDSFLAALAQVIDRHDVLRTSLAWTGLPHPVQVVHRHAELPVTETDLGDGPDPVARLLAHGDEPLDLRRAPLMDARTATEPGTGRRLLAVRMHHITQDHTTLDLVLREATAVLAGRGGTLPAPRPYREFVGRALLTTPAEEHLAHFGRLLGDVTEPTAPFGVWEVRGGGTDVTERRTVLGEPVAARLRAQARRTGVSAATVLHVVWSRVLAAVSGRDDVVFGTLLLGRMQAGDGAGDVPGMFINTLPVRARTAGTDVAQAVHAMHHQLAELMVHEHASLAVAQRAGGVRPPAPLFTAVLNYRHNPEGGPGTVLPPGTELLAFRERTNYPLLVSVDDDGGALAFDVQAATPIDPDLVTRLLHATTERVVDALEQAPDTPLADVDVLPAAERHRVLTEWNDTGRPDTARTLADVLADRATATPHAPALTHDHDGVPEQLDYAELFARANRLARHLIGQGVGPEDRVVLLMDRSPDLVVALLAVVGAGAAYVPVDPDQPAVRVAHLCVDAAPAAVLTGRAHAASVPRSAPAPIVVDDPEVRSAVAAHAPDPIGQDERTCPLRPSHPAYVIYTSGSTGIPKGVVVPHSGAVNLLAFRWPGLTADSSLLQFASIGFDVATWEIMTAFAAGARLVVAPAARLLPGAGLEDVVERHAVTHLQLPPTVLGMVADDHRLASVRTLLVAGEALGQALVDRWGAGRWFGNAYGPTEITVIAAADGPLRPGDAPTIGRPLPGVRLYVLDARLRPVPDGVDGDLYVAGAGLARGYLDRPGLSAERFVADPHGAAGTRMYRTGDTVRRTADGRLLYTGRADDQVKIRGFRVEPGEIETRLTEHEGVAHAAVVARDDVPGAPGDTRLVAYVVPSGPGVPAALRDHLAALLPAHLVPSAFVALDRLPLSVNGKLDRAALPVPDPATGTGAARPAGTYDELLCAAMAQVLGVPRVGADDDFFALGGHSLLAVRLVGRIRAVLDVEIPVHAVFEAPTAARLAARLDEWTGAQVRPSVVAGERPGRLPLSYAQRRLWFVDRLEGASALYNIPLVVRLSGRVDVGALGAALGDVVGRHEALRTRFPQVEGEPYQEVVPVAEARVELPVVPVAAGELEARIEEVSGHVFDLAGELPVHAALLTSGEESSVLVLVVHHIAGDGWSLAPLWRDLSAAYGARRAGGTPRFAPLPVQYADYTLWQRDLLGDAADPGSVLAEQVAHWRTALEGVPEELSLPADRPRPSAKTHRGAAVPVRVPAGLHARLAELARSEGVTMFMVWQAAVAVLFSRLGAGEDIPLGGPVAGRTDESLEDLVGCFVNTLVLRTDLSGDPAFTDVLARVRRDTLSALHRQEVPFERLVEELAPPRSMGRHPFFQTVLEVQSTPLLAPELDGVNVAVLPHAVRDAKFDLDLQIAESFDAEGRPTGMAGELVYAADLFDHATAETLTARLLRVLDAVADAPGRPVHTVDVLDDAERRRLVGEWSRRQPAIAGPDVRVFVLDDHLMPVPPGVTGLLYTTCDASADSTVACPFTEEESVMRPTGAQARWDDEGRVHVVPADDAAAPEADTQPSGAPVPRGSGTELREELLRTVFAQVLGVPEVGADDDFFALGGHSLQAVRLVSRIRAVLGVELLVRDLFETPTVAGLAARLDDTAGAQVRPSVVAGERPGRLPLSYAQRRLWFVDRLEGASALYNIPLVVRLSGRVDVGALGAALGDVVGRHEALRTRFPQVEGEPFQEVVPVAEARVELPVVPVAAGELEARIEEVSGHVFDLAGELPVHAALLTSGEESSVLVLVVHHIAGDGWSLAPLWRDVSTAYAARRSGKTPDFPPLPVQYADYALWQQRLFGDEDAAGSRLAAQVEHWRATLDGVPHELALPFDRPRPARPGRGGGWADIEVPAELHARMAELARSEGVTMFMVWQAAVAVLLSRLGAGEDIPLGSPVAGRTDESLEDLVGFFLNTLVLRTDLSGDPAFTDVLARVRSTALDALDHQDVPFDRLVEKLAPARYTDRVPFFQVLVAVQnMPQAQVALPGLDVDAGPGKPTTAKVDLDVQVVELHDADGAPSGMAGGLTYATDLFDHSTAESLVARLLRVLDAVTADPARRVSRIDVFDPAERRRLLTESNGARSDTLALTVPELFAVRASRAPKAVALDTGAEPVTYGQLDARSNRLAHHLIDLGVGPETVVAVVMDRSPDVVTTLLAVLKAGGAYLTLDPAQPDSRTAEMIALAGAEVCLADQRYAEAARGRFATVVVADAGDAEWADRPAGTVAGRSLPDQLAYLMFTSGSTGEPKGIGTTHRDIVDLAGDRCWQFPGTARGMFAAPHTFDGSTVEVWVRLLTGGTLIVTPPGRTDAARLRSLVADHGLTHAHLTAGLFRVIAEEDPAAFTGVHDVLTGADVVPREAVRRVLEAVPGIVVRSSYGPTEATVIATQIPLTEPDALGDVVSIGRAMDNTGVYVLDDSLQPVPAGVAGEAYIAGAGLARGYVARPGLTAERFVACPFDVPGARMYRTGDIVRRRADGALEFVSRADDQVKIRGFRVEPGEVEKILAGHPAVAQAVVTVREDTPGDKRLVAHLTAAPGEALPDVREFVAGRLPEYLVPDAVVVLDRLPLTANGKVDRAALPAPEAASTGAARRPPSLREDLLCSVFAQVLGVPRVGVDDDFFALGGHSLLAVRLVSRIRSVLGAEIPVQAVFETSTVAGLAPTVEAAGSTGVLRPALAAGPRPPRLPLSYAQRRLWFVDRLEAAGPLYNVPLALRLTGALDTGALRAAWTDLLTRHESLRTRFLHADGDPYQDIVSLDDFPPYFAVESVGRGELEARIDEAAGHVFDLTAGPPVRATLLDVDGPDTDEAVLVLVTHHIVADGWSMVPLLRDLSTAYTARRAGRAPGWEPLPVQYADHTLWQRGLLGDGDDPDSVLAGQVAHWREALDGSPEELALPTDRPRPAVASREGGWVPMSAPADLHARLTELAVAQGATAFMVWQAALAVLLSRLGAGQDIPIGSPVAGRTDEAADDLIGFFVNTLVLRTDLSGDPTFTEVLGRVRRSALGALGHQDVPFERLVEELAPTRSRARHPLFQILLAVQNVPAATVDLPGLRVEALPTELGRAKFDLDLHVAEAFDDEGRPAGIDGGITYAADLFDRTTVEALLDRLLLVLHAVAADPSRRVHDIALLDSDDRHRVLTEWNRTERAAPAATVPDHFRAQAARTPDAAALVTDGARTTYAELDAASDRLARYLTRHGAGPGRLVAVVMERSPETITALLAVLKTGGAYLPVDVGYPAARIELMLRDAAPALLLTTTDLADRLPGSAGGPDRIVLDDPSVRDAVAAEDATPTATPPHLDSAAYTIYTSGSTGTPKGVVATHRAVDRLVRPADYADLRAGDVVSHLGSVSFDSTTFDIWATLLNGATLAVGPAGSPSVADIRDYLARHRVTVALLPTGLLHQVIDLDVEALRGVRSVLTGGEALSVEHCRTLLDTLPGTRLMNGYGPTESVTYTHTHPVTRADVDSGRAIPLGRPLARTRAYVLDSALRPVPVGVPGELYIAGDGLARGYANRPGLSAERFTACPFEDGGARMYRTGDLVRWRADGVLEFVGRVDDQAKIGGFRVEPGEVEATVSAHPDVAQAVVVVREDTPGDKRLAAYAAPADPAVSGRELADRIRHFVADRLPDHLVPPFVTVLDRLPLTPNGKVDRAGLPVPDPMAAVSVARGPASPYEELLGVVFADVLRLPRVGVDDDFFALGGHSLLAVRLVSRIRAVLGAETSVATVFENPTVSGLARQLTRAGGRARPALVPMPRPPVLPLSYGQSRLWFVDRIEGPNHLYNICLVLRLTGDLDPELLRLALADVVARHESLRTTFPLVDDEPSQHVLAVEEAAVDLPVTAVTEEELAGRLDALAAHPFDLARELPLKTELFSLRPGEWVLSATVHHIAGDGWSMGPLWRDLSQAYLARAAGRAPEWEPLPVQYADHTLWQRDFLGDVDDPDSVLATQVAHWKERLRDAPQELALPVDRPRPAVSDHRAGLVPLNIPAPLHARLAELALGQGVTMFMLLHAAVAVLLSKSGAGRDIVLGSPVAGRTDQALDDLVGYFAGTLVLRTDLSGDPDFLELLDRVRTAGLDAFEHQDVPFERLVEELAPARSMARNPLFQVMLAVQNNQRGTLSLPGVQVREEPAGALTARFDLDFEVRESFDESGAPAGLDGEVVYAAELFDRSTVQTLTARLLRVLETVAADPTLPVTRVDLLDDAERRRVTEEWNDTAGPLPDGTLAGLFDRQAARTPDAVALVHDGAEITYAELDERSGRLARHLIGLGAAPETLVGVALDRSVEQIVALLAVVRTGAAYLPVDPGQPRRRTDLVLTDASPVLVLSTAETTARLGGTEAGTPARWIDLDGPLADGLRDTPAPAAVTDADRGTPLRPHHPAYVMYTSGSTGTPKGVVVPHSGVVNQLAWMQEEYRLEPADRMLQRASFGFDASVWEIFWPLLNGAAVVLSGPGSHADPEYLADLVDRERVTVAQFVPSVLRTFLDGGAAGRCTSLRTVLCLGEALPAAVRDRFRQTLDAELHNLYGPTEASVAVTAWPCDAAQDGASVPIGRPLRNIRAYVLDDGLLPVPPGTAGELYVAGTGLARGYLGRPVLTSERFVACPYGPAGERMYRTGDIVRWTAGGHLEFLDRADDQVKIRGFRVEPGEVEATLATHPEVAQAAVVTREGPGGDPALVGYLVPAAAGDDGADLVARVREYLAERLPEHLVPPVLTPLDTLPLTPNGKLDRAALPAPDYTALATGGRAPATLREQLLCSVFEQVLGVSPVGVDASFFDLGGHSLLAVRLVNRIRVVVGADVPVRAVFEAPTVAGLLAWIAREGRQGTADVLVPMRSTGERPPLFCAHTVLGLGWEYGWLTDAAPGDQPLYALRPRGMDTGTAELPDSLPRMAADYVEQIRTVQPTGPYHLLGWSFGGNVVQEMAAQLQDAGEEVAALVLLDSSPVDGPATAEQRAGFAEQEETVAGALTGEEHEAYLRIVRNNTRILLAHRTRKTTGTLLLVSADSETKAALWRPFVSGEVREHVLDCAHRDMLLNPDVVRRIWDIAADELEPTDTDDTDNDPDRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04895 Non-ribosomal peptide synthetase MTKQSGLQDILPLAPLQEGLLFHSVFDEKAPDVYLVQQAIDLEGDLDTAALAAACRTLLRRHANLRAAFRYQGLKRPVQLIPHQVELPWEETDLSRLPEPERSAAADRLLEEDRLRRFDLGRPPLMRFTLMRLGDGRYRFVLTNHHILLDGWSRPMLVRELLALYRTRGDDSALPRVRPFRDYLQWLAGQDRDSAVAAWREVLAGLDGPTLVAPQAGERTPVVPGRLETELADADHAALTRLAREHSLTLNSLVQGAWAVVLSGLTGRDDVVFGTTVSGRPPEVAGIETMVGMFINTLPVRVRLRPDEPFLDAVRRTQDEQTRLQSHQQLGLAEVQRLAGEGELFDTTMVFENYPVDIGAERDEPGGIGGVTVTGTRNRDATHYPLALVAVGRDGLRLRLDHQPDLVPPAAARAVLERLVRVLRGAASEPHRTVGRFELLSAEERGAVLSLGRGTDTGPADTTLPAAFRAQAERTPHADAVRCGTTVLDYAELDVRSDRLARALVAHGVRTETPVGLLMDRSEHLVVALLAVLKAGGAYVPLRQGDPLDRLRQVTALAGVRHVLTDAEHAARAGELGVTAVRADAADAPAGGAELPSGPGHADRLAYVMHTSGSTGMPKGVAVTHRDVVELARDRSFACGAHARVLVHSPHAFDASTYEVWVPLLSGGTAVVAPPGDLDADTLGKVLTEHEVTGLWLTAGLFQLVADEAPHHLAGVREVWTGGDVVQAAAVRRVREACPGTVVVDGYGPTETTTFAVRHRIPANAPVPDTVPIGTPLDNTRLLVLDTALRPVARGVAGELYLAGAGLARGYWRRPDLTAERFVADPHGPAGTRMYRTGDLVRWTPDGTLEYLGRADEQVKIRGFRIELGEIEAVLGLHFEVAQAVVTVHEPRPGDKRLVAHLVAEEGSDPTPASLRDHLAAELPDYMVPSAYVSLDALPLTGNGKIDRRALPVPDLTAADATVESRAPRTPREEILCGLFAELLGMPRVGVDDDFFALGGHSLLATRLVGRIRAVLDAELTVRQLFDAPTVAALSRALDTAGAARPALRPAEPRPERVPASPAQRRLWFLHRFEGPSPTYNIPFALRLSGDLNRSALRAALADLTDRHESLRTVFAEDAEGPRQIVRPAAEARPELTVVPSAPSDGLEAEVARAASYSFDLAAEIPLRAWLFETGEREQVLLLLVHHIAGDGWSVPLLARDLTTAYTARLGQRAPQWRPLPVQYPDYTLWQREALGSEDDPDSPAARQLAYWRDALAGLPEELALPADRPRPATAGGRGGRVLYEVPEELHARIVTVARTCQASPFMVVQAAVAALLTRLGAGEDIPLGTPVAGRTDDALDGLVGFFVNTLVLRADTSGNPAFRDLVARVRETDLAAYAHQDVPFERLVEVLNPKRSPARHPVFQTMLTFNNTDRRPGDGLRLPGLDAESLSADTGTAKFDLLFSFAERHDAEGRPAGLGAGLEFSTDLFDPDTAEALVARLLRLLDAVTAAPDRAIGAVPLLGDEERARALSASLGPARVPVGGSLPERFAVSVARAPHAVAVETAEGVLTYAELNARANRLARLLVERGAGPESLVAVAMHRSAELVTACLAALKAGAGYLPVDPEYPADRIAYMLDDARPASVLTTRDLAGALPTGPAGTPLVVDAPATVARLGSLPDSDLTDTERTSPVGPAHPAYVIYTSGSTGRPKGVTMPVRALANLLDWHERTLPGGPGTRVAQFTAVSFDVSVQEILSALLAGKTLVVCPEDVRRDPERLAGWLGERQVQELYAPNLVIDAVCEAAVAARLDLPHLTDLVQAGEALTPHGAMRAFCAARPGRRLHNHYGPAETHVVTAHRLPADPAGWGPSAPPIGRPVDNTAVRLLDPWLNPVPPGVPGELYIGGDALARGYLGRADRTAERFVADPYGADGARMYRTGDLARLTPDGLLVYLGRADSQVKIRGFRIEPGEIEAALTAHASVAQAAVVVREDRPGDRRLVGYVVAAHQEAPDSARLREHLSGRLPAHMVPAAFVVLEALPLTPNGKLDRTALPVPEYAAGGGSRAPRTPAEHRVCTLFAEVLGVERAGVEDDFFELGGHSFLAARLVARLREEFGQDLPVRTVFDSPTPEGVAAVLTGTADGGPGRSSESLLALRARGTAAPLFCLHPGGGFSWCYAGLVRHLGPDVPVYGIQARGLDGSGPLPSSMAEMTAEYLALIRSVQPSGPYRLAGWSFGGLVAHALATALRAEGEEVSLLALLDAYPPGENADTSEPVEHEVVAHNLRAMGFEFDMAELIADQEGVLRRFREFLQSGDQALAQLEARDILALKDVYVNNVRLMRKFTPEFFDGDVLFVSAERKSADDREGRLNVSLWQPFTGGSVEVCAIDSTHGNLMTDARHMARIGQFLADRL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp04900 Non-ribosomal peptide synthetase MTEQSAVGLPLTPAQESLWFAHQSRPLDAGFLIAEYVDIEGELDLTTLRRAVASVARETEALRTTITDAPDGGTAGQRVHDGMALDVPLVDLSASANGEADAHRAMLQDLATPVDVTRGPVTALVLYRLSTSRHLLYLRTHHLVLDGYGAAAALGRIATTYGLLATGEEVTAEPLPLEPLVADARQYARSAEYAEDGAYWRESLAGAPHAERLTDRTGPPGTEVLRRSVALDPARWRRLREGARQGRVAWPALFVAGTAAYTHRMRGAHDLLLGMPVTGRRSRIARRTPGMTSQIVPLRLRLDPAVPVRDLLRQVTTAMRGALRHQRFPVEELRRELGLGRGDSLVGPAVNVLAFDENLRFGPATGTLHNLSLGPVEDLTLAVHPAPGGAGARVDVLANAALYDGTSAAGHLERILRLTEEFAADPDRPLSALELTGPEERDRVLALGTGPRERSRIPAPRTDAPVDGGVDGRPGPATAPTEHAGSTEHADVPEPTLPEVLARLARETPDAPAVDDGTRGLTFAELDRAVDAAASALRADGAGPGTTVAVALPRSVDTVVAPLAVLRSGAVYLPVDVTYPAERIAHLLADAAPVVLLCAPGGPVAGMAPAGTAVRSLSRSGTTAPGAPFDGPRAEDAAYLFYTSGSTGRPKGVLVEHRSISNLLAHHRRESHASAESAGGRRLRVALTASTSFDASWDPLLWMLGGHHLHIADDTTRRDPEALVAFLRAERIDVIETTPSFLGQLLAAGLTAETPTADGADGAPVHRPTVIALGGEPVGDELWQRLSSQPGLLAYNFYGPTETTVDAVTARVRGTDPVIGRPVRGARAYVLDTALRLLPYGATGELYLAGEGVARGYTGRPGPTADRFLADPFGEPGSRMYRTGDLARWHENGSLEFAGRSDTQIKIRGQRVETGEIEAALAALPGIAQAAVALHADGPAGETLAAYLVPTPDEAGDGVRRDRRRVRDALAASLPAYMVPAAYAATDRLPLTPNGKLDTAALPRATAVSTGPKSPPRTATERAVCAAVADLLGLADVGRDDDFFSLGGHSLLATGLLADLAGRTGVRLPVRALFEAPTVAGLAARVDAGRRSAGPEDPPGGRAVAERPARLPLSAAQHRLWLLEHMGEGGDRYHIPVAVRLDGDLDVPALRAAFSDLLARHESLRTVYPQDAEGPHQVVLPAGGCGVELRTAPVLPDARPEDVPAPRFELAERPPVHAVLVPTAEPAGDGPGSHLLLLTLHHIVTDGWSMGPLVHDLCAAYRARTGGHAPRWQPLPAQYADYALRQRARLGDREDPGSLAARQLAASRAALEGLPPELPLPHDRPRPERATARGGRVPVRLDAADHRALGALAREAGVSPFMVLHGVLATLLHRLGGGDDIVVGTPVAGRDEEEFHDVVGFFVNTLVLRVGVGGDPTFRELLDRVRETDLSAYGRQDLPFEQLVEALAPPRSLSRHPLFQVMLALNNTPAPRLDLPGVHAEPLRSGRTTAKFDLTWDFTETHDAHGRPDGLTGEVEYSAELFDESTVRRFAGHFVRLLRSVLRSPDARLGALGMLTEDQRLAALDTGARDDSAERGDELVHSVCDVLETQAAVTPDRTAVAEGRRTVSFGELATGLRDTARLLAAAGVRPGDRVAVALPRSARQIAAVFGVLRAGAVYVPLDPAHPAARNARILESARPALLLTERERAAALPASRTPTLYLDEAPDAAPAAEALPADGPRGADPAYVLYTSGSTGRPKGVVVEHRALANLLRHHGRHLIEPAERANNGRPLRVALTAAATFDASWDPLLWMVAGHELHLVDDASRHDPEALVRILHERRIDVLETTPSFLEQLRVCGLFAPGRPWPRVVALGGEPVHEKLWRELAELSGVSVWNLYGPTETTVDSVIAPVTAGTGPAIGHAVTGMRARVLDSRLGPTPPGVTGELYLAGAGVARGYDGATGLTADRFLADPYGPAGSRMYRTGDLVRRRPDHSLVFVGRTDSQVKVRGFRVETGEVEAALTAHPAVRRAVVTVRQAEGGGRLVAWAVPETGARPTPAGLRAFLGDRLPAYMTPSHLALVPEIPLTAHGKTDFGRLPDPAPALAEQGERPRTPQEEILCALFAECLGTDSVGRDADFFALGGHSLLATRVVNRVRSAFGAEIPVRALFEDPTPAGLARHLDGAARGRPSLHARADRPAELPLSFAQRRLWFLNRMRPDDASYNLPMAVSLCGRLDVAALHGALGDVVARHESLRTVFREAADRSGTPVQRVLSPGAARPALTVTPSTPDQVAGLLREAARAGFDLGGDLPLRAELLRTGADEHVLLLTVHHIAADGWSMGPLAQDLAAAYAARVAGRAPDWTPLPVQYADYALWQRDLLGGHDDPDSVYARQLAYWRGALADAPTETALPADRPRPDAGSGLGGSVPLPLSGSDGRRLAELARREGASTFMALHAVLAALLDRYGAGDDVVVGSPVAGRTDEALAGLVGFFVNTLALRVRTDGDPDFRALLERARETDLAAYAHQDLPFESLVEHLAPPRSPARHPLFQVMLSLNNAGRPALDLPGLHAEVRGVDTDAAKFDLSFSFSEQSGDGELTGQLEFARDLFDTATAQDLADSFVALLRLVVADPDSPLSRHDPLDASRLAGPLGHGDGPQAAPRHPTVVAGFAATAAAARSSDIAVRCGAQALSFAELARDGARLAHLLRGRGVDADRTVAVLLPRSTGSLTALLGVLAAGGAYAPLDDALPPARVAAVLSDARPAVVLATAATADRIPDGPWQTVLLDSPGTWAELAALPAEFPDGAAPGPRDPAYVVHTSGSTGRPKGVVVEHRSLAQLAEHHRRTLFDPARAATGRHRLRVALTASLSFDAAWDPVLWMLDGHELLVVDNDTRRDPAALVRAVREERVDVLETTPSHAAALLDAGLCAEGSPGHRPAVLALGGEDVPPGLWRRLREVPGLTVWNLYGPTEATVDTLYARLDRGDRPELGEPVAGTSCYVLDRLLRPAAPNTTGELYLSGASLARGYLGRPAETAARFVPDPFGPPGGRMYRTGDLVRRTADGRLEFRGRADGQVKVRGFRVEPGEIVTALEAQPGVRRAAVALRPVGSGAAHGTEQLVAYVVPGDGPGASGGPAAPDRDALRAALAAELPGYMVPAAFVVLDALPLTASGKLDAGALPAPRGEHLAHAAGRAPSGPREDLLCALFAETLDVERCWSDDDFFTLGGHSLLAARLLARVREATGVELGIRELFEAPTPAGLATALTAREAEAGTGTGPGADLACLLPLRSGGSLPPLFCVHPAGGLAWPYAGLLQHVADRPVYGLQTPNLDGTEHFPDSIEAMAAYYVDQLRTVQPHGPYRLLGWSFGGNVVQEIAVRLQEAGEEVALLSIMDAFPVPPADGLEDAGHDVVFRALLTALGVDLSAWDADAPLDAAVVRDALRESGSPLGALEPAAIETMVGNFADQARLMRRHVPRTFRGDVLFFRATEEDPASGLVPSLWDPYVDGALVVHDVPCGHAQMLRPDARAVVGPVLDAALRAT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05082 P5317-28 QETFSDLWKLLP E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 4.7 µM
dbacp05083 P5317-28 QETFSDLWKLLP E3 ubiquitin-protein ligase Cell cycle arrest or apoptosis of cells Immunoprecipitation assay HCT-116-p53+/+ Colon cancer IC50 : 30 µM
dbacp05227 Penicillin acylase family protein MPPNNTASTGQQPGTSGRKKGRKGRLLVVVLVLAVVGGLVFGGYWSVSTVRASFPQTKGSITLDGLSGPVDVKRDGYGIPQVYASSEEDLFMAQGYVQAQDRFYEMDVRRHMTAGRLSEMFGKDQVGNDEFLRTLGWHRVAKKEYDEKLSDSAKKYLQAYAKGVNAYLKGKDGADLSLEYAALGFTNDYKPQEWTPVDSVAWLKAMAWDLRGnMQDEVDRALMTSRLGPKQIADLYPAYPYDRNKAIVQEGQYDELTQTFDGSGSSGGDSGTGTGAGTGAGSGTGAGAGTGAGSALEGQLAGLQNVLDDVPTAVGVNGNGIGSNSWVVSGEHTITGKPLLANDPHLSPSLPSVWYQMGLHCRTVSDKCRYDVAGYTFAGMPGVVVGHNQEIAWGLTNSGADVTDLYLEKITGEGYQYDGKVVPFETREETIKVAGGDSKKIVVRETNNGPLLSDRDDELVKTGKKATVETAAPDRGDGYGVALRWTALDAGTTMDAVFAIDRAQNWSEFREAATLFDVPSQNLVYADSEHIGYTLPGKLPVRAEGHDGSVPAPGWDPKFRWTGEYIDQDELPHEYDPERGYIVTANQAVVDEDSYPYTLTTDWGYGTRSQRITSLIEQKIKDGGKISTDDMRQMQLDNSSEMAKLLVPQLLKIDVADKDVREAQKLLEGWDYTQDADSAAAAYFNAVWRNVLKLAFGNKLPKELRVKGQCLWVDPVNTTGPADATNKVYECGQRDADQAQPDGGDRWFEVVRTLLDDPKSDWWSTPKYGTRKGADKNRDDLFKRAMVDARWELTAKLGKDIDSWNWGRLHRLFLKNQTLGTEGPGFLKYALNRGPWKLSGGEAAVNASGWNAAGGYGVIWVPSMRMVVNLGDLDKSRWINLTGASGHAYSAHYTDQTDKWAKGELLPWSFSEKAVDESTSDTLVLKP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05232 Penicillin acylase family protein MSAETYRDAWGIPHLRADSPEELARAQGRVTARDRAWQLEAERHRAQGTSAAFLGPEALSWDRLARRARLADTARRCFIALEEKDPETAAWVRAYVHGVNEGLALHRGGDGPGDREGPGDREGSHPLDGSPRRDDPRRPPAPEFARAALAPGRWEPWTPLAVWLATHILFAGFPAKLWREHITARLGPDAVALFAADGPGTTGSNGWLLSGERTTTGHALIAGDPHRWIEDPGVYQQVHLSCPEFDVVGLAVPGVPGVAHFGHTGTVAWAITNAMSDYQDLYHERLRRTGAGVEALGPDGTWRRAARHTETIRVAGEGTVEVEVIETDRGPVVAGGPEGLDDGTPAALSLRYPPRVTSDLGFGALLPLLRARTVADVDRALDAWAEPVNVVQAADTGGGLLHRVAGRVPVRAEANGLRPVPAWEPGHEWTGWHTPPRAGLADGAAVMANQRGLATPLGVEFAAPHRADRIAALLAGRRRWSAADLSAIHTDTHLGSAGPLLAHLTALTGLGPEATDLRDRVLAWDRRMDARSTGAAAYAAVRAAVVRRLAAHPVLAPASVAPAYPEVLQPWLALVPRVAYALEHLLRADDLYGIDRAAVVRAALEEVAARPPAGPWGDTHRLTPWRALPDPAAPADAPALSGDHDCVLCTSSVPGLTDRAARGPAARYVWDLADRGNSRWVVPHGASGTPGSSHHRDQQPLWLAGELVPVITDFDRLTLICTHTHTHTSTEETDA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05237 Penicillin acylase family protein MAAGTSPSAGTTAAEPAEAAANDHCGGQCSDILPPGQNGNATLAQILLNQAFGTQPEHAEDQLGPYANLATGYTGLTNDKINTFFNDASFGVPDGQAASTLRPAGRDDVTIVRDKKTGVPHITGTTRYGTEFGAGYAAAQDRLWLMDLFRHVGRGQLTPFAGGAPANQGLEQQFWRSAPYTEADLEAQIESAAAKAGERGDLALADVDAYLAGVNAYIDASDRGRYFPGEYVLTGHKDAITNAGTIERFQRADLIALASVIGSLFGAGGGGEVDNALSLLAAQEKYGVAEGTEVWESFRQRNDPEAVLTQQDGSFPYLPTPDDPQGRALPDAGSAEAEPLVYDRTGSAAGASATGASTTAAQSATASARRGMSNALVVSGEHTASGHPVAVFGPQTGYFAPQLLMLQELQGPGISARGASFAGLSMYVELGRGQDYAWSATTSGQDIIDTYAVELCQDDYHYLHRGTCTPMEKVERHNAWKPTVADSTAAGSYTMRVWRTAYGPVEYRATVGGKKVAYTTLRSSYLHEADSIIGFQMLNDPDYLDGPERFKGAVQHINYTFNWFYADSEHTAYYNSGDNPVRADGVDAEFPVWARQAYEWRDWDPAANTARYTGASAHPQSADQDYYISWNNKQAEDYPAASWGNGSVHRGNLLDDRVKKLVADGGVTRTALVGAMAEAALADLRAEDVVPGLLKVVESAPVTDPAAKTAVDGLKAWLSAGGLRTETSAGSGKYAHADAIRTLDAWWPLLVKAEFEPGLGTGLYTAFTRNLPVDESPSAAHGPTGAHAGSAFQYGWWSYVDKDIRAVLGQNVKGPLAHPYCGDGDLAACRDTLVTTLKEAAGRTAGQVYPGDENCSAGDQWCADSVIHRTLGGIKHGGIGWQNRPTYQQVVEFTSHR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05317 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer 16.5 % inhibition of cell proliferation at 1 nM
dbacp05318 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer 14.2 % inhibition of cell proliferation at 10 nM
dbacp05319 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer 16.8 % inhibition of cell proliferation at 100 nM
dbacp05320 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer 21.7 % inhibition of cell proliferation at 1 µM
dbacp05321 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer 27.9 % inhibition of cell proliferation at 10 µM
dbacp05329 Peptide 5 fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin Not specified MTT/MTS assay PTC Colon cancer ED50 : >10 µM
dbacp05332 Peptide ABC transporter permease MPGRITPRRPGPHRRSGRPRATALGAALATVLVPALSACGGDAASASGDATLKWTSTYFPAHWDPVVGGSGAQFRELSLVYASLTRTDESGKAVPDLAESWEYNDEGDRITFHLRPGLKFSDGEPVDGAAVKAAVERAQKQKNSALFGDLTSIESVDAKGLDATVNLNQVDYQIPQLLGQRVLQIASPKAAAAPEKLDQNPVGAGPFTVTQIVPGTKAVLKKNPEYWDADNIHIDNVELTSAPDASTVVSGLQTGVYNFADIAPSQADAAKKAGLDVFVQPGFNASNISLNVNKAPFDNDKVVDAVRHAVNRQEFVDKLTFGYGEATNQPFPKGYVAYDPESEDAYPYDPAKSKKLLAEAGYRSGDIKLDLVIPEEDPQAEIVQSQLAAVGITVDIRIDKNWSTPFFAKDLTFSLYGTTGRDSAAQTLTAHFGPDGPLNLSTPYEPEGFESAIAKVRQTPLDAPEYPQVLQEATRAGLDSKALVFTYSQPNLIAKSKSVSGLPKNPAHLDWTGVTIGGKGAAS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05337 Peptide ABC transporter substrate-binding protein MKSSVSSTRRAAPGRPRAVGAMLLAGLVFVSSGCAVAGSAGGDAGRADGRTLRVVLTQEPPTLEPCEASLTGTGVVVRSNITEPLVERDPASGELDPLLATGWKQTAPRTWTFDIRSGVTFHNGAPLTAEDAAFSIDRAVNSDLACNVEGYVFGNDDLDVEAVDDHRLTVTTEEPDPILPLRISFVEIVPRTTDTEAKVRVPVGTGPYAVGSWKAGAAISLDRYDGYWGEAPDFARARYVWRSDASVRAAMIDKGEAEIAVALDPTEAGKDTTAAYPNNETTALRLDGREAPLDDLRVRRAVDLAVDREGIVDALLGGLAEPAGQLVPPGVVGHNDEISPTRQNVTEARALVERAAADGVPTGRQITLVARNGMFSGVSETAEALQYQMQQIGLNVKVRMADTATHLQYQLRPLPEDVGPIALLIMHGNQAGDAGFTTSQYLLGDGPQSTFGTEALDRRITEAGALSGEKRQRAFAGLLAEQNEDVVQYAHIAHMSGLLGLSRSIRYEPNSATGDELRLSEVHPAKGAKD Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05342 Peptide ABC transporter substrate-binding protein MSPARTAARRRRALAVGACAAVGVLLSGCAGGVSAPSGSKNEINYALPANFTPNWIVPIGTPGHLNTNNASISQSLWEPLIAYDGSTGEIGWNKDNSLATEAEFAADNKSVTVTLGDRHWSDGEPVTARDVEFWFNLVRENKKSWASYSPGKAPDVWTSFRTLDDRHFTLDFDRAYNRQWMLANELSMIRVMPQHAWDRTSDSGDVSDLDRTPDGAKKVWTYLIDAGKKISRYASDPLWKTVSGPYRLKSFSTSGRVELVENEKYDGGGAAHVKQVNLLSFTTVAAEENALRAGTVDYGYIRASDLGIKKSFTDLGYHVERWSGWAVTYMPYNFNNPEMGAVFRQPYARQAVQMSVDQKTLAKVLYNGTAVPTYGPVPQGQASAFLSGEQKAEPYPFSNSRARALLTDHGWSERDGTMVCTSPGEGAGHCGEGVEEGTEFRMRVLYQSGSTETDnMMSALQSSFEETGIDFDIKTAPVNSVLSQTGQCEEDDPACDWQLSFFGSAGSWYFPAYPSGDALFASGGGSNFGNYSNPEVDELIDRTTTSSSPDAMLDYSKALAEDLPVIWLPEPDYQVSVIRDGLGGFAQDSLANFHPAMWAWTE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05347 Peptide ABC transporter substrate-binding protein MKILISADMEGATGVTWPADVLPGTPQWERCRSMFTSDVNAAVQGFLDGGADEVLVNEAHWSMRNLLLERLDERTQMLTGRHKALSMVEGVQHGDVDGIAFVGYHAGAGMEGVLAHTYLANQLTGVWLNDVRASEGLLNAHVVAEYGVPVVLVTGDDVACEDALGYAPEARKVAVKDHVSRYAAVCRTPARTAADIRAAAKEATPLAVRHEPVTGGPFTVAMEFDAEHLAAASTVVPGVAQVGERKVAYTHDTMFEAIRTFKAVTTIASAAVEEQYG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05352 Peptide chain release factor 1 MFEAVEELVAEHADLEKKLADPSVFADQANARRLNKRYAELTPIVATFRSWKQTGDDIGTARELAADDPDFAAEVKELDKQRDELTEKLRMLLVPRDPSDDKDVILEIKAGAGGDESALFAGDLLRMYLRYAERVGWKTEIIDSTESELGGYKDVQVAVKTKGGQGATEPGHGVWARLKYEGGVHRVQRVPATESQGRIHTSAAGVLVTPEAEEIDVEINPNDLRIDVYRSSGPGGQSVNTTDSAVRITHIPTGVVASCQNEKSQLQNKEQAMRILRSRLLAAAQEEAEKEAADARRSQVRTVDRSEKIRTYNFPENRISDHRVGFKAYNLDQVLDGDLDSVIQACVDADSAAKLAAA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05357 Peptide chain release factor 1 MDLAFLHPLYEHQGPWASVYLDLSRHTEDTPHERELTAAAVARELAEQGADDATCEAVREAVDGLRHASDPHGRALFARAGEVVLDPRLARPPYGGTTADWAPLPHVAPLLDLAGEDPVCVVAYVDRKGADFELRSALGSSDAGGVTGRQWPVHRTSSADWSERHFQLRVENTWEHNAAEIADALAVCQEETGADLLILVGDDRERRSVHERLPKRLQGRVAEASRGAGSRLLDDEVERLRADHVRSRAREDLDRFLAARSPDDEGRAGAAEGVPALVEAAREHRIDELLVIPDAPDTHREVWIGEDADQLAVRRTELKTLGEQNSWSARADDALLRSAVMTGAPAISVTPVLPPETAGKAPVGGLGALLRWK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05362 Peptide chain release factor 2 MAVVDVSEELKSLSSTMESIEAVLDLERMRADIAVLEEQAAAPSLWDDPEAAQKITSKLSHLQAEVRKAEALRGRIDDLGVLFEMAEEEDDPDTRAEAESELAAVRKALDEMEVRTLLSGEYDAREALVNIRAEAGGVDAADFAEKLQRMYLRWAEQRGYKTEIYETSYAEEAGIKSTTFAVQSPYAYGTLSVEQGTHRLVRISPFDNQGRRQTSFAGVEVLPVVEQTDHIEIDESELRVDVYRSSGPGGQGVNTTDSAVRLTHIPTGIVVSCQNERSQIQNKATAMNVLQAKLLERRRQEEQAKMDALKGDGGNSWGNQMRSYVLHPYQMVKDLRTEHEVGNPESVFNGEIDGFLEAGIRWRKQREK Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05367 peptide chain release factor N(5)-glutamine methyltransferase (EC 2.1.1.297) MPSSPPGPATPAGTPSGDVLARAVATLRGAGCVFAEEEARLLLDAAPAPADLERLVGRRVDGEPLEVVLGWAEFCGLRVRVEAGVFVPRQRTRFLVDAAAELAGRPGAVVVDLCCGTGAIGAAVAARVPGIELSCADVDPAAVRCARLNVGPDARVYEGDLYDALPDALRGRVDVLVVNAPYVPTDEIAMMPPEARDHEPRHALDGGGDGVEVHRRVAAGAPAWLAPGGTLLIETSEEQAPLTARAMKDHGLVPRVSTNDEMYSTIVAGTRAVR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05378 Peptide deformylase MRHGSIPGAHGRVRPLALLGDPVLHAPCAEVTDFGPELAALVEDLFATMYASRGVGLAANQVGEGVRVFVYDCPDDEDERHLGHVVNPRPVEAGGVVVRGPEGCLSLPGLEAGVERYDEAVVTGVTVTGEPVTVRGTGFFARCLQHECDHLAGRVYPERLSGLRHRRLMRKAARAPWSR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05383 Peptide deformylase MPSVFVQGRPTASYPPFAPEARRGSVRRVTEVGEEVLHRPCRDVTEFGPDLAALIDDMFRTMYVAEGAGLAANQVGLGLRLFVYDCPDDEGVRHVGHIVNPVLDALAPAARRLLDEGEGCLSVPGAVMAVPRPDRAVVRGLDKDGAPLLVEGTGYFARCLAHETDHVNGHVYLDRLSARERKTALRQSADRREEVFARRSANAAAFA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05388 Peptide deformylase MAQQDTDQQHTGVLPVDDEGFVVDTEECEQREADWRGRGTSRPITVVGNPVLHKECEDVTDFGEEFQQLVADMFASQRTAEGVGLAANQIGVSKKVFVYDCPDDDGVRHVGVVCNPRLVELPADRRRLDDSNEGCLSVPTAYAALARPDFAEVTGQDEKGNAVRVRGTGYFARCLQHETDHLYGYLYIDRLSKRERKDALRQMAENEPRYPVVAND Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05393 Peptide deformylase MGTPSDRAPLAERVEELLALGGPLPIVAAGEPVLRRAAEPFDGQLAPALLARFVEALRLTMHAAPGVGLAAPQVGVGLRIAVIEDPAPVPEEVRAARGRVPQPFRVLVNPSYEPVGAARAAFFEGCLSVPGWQAVVARHAEVRLRARDEHGRAVDEVFTGWPARIVQHETDHLDGTLYLDRAELRSLASNASMADLWSQPTPERAASALGFELPGRPGPSGSPGLPGSAS Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05423 Peptide methionine sulfoxide reductase MsrA MAAQTQRAVLAGGCFWGMEELIRRLPGVTATRVGYTGGDVPNATYRNHGTHAEAIEILYDPEVTDYRAILEFFFQIHDPSTENRQGNDIGLSYRSAIYYVDDEQKRIAEDTIADVDASGLWPGKVVTEVEPAGPFWEAEPEHQDYLQRYPNGYTCHFPRPGWRLPVRTEG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05429 Peptide transporter permease SapC MKLTTAVLAAGAAVSLTTAVVGATRLRQNARHQAERNEAFLTRNQLDWLAQMSTNPDLAKLWAPEDMDVEEYMQLLAANRLICILSVRDRLGFVRTGHLPWHAAKLMENDACRRYWQRFGDLRAEEAEGDEQGEHFTRVLDQAAKQHPRAQAAAT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05448 Peptide-binding protein MAWSEGGFGRLGAAVWSADPWYGGSRSAHVFNRKRRLRRVVAIVSLSSLATGCGLLSPDDPEDDGPIVVGTTSAPSTLDPAASWDGSWELFRNVYQTLLSYPDGATAPEPDAAEQCAFTDSANQVYRCELREGLTFSNGHSLDALAVKHSIDRIKEIDVNGGPAGLLGSLERVQAPSAREVVFHLDKPDATFPFVLATPAMSIVDPSGYPADALREDGEAVGSGPYTLRSYEDGVRAELVRNDRYQGFAERRNNAVTVRYFKDSAGMVEALRDDDIQVTYRGLAADDVIGLQAKDAGDEALRLVEGSGTEISYLVFNPEDPWAGRREVRRAVAQIVDRATLAHEVYQDTVDPLYSMVPKGLTGHTTGFFDDYGDPSVPKARKLLTEAGITERVPLTLWYTSDRYGSETATGFKEIKRQLDASGLFEITLESRPWKTYVTGYQKGEYPVFGRGWSPDFPDAENFIAPFVGEQNALGTPYPAPEITGELLPRSRRESDRADVEREFERAQQIIVDDARLLPLWQGKQYVAVSTEISGVEQAMDPSTIMMVWQLSRKTGW Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05453 Peptide-binding protein MNRKTLVLPAVVGLLAPVLAACGGSDGGSGGGDAIAVGTTDRFTITKDVPAPFDPAYAYDIGAWNIMRHTAQTLMTQPRGDGEPVPEAAQQCGFTDTGNERYACTLRDGLKFSNGDDLTAEDVKYSIDRAVSLEADTEVGKVLLSTVDTVETKGDREVVFHLKTADATFPYKLSTPVASILNKEQYAKDKFRDGFDLDGSGPYEMKSESKNGVLSKIVFTKNPTYKGSVKVNNDKVELVSFEDAESMGNALDKGDIDVMTRAMAPEQVKKLSDSSQGAVKLVEVSGLEIRYLGFNVDAASVEDKAVRQAMAQVINRAELVSRVYGSQAEPLYSMVPAGITGHSNSFFNKYGDPSVAKAKQTLKSAGIDSPIELTLHYTTDHYGAATKLEFEELQRQLNASGLFDIKLDGKPWDIFRPAERRLEYDVFGMGWFPDFPDADSFIAPFLDEDNTLKSPYLNQKIIKDLIPESRSEADRLSAADSLTEIQDITAADVPLIPLWQGKQYVAARDDVTGAAYLLNSSSTLQLWELGRGVSG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05458 Peptide-methionine (R)-S-oxide reductase MSYDVEKPDEQWRKELAPAEYAVLREAATEPAFTGEYTDTKTEGVYSCRACGAELFTSTTKFESHCGWPSFFDPKDTDAVELIEDRSHGMVRTEVRCARCGSHLGHVFKGEGYPTPTDQRYCINSISLRLEPERG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05475 Peptidyl-prolyl MAEQLYATLKTNHGDIEVRLLPNHAPKTVRNFVELARGEREWTNPETGEKTTDRLYDGTVFHRVISGFMIQGGDPLGNGTGGPGYQFEDEFHPDLSFNKPYLLAMANAGPGTNGSQFFVTVSPTTWLNRKHTIFGEVAGEAGQKVVDAIAALPTNPRTDRPVNDVVIESVTVETRQG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7µM
dbacp05480 Peptidyl-prolyl cis-trans isomerase (PPIase) (EC 5.2.1.8) MSNSKVYFDIDIDGQDAGRIVFELFEDVTPRTAKNFIELSTGEHGFGYAGSSFHRVIPQFMLQGGDFTAGNGTGGKSIYGAKFEDENFKLKHTEPYLLSMANAGPNTNGSQFFITTVVTSWLDGKHVVFGKVVEGTEVVDKIEGYGSSPQGTTSAKITVRASGKL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05493 Phenyloxazoline synthase Mycobactin synthetase protein B MNIPELLARYADEGVVLWAQDGQLRFRAPQGRLTDTHRAELRTHKQDILRHLEAGRPALRPDPDSRHEPFPLTDIQAAYLIGRTDAYAYGGVGCHAYVELDHPELDVERVTAVWRELVERHDMLRAVVHHDGYQQVLADVPDLHVACDDLTGLPAADAEAELARTRARLSARETPTDQWPLFDVHVSRTAGRAVLHLSFDMLVVDHASLRILLAEFRHRYGGGVLSAAPRITFRDYVLARRAQTGIDGHARDRAYWTERLDTLPPAPELPLAEPWEAAVSASTGTRGAPTDAVTFRRLEVPLSAADRERLTERAARRGLTVSTALLTAYAETVGRWSRTSRFTLNVPTVDRPDLHEDIGRLVGDFTSLELLAVDLDTPAAFAERTGALGQQLLEDLAHPLFTGSEVLAELSRRAGAPVLMPVVFTSALGTGGTAEGVPPEVAHAATRTPQVWLDCQVMHRGDALILSWDVREGALAHGVAEDMFGAWTSLVRLLSAEGEEGDAAWDAPVDIPLPAAQRDRRAAANATGGPLPDALLHEPLLDRARTTPDAIAVRTPETALTYRQLADRAGGVAETLTASGLRPGEPVAVWTDKGWEQVVAVLGTLMAGGAYLPVDTAQPPARRDTILADAGVRTVLTQSWLAETDDLPATVSAVAVDLVPAAPATREPRTAPRRDPDDLAYVIYTSGSTGTPKGVMISHRAALNTVQDINRRYAVTDRDRVLGIAGLGFDLSVYDLFGPLAVGATLVLPRADRRGDPSHWAELVRDFGVTVWNSVPGQLHMLCDWLRSEPPADDGTLRLALISGDWIPVALPDQARALLPGLEIISLGGATEGSIWSIAHPIGEVDTDRPSIPYGTPLTNQTFAVLDRHLRPRPEWVPGELFIGGAGVALGYLGDEARTAERFLTDPRTGQRLYRTGDLGRYLPDGTIEFLGREDAQIKIRGYRVELAEVEAAVQAHPAVAAGAVVVDDSAAGGRRLAAFVETARRDGDRRAAPGARQAREAAADAVREASAAVDGARLADFLAALDEVALDGMTRVLAGSAVFEDGAARTADEVGTALRATPRHRHIVRRWLRALAARDRLTHRDTDDTYSGLVAVSGPDTERRWRLAADLEHEVGWSSELLTVMRTCAERLPELVAGDVGIRDLLFPGAATDAADAAYRDNLAIRHLNRAVVAALREIAASHTGEERLRILEVGGGVGGTTGELVPVLAEYGVDYLFTDPSAFFLNEARERFADHTWVRYQRFDVDQDLRGQHLPPNTFDVVVCANTLHAAADADAAVGRLRELLVPGGQLVFVENTRDENLPLLVSMEFLEVAGRPWTDVREHTGQSFLTHPQWRELLGRHTASDVTSLPEGQDALARTGQEVFLATMKDDRHHVPTGELARTAATRLPEYMLPAVWQVVDTLPRTANGKTDRARLVDWLPRESAPVVVDERPRDELENSLADLWSELLAVEGVTRNDDFFDLGGDSLLVARMVGRLRERVPRAADLEWEVVLRHMLRRPTVAGLAGFLRSLADPKDAPAPGAVRTDPVIHLHGARSDDEPTTVLVHAGTATIMPYRALITEIRRRSPGLAEVVGVEVPDLNGFLAAPPQGLIEQLAADYARALTADGRSRFHVVGYCLGGLIATEVARNLAESGAEVESLTVISSHSPRFRLDDELLAEYSFAVMMGIDPAELGFPDDQYRVAAAADAVLASSPGILPDGGLAALPEEFEDVAGRFRSLAEVPRATRIARMCEAVPASAGSYEPDHMSRLFLAFRQSVFAITRYTAEPYAGDITFLRHDGAYPFPGSKDAVTTYWEELTLGDLDIVDIGGDHYSCLSVEHAPGILKTLGELTRGAITR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05498 Phenyloxazoline synthase mycobactin synthetase protein B MSDEAVVEARTAEGDAGRRGPHTAPAVRDAVARALDLAPQELDDDRDLFELGLDSLLLMSLVGAWRREGSTVTFQDLTRVPTLAAWTALLARAPHGDAPAAARPAPVPRQADRSVPRQADRATERSAPQQAERSAPRRSVRQADRQQNRQADGAAEPFPLATMQHAYWIGRQDGQPLGGVAAHFYVELDGREVDPARLDAALRALVHRHGMLRAVFDEEGRQRYGATGAPLTVHDLRARTPEEADSALESLRERNTHARGDVAGGEVFRAALCLLPDGRTRLQIDLDMMAGDALSLRVLLSDLRRFYACPDDPPPVLGLDYRRYLAEHDARRRAERERDAVWWRERLHELPRGPRLPTTVDPLTPVGAGDTALTRSRRLHHWLGPDDKAALIKAAGRHGLTPAAALATAFAETVAAWSDSRRFLLNLPLFDREMFSPEVAHLVGDFSSSVLLDADLGAPLPFARQARRLQERLQEGISHGAYGGVEVLRDLARAEGAPVLAPVVYTSAIGLGEIFEQDVQKSFGRPSWIISQGPQVYLDAQVTELDGGLLLNWDVRDGVFEAGVPDAAFDAYRRLITCLRTDPDAWDRPVDGLLAPGVLARRAVAALPPAPVPHRALHTRFFELAETEPDRTAVVRTTGAPLTYGQLADTARRIAALLGDHGVGEGDTVAVTLPKGDGQIGAVLGILAAGAAYAPVGVEQPAVRRRRIHSVAGAAAVLTDRAHADLCADAAAPAPVLLVEDAPAAGPAPVVLPDPGLPAYVLFTSGSTGEPKGVEVPHRAVVNTVEAMAEQLGLGPDDRTLAISALDFDLATWDIFAPLSLGGQVVAVGQEHRRDAHHWAELVRTHGVTLVQCVPALLDLLMAAGEDAAGGEGLGTSPRMVLLGGDWVGLDQPARLRALVPGCRFVALGGMTEAAVHSTVFEVTETDPAWKSVPYGVPLRnMRARVVDGRGRDCPDMVPGELWIGGPGVASGYRADPARTAERFVEYDGERWYRSGDLARYRPDGVLEFLGRADHQVKIGGHRIELGEVESALESDPAVRHAVATVLDTPVRRLAAAVSSRDGAAPEPDAVRDRAAERLPAHMVPERVLVLDALPLTENGKLDRAAVRRALTEAAGHATARASAPEGPVETAVAAEWSDLLAVDRVGRESSFFLLGGDSLVATRMIGRLRAAGFPDARVADLFARPVLRHFCETLRAGTADGREQEPPAPALVPDPDHAHEPFPLTDVQAAYHTGRDPRFALGGVGTWHYTEFDGTDVDLDRLERAWNTLVRRHGMLRAVVEDGHQRVLPDVPPVRIPVREATAADAPEALAELRARLSQQVRDPARWPLFAVEAVRHPDDGDGHGDGDGTVRTRVGVGLDYLVLDALSITTLYAELNALYADPDHQLPPVDVTFRDYLTRLPADPASVDRARAHWQARLAELPPPPALPYDRDPATLDAPVFTRRRLTLSAEDWQAVKRRAARHGLTPSTVLLALYGEILAAWSGTDAVTVTLTLFNRRDVHPHIHRVLGDFTSLSLAGHRREGASWLAAALALQHRQAEDLDHADVPIDWLLREFGRRTGTVDAAAPVVFTSAVGVGDATLARAGTGLPEKVWGISQSPQVCLDNQVTEESGGLVVTWDAVEELFAEGVLDAMFDAHARLLRHLVTGDWEAPLPDPLPAAQHDRRAAVASGAALEPVAPRLLHEAFFAHAAGRADRTALVTTAGEELSYGALAERALRTAAALADAGVGPGDLVAVTLPKGPDQIAAVLGVVAAGAAYVPLGLEQPAARLARVRAAARFRVVVGEWPDTGDGTAPRALSFARTQRSEPWRSPRETSPEALAYVIFTSGSTGRPKGVEISHAAAWNTVADISARHGIGAGDRVLALSALDFDLSVYDLFGLLAAGGSLLLPTEDQRREPARWPDLVDRYGVTVWNTVPALLDLLLDADEQGTGGLRGLRTALVSGDWIGLDLPGRLRARTARPCAFVAMGGATEAAIWSNTLTVTDVDPRWASIPYGRPLTGQHYRVVDRDGRDCPDWAPGELWIGGAGLARGYLAEPERTAEKFVVRDGRRWYRTGDLGRFRGDGLLEFLGRLDTQLKIAGHRVEAGEIEAALEAHPAVARAAVVAVGERTAKRLVAFAVPLATPATATEPPTADDLLGHLADRVPAYAVPSRIALLPALPLTANGKVDRKALTDTAGPAPVPAGAEPPRGGTETALAELWREHLPEPVRDRNANFFTLGGGSLAALRLLTAIERRLGAAVPVRRFFAAPTVAALAADITRTLAAHGTAYETGEL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05551 Phylloseptin-PHa FLSLIPAAISAVSALANHF Northern orange-legged leaf frog Disruption of the membrane MTT assay, Lactate dehydrogenase (LDH) assay HCT116 Human colon cancer LD50 : < 5 µM
dbacp05599 Polysaccharide deacetylase MSSEGFGLPKESWRWPETAWRGHVDAVRAGRRLVPDRWPGGARVAVALSFDSDHETIPLRDGETSPGRLAQGEYGARAGAPRILRLLERYGVPATFFMPAVSALLHPEEARAYTRDGHELAVHGWIHERnMLLDREEERELTARALDTLTTVTGQRPVGIRTPSWDFSDSTLDIMLELGFAYDSSLMADDEPYEIVAGGRSTGLVEIPVDWIRDDAPYFTMDRYGSVRPHSRPRGVGEIWRDEFDAAYHDGGVFQLTLHPHVIGHRSRLVVLRELLDHIASHQDVWFATHAQLADAARSMLPASGPDRP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05604 Polysaccharide deacetylase MITLVRRAAALCVLGAALTACGTTAAEVAPRPAPSAPAPSSSASRTPTPTLAPGPGGLTPVFEHGPRTDGTNHGEQDGTRDGKLIALTFDADMTADQGPRAASGERFDNPQLIAALRELKVPATVFMTGRWAEEYPDEARSIGRDRKFEIANHSYSHYAYTDDCYGLPTVAEDDMRADLERAYTAFEKAGVPNPMPYFRFPGGCYDKAALKELSATGVTAVQWDVVSGDAFATDADAVTRQVLDGARPGSVVVMHCTRSAAPVTEEVVRAVVPELRSRGYRFVKVSDLVGAANGRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05609 Polysaccharide deacetylase family protein MPVLMYHAVAAGPNDATRALSVTPQAFAEQMAAVADRGRTPIGTAELAAAWRSGRPLPRRPVLITFDDGYAGVHRHALPVLARHGFPATLFVSTGWLRGPHDTGGAPDTMLDWAQVRELAAAGVEIGGHSHTHPQLDQVGEERLRHELIHSKEIVADQLGVVPASFAYPYGYSDRRVRRAVRETGYAQALAVGNGLARRAQGPYALRRVTVRRSTGTEEFARLVEGRAIARTFALDRALTKGYAVLRRTRQARRKVLGAGA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05614 Polysaccharide deacetylase family protein MYHSVGDRSDDPYRITVTPDRLEAQLRWLRRRGLRGVPVAELLAARAGGDGGDLVGLTFDDGYADFVEHALPCLRRWGCGATLFVLPGRLAGDNAWDPLGPRKPLLSADGIRHAAAEGVEIGSHGLTHVDLTTADDAVLTAETAGSRALLAELTGTPVTGFCYPYGTVDARAADAVRAAGYTYACAIDPGPLTGPYALPRVHVGQRDTSVRLLLKTRLHRLRRRASAGV Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05619 Polysaccharide deacetylase family protein MDDPPAWIAEFTVTPKEFAAHLDAIVGSGRTPVTIGVLADHLAGRAPLPPRPVLLTFDDGFADLPGPTAEALAERSLPATAYLTTGAIVPGGRSLLPPAPMMTLAAVAGLERSGMEIGSHTVTHAQLDTLPGTDLAYELRTSKAVLEDALGHPVRHLAYPHGYNSAKVRSWSARAGYETATAVRHALSSERDERYRIARLIVRRGHTVADVESWLAGGGVRTAPYRDGPKTVAWRWYRRGRAMVRGPEFAG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05624 PPL-C VSVSHFQKVWVV Not found Not specified Not specified CT26 Colon cancer MIC : 11 mg/kg
dbacp05628 Prepilin peptidase MGPGLGVDLDLLVVLVAALWGAGAGALLPRAVYRFAAPSGEAWRERCPGEHPVRGWLGRARCAQCTGERQAYGPGAGLLAAVTAVVCVALAGATGARPEVAVWLLLAPVGVLLAAVDLRVRRLPDPLTLPLAGAALVLLGLTALVPEHAGEWTTALLGSLALGAGYLVLFLINPAGMGFGDVKLALGAGAVLGWYGWPTLILGTFAGFLLGAFYGGVLLVTRRAGRKTAIPFGPFLIAGAFLGLLVGAFTA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05635 Proline iminopeptidase MGLYPEIEPYDHGMLDVGDGNHVYWETCGNPHGKPAVVLHGGPGSRATPGHRRYFDPAAYRIVLLDQRGAGRSRPRASAHDTDMGVNTTAHLMADLERLRAHLGIERWLVWGVSFGSFLGLRYAQTHPGVVTELVLTGVATGSNREVDLLTRGLGKLFPEAYEQLLAGLPPDEREGNHAAAYHRLLESPDAAVRERAARAWTDWETATIPAPPRSVARYEDPAFRLGFARTVTHYWGNDHFLGDGNDEGVVLRDAPLLKGVPGTLVQGSLDFGNLLGTVWRLHHAWPDSELVLVDEAGHDAGAVGDEVLVAATDRYARGAA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05640 Proteasome accessory factor PafA2 MGIETEYGISVPGHPNANAMLTSSQIVNAYAAAMHRARRARWDFEEENPLRDARGFDLARETADSSQLTDEDIGLANVILTNGARLYVDHAHPEYSAPEVTNPRDAVLWDKAGERIMAEAAERAAQLPGAQPIHLYKNNTDNKGASYGTHENYLMKRETAFSDIVRHLTPFFVSRQVFTGAGRVGIGQDGHEHGFQLSQRADYFEVEVGLETTLKRPIINTRDEPHADAEKWRRLHVIIGDANLSEISTYLKLGTTALVLSMIEDGFIAVDLAVDQPVRTLHQVSHDPSLKHLVTLRSGRTLTAVQLQMEYYELARKYVEERYGADADDQTKDVLGRWEDTLNRLENDPMSLAGELDWVAKRELMEGYRRRDNLDWDAPRLHLVDLQYADVRPTKGLYNRLVDRGRIKRLLDENEVERARTKPPEDTRAYFRGRCLEQYADDVAAASWDSVIFDLPGRDSLQRVPTLEPLRGTRNHVKELLDRCRTADDLVRVLSGG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05645 Proteasome subunit beta MEANTRSTGRLPAAFLTPGSSSFMDFLGEHQPEILPGNRQLPPVQGAIEAPHGTTIVAVTFPGGVVLAGDRRATMGnMIAQRDVEKVFPADEYSAVGIAGTAGLAVEMVKLFQLELEHFEKVEGAQLSLEGKANRLSTMIRSNLGMAMQGLAVVPLFAGYDVDRGRGRIFSYDVTGGRSEELNFATTGSGSIFARGAMKKLFHDELTEEQATTLVVQALYDAADDDSATGGPDVARRIYPIITVITEDGFRRLGEDECSALARSVLERRLEQPDGPRAALL Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05655 Protein GPR15LG MRLLALSGLLCMLLLCFCIFSSEGRRHPAKSLKLRRCCHLSPRSKLTTWKGNHTRPCRLCRNKLPVKSWVVPGALPQI Mouse Not specified Not specified Not found Colon cancer Not found
dbacp05656 Protein GPR15LG MRFLALTSLLCILLLCLSFFSAEGRRHPRNPAKPGKIRICCPRLPGPDLMPQKGHHMRICRPCKFKQKPQLWVVPGALPQV Pig Not specified Not specified Not found Colon cancer Not found
dbacp05761 PUMA BH3 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified MDA-MB-231 Colon cancer Not found
dbacp05762 PUMA BH4 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified HCT116p53–/– Colon cancer Not found
dbacp05763 PUMA BH5 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified HCT116p53+/+ Colon cancer Not found
dbacp05764 PUMA BH6 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified GLC-82 Colon cancer Not found
dbacp05765 PUMA BH7 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified SGC-7901 Colon cancer Not found
dbacp05766 PUMA BH8 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified HEK293 Colon cancer Not found
dbacp05767 PUMA BH9 LRRMADDLN BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis Not specified 2BS Colon cancer Not found
dbacp05770 Putative ATP-grasp-modified RiPP MFAHSDRLPSGTPLPNGISTPTPWGLRRMAPYPALAPSYARVELDPATQTGRYFDASGAVLEMPGHGTSTGTRPATNTGNSSDGAGPGGNGGGDQDSGNDTDQ Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05930 Release factor glutamine methyltransferase MNLLLAEVAQAAQRLADAGVPSPRTDAEELAAHLHGVKRGELHAVPDADFDARYWEVVARREAREPLQHITGRAYFRYLELQVGPGVFVPRPETESVVGWAIDAVRAMDVVEPCIVDLCSGSGAIALALAQEVPRSRVHAVELSEDALVWTRKnMEGSRVDLRQGDALTAFPDLDGQVDLVVSNPPYIPLTEWEYVAPEARDHDPQLALFSGEDGLDLIRGLERTAHRLLRPGGVVVVEHADTQGGQVPWIFADERGWADAADHPDLNNRPRFATARKALP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp05936 Retro LGGIVSAVKKIVDFLG Amphibian skin secretions Penetration and disruption of the membranes Sulforhodamine B assay Colon tumor cell line Colon cancer IC50 : >10 µM
dbacp05977 rRNA methyltransferase MNRPVPVPPLADVLRAALAELVDGLPPRQAGRAVERLIGHYRGDTPTDAPILRDRADVVAYAAYRMPATFAAVRSALDAFADAVPGWAPGSHVDVGGGTGAATWAVGDTWAGPRQVTVLDWAEPALALGREIAAAHPALRDVRWQRSRIGAALTVEDTDLVTVSYVLNELTSADRAALVDAAASAARAVVIVEAGTPDGYARVIEARDRLVAAGFHVAAPCPHSAACPIVPGTDWCHFAARVSRSSLHRQVKGGSLAYEDEKFSYVAATRLPVSPAPSRVVRHPLIRKGQVLLDLCEPDEQLRRRTVTKRHGDLYKAARDAVWGDAWPDAANPPTE Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06015 S9 family peptidase MGEPVRTLSYGSWPSPVDAALAAAHDGRPDEVGFVGDEVWWTAPRPAEGGRRTLVRRHADGTEEAVLPAPWNVRSRVIEYGGRSWAAVTTDAGPLVVFVNFADQRLYSFAPGGDAPRPLTPLSAVGGGLRWIEPDPRPEHGEVWCVLEEFTGEGPTDLRRVLAAVPLDGSAADDRDAVRELTAERHRFVTGPRVSPDGSRAAWLAWDHPRMPWDGTELIVADIGPEGTFRDARAVAGGPEESIAQADWAPDGSLLYASDRTGWWNLYRDGRPLHAREEEFGGPLWKLGQRWFAPLDSGLIAVLHGRGAAVLGVLDPETGEVVDAAGPWTEFAPALAAHGERIAGVGAGAHSGFEVVELDARTGRARVIGAPYEDATDPAYYPPSRIRTFTGPGGRDIHAHLHPPHHPGCRAPDGELPPYVVWAHGGPTSRSPLVLDLEIAYFTSRGIGVAEVNYGGSSGYGREYRNRLRGQWGVVDVEDCAAVALALAEEGTADPRRLAVRGGSAGGWTTAASLATTDVYACGAISYPVLDLAGWGAGETHDFESQYLESLIGPRAEVPDRYTERSPAEHAESVTAPFLLLQGLDDVICPPAQCERFLARMAGRGVPHAYLTFEGEGHGFRRAETMVRALEAELSLYAQVFGFTPPGVAALELTR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06022 San A-amide NA Marine fungus, Wilt of banana Apoptosis induction Not specified HCT-116 Colon cancer MIC : 0.98 µg/mL
dbacp06037 Sec-independent protein translocase protein TatA MFGRLGAPEIILILVVIILLFGAKKLPDMARSLGKSARILKSEAKAMKGENKSDDSAPADPPNPEQSAAQRTIQASPGDVTSSRPVAEPTDTTKR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06042 Sec-independent protein translocase protein TatA MLRNGLEPWHLLIVAIVFLVLFGSKKLPDMARSLGKSARILKSEAAAMKSDGGPAAERASGGGPAAPAPAATQPSGSAPAGDRDRARDR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06048 Sec-independent protein translocase protein TatB MFNDIGALELVTLVVLAVLVFGPDKLPKVIQDVTRTIRKIREFSDSAKQDIRDELGPEFKDFEFEDLNPKTFIRKQLDNDELGLKELRSGFDLKKEMAEVTDAVHGRDTEASSASSAAASSSGGRIDMSKKADLSKRPEKAEKPAADDRPPFDVDAT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06054 Sec-independent protein translocase protein TatC MLKPARSKEKDPEGRMPLAEHLRELRNRLAKALLAIVVVTVVAAFFYRDIINFLTDPILESVGCEKSFEELAEAKAGSEPCAQITINGLLGPFTLALKVSLTAGIVLASPVWLYQLWAFVAPGLHRSEKKYAYAFVATGAPLFLVGAYFAYAVLPTSAKVLIEFTPSDVDNLLPLDELLDLVTRMVVVFGLSFELPLLLVMLNLTGVLSGKRMLGWWRAMIMGITLFAAIATPSTDPLTMLMLAGPIWVLYFAAVTIALLNDRRKSRREALEPDDDEASDLDLTPEDVGEVEPVTTARALPEQATRDRVNGYDDVT Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06077 Shiva-1 MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG African clawed frog Pore formation at the cytoplasmic membrane MTT/MTS assay HRT-18 Colon cancer IC50 : 49.3 µM
dbacp06078 Shiva-1 MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG African clawed frog Pore formation at the cytoplasmic membrane MTT/MTS assay DLD-1 Colon cancer IC50 : >100 µM
dbacp06093 Signal peptidase I MDIETQPTERDRSSRSSGSEQPSDPAGPEERSRSALAGRIADWVPGGRITVTLLVLLLFLLLVSTFVLKPFQIPSGSMERGLRIGDRVLVNKLAYRFDGRPQRGDVVVFDGTGLFGHGDYIKRVVGVGGDHVVCCDREGRIRVNGRSVDESAFLYPGDRPSTVGFDVVVPDGTLFVLGDHRSGSSDSRDHLGSPGGGMIPVDRLIGRADWIVWPFGHATHLDRPDAYADVPDAEAGGVSGAAGGREASAVSGPAGEREAGGDSGAAGERAAGEDSGAAGGGVRRAESVDG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06098 Signal peptidase I MGSRGKPRGAPSSPAENLLPTGSRRTAAPSGGRSRAERRKLQRKVKRRRRRGAVKEIPLLVGVAVLIALVLKTFLVQAFVIPSGSMEQTIQIGDRVLVDKLTPWFGSEPQRGDVVVFRDPGGWLAGEQTTKQDDPVVVKQVKEGLAFIGLLPSDDEKDLIKRVVGVGGDKVKCCDTQGRVTVNGVPLTEDYLYPGDTPSRTPFEVTVPEGRLWVMGDHRSNSADSRAHQETDFGTVSEDEVVGRAMVIAWPFGHWTTLDEPKTYASVSDSVSGSTAAPRLSHRVAPYDPNAMIQLPIPAELPLVMGVVGLRRVRRGRWQRVRSWRGGCSGWRTVRTRRRGEPRTPRGDGRPGPGRSPGLRVRLRLRNRGRQGDRRTERRDPARGSGRDASRDAHPGQEAALLLEGAADPDRYRAGSRPADQDVPGPGVLDPVVLDGEHPADR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06103 Signal peptidase I MGGESTTRTAPRGGGAKNTPVGSRRGQRLSGLAVALGMVLFLGGFVWGAVVYRPYTVPTGSMTPTIAAGDRVLAERVSGSDVRRGDVVVFKDAAWADAPMVKRVVAVGGDTVSCCQKGKLQVNGKVIDEPYLPAGTPAEISDFQTVTVPEGRLFLLGDERDNSVDSTAHLTDAAGGTVSRGAVDARVDAVVWPMNGMLERPTGFETLGGLSSPGPLWTVVALVTGGAVLILGGAAYGPVAKRAEASRARRGTEAAGGR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06108 Signal peptidase I MGGTPPATPTPAKKQRSFWKELPILIGIALVLALLIKTFLVQAFSIPSSSMENTLQIGDRVLVDKLTPWFGSEPDRGEVVVFHDPDDWLAGEPTPDPNALQTVLSWIGLMPSADEKDLIKRVIGVGGDTVECNKTGPLKVNGKALNEPYVYAGNTPCSEDEQGGQFKVTVPEGKIWVMGDHRQNSRDSRYNQSDKNGGMVPVDEVVGRAIVVAWPMNRWGTLPVPETFDQDGLQARASAAALSVAPQGLAVAGVVPVVWWRRRRRAVSVETR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06113 Signal recognition particle protein MFDTLSDRLSATFKNLRGKGRLSEADIDATAREIRIALLEADVALPVVRAFIKKVKERSMGAEVSKALNPAQQVLKVVNEELVGILGGETRRLRFAKQPPTVIMLAGLQGAGKTTLAGKLGRWLKEQGHSPLLVACDLQRPNAVNQLSVVAERAGVAVYAPEPGNGVGDPVKVAKDSIEFARTKVHDLVIVDTAGRLGIDQELMQQAADIRDAVSPDEVLFVVDAMIGQDAVNTAEAFRDGVGFDGVVLSKLDGDARGGAALSIASVTGKPIMFASNGEKLEDFDAFHPDRMASRILDMGDLLTLIEQAEKTFSQEEAEKMASKLASKKGQDFTLDDFLAQMEQVRKMGSISKLLGMLPGMGQMKDQINNLDERDVDRTAAIIKSMTPGERQEPTIINGSRRARIAKGSGVDVSAVKNLIERFFEARKMMSRMAQGGGMPGMPGMPGMGGGPGRQKKQQKKAKGKQRSGNPMKRKQQEQEEAARRAAAAQGGGALGLPQQGGQDFELPEEFKKFMG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06149 SsrA-binding protein MAKEKGRKLIAQNKKARHDYQILDTYEAGLVLSGTEVKSLRQGRASLADGFVQLDGHEAWLHNVHVPEYSQGTWTNHSARRKRKLLLHRVEIDKLEAKSQETGHTIVPLALYFKDGRAKIEIALARGKKEYDKRQTLREKQDRREAERTISAIRRKQRA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06189 T Peptide TKPRKTKPRKTKPRKTKPR Tuftsin derivative Immune regulation MTT/MTS assay HT-29 Colon cancer 70% maximum inhibitory rate at 8 mg/kg
dbacp06195 Tat RKKRRQRRR HIV-Tat (49-57) Apoptosis inducing MTT/MTS assay HCT-116 Colon cancer ~10% cytotoxicity at 100 µM
dbacp06199 Tat-a5 KAQIRAMECNILGRKKRRQRRR HIV-Tat (49-57) Apoptosis inducing MTT/MTS assay HCT-116 Colon cancer ~80% cytotoxicity at 100 µM
dbacp06208 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay HCT116p53–/– Colon cancer Survival rate : 32.19 ± 6.42%
dbacp06209 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay HCT116p53+/+ Colon cancer Survival rate : 34.28 ± 8.93%
dbacp06210 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay GLC-82 Colon cancer Survival rate : 63.64 ± 4.80%
dbacp06211 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay SGC-7901 Colon cancer Survival rate : 64.75 ± 33.48%
dbacp06212 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay MDA-MB-231 Colon cancer Survival rate : 69.79 ± 6.71%
dbacp06213 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay HEK293 Colon cancer Survival rate : 115.85 ± 23.03%
dbacp06214 TAT-DV3-BH3 YGRKKRRQRRRGGGLGASWHRPDKGGGGLRRMADDLNAQY BH3-only, Direct activators (PUMA, Bid) Inducing apoptosis CCK-8 assay 2BS Colon cancer Survival rate : 124.38 ± 22.05%
dbacp06289 Tetrahydrofolate synthase MSDNPGENGQPDPSDPLDSFDEIIDAETTRDPDLAVIEAGSRTLRTQGGPPEADVPGRPEDPETDAALRAVETELATRWGETKLEPSVTRIAALMDVLGDPQRSYPSIHITGTNGKTSTARMIEALLGAFELRTGRYTSPHVQSITERISLDGAPMSAERFIETYQDIKPYVEMVDAQQEYRLSFFEVLTGMAYAAFADAPVDVAVVEVGMGGSWDATNVIDGDVAVVTPIDLDHTDRLGETPGEIATEKSGIVKQDATVILAQQPVDAAQVMLKKAVDVNATVAREGLEFGVVARQVAVGGQLATLRGLGGEYDEVYLPLHGAHQAHNAAVALAAVEAFFGVGAQRPEPLDLDTVRKAFAAVASPGRMEVVRRSPTVVLDAAHNPAGARVTAEAVGEAFQFSRLIGVVGASGDKNVRGLLEAFEPVFAEVVVTQNSSHRAMDADELAGVAVEVFGEDRVQVEPRLPDALEAAITLAEEEGEFAGGGVLVTGSVITVGEARLLMGKG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06297 Tetratricopeptide repeat protein MPRGAPARGSAHRYGDGPRFTQCPRPPGVPGREVAYCDLVDQDWEERVTAAWAAIDDYADDGAAEFRAVIDALADELPADSPLGLFERACAWDSTGHSDRAVPLYREALERGLGEVSHHKGRRAKIQLASSLRNTGHPEEGVLLLSPELVSTSDELDDAVRATLALCLSAMGRDREGLSLVLGALAPHLPRYQRSMAAYARQLVEPEDPED Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06310 TOMM leader peptide-binding protein MHDEQHHGPGLGGSDGLWDEALRGLGDALDAKVVANRGWDLSWERLQWEKASADGEDLVSVRVYDDEVVVGPRWVPGTDSGCASCAEVRERTTAEHPLATALDTPRAVPRAARPLLPLLLAAAAANLADHPLGPGELYAVGAQYVRRHRVPRSFFCPACADHGSVAADDWRPEPLELPAEPLSSKDPTRGAGGAHLVEPGALRERLLDARYGPIQVIMRESDVPFAMSMCLAPDAAAPGHGRAGTFAEADPVGIIETYERLGSFPFDTPLLLERSHREVAAHALDPVTLGEHTEKQLEHPDCQVLPYTPDTPMDWVWGHDLATGEPLLVPAEAGFYQYEQRFKLSRHAARAARVEARRARAAGHRPAPGTLRKYFHDSSSGCAAGSSLTEAALHSLLELAERDAFLLSWHRREPLPRIADASITDPESRSLIDLIRTRGFDVHVLVARQDIDLPIVWVLVVNRQNPFPASYSSGGSGADPDTAIRGALREVAQLVTNKMQWNREEAEQMLDDPWKLVELEQHPQLYTLPEKLARVTEVLGGPQTTVQDAFPGWPQVLRRASGGTVRGALDHVRALYAAAGLDRIVLVNQTTREHADAGISVAKAVVPGILPMCFGHAQQRLKNLPRLVAALAGTPQENREIPYDPHPFP Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06315 TOMM leader peptide-binding protein MHPMVKPALRRGWRDLNTVQFGMTPAHALTLAPVDTATGGFLELLNGTRGPALLREEGHRMDLPEGHVDRVVDRLAGAGLLDDSRGGGPAAEALREKKDVLDRLRPDLATLSLTTSAPGDAIRHLAARRALRVGVRGAGRVGAALAGLLSGAGVGEVDVRDGGCVEPWDVAPGGLPARSVGDRRDAAARRVVRAAAPGGPPRRSPAAPPDGSDPGLSLVVVAPRDDVAVHTPDPASVESLMASGTPHLYAGVVEGTGVVGPLVLPGETGCAGCLYADRTDRDPAWPRLVAQWRSGRPRPVPPCDLTLAATVAGLAAAHALAFLDGGTPAGTGVRWEVSLPALRWHARPVAAHPACPCGAAAEGKAEGKQEHIAEDGAGGATMAGQGPPSAARHGVGPTRPAGTWRAHV Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06342 Trigger factor MKSAVETLNPTRVRLTVEVPFEELKDSLDAAYKKINQQVTVKGFRKGKIPARVIDQRFGRGAVLEEAVNDALPKFYTDAVNEAELNPLGQPEVDITELKDGETLNFTAEVDIRPTVEIPDYSGIEVEVDAVEVSDEDVEKSVEQLRERFASTSPVERAAQDGDVLTLDLQAKVDGEVLEDGVADGVSYTIGSGELLDGIDEAVKGLEAGGEATFASELKGGSAAGKEAEVTVKVSQVAARELPELDDDFAQLASEFDTLEELQADSRKRLAnMKQYDQATQAQERVLDKLLELVEIPVPEKLLEDEINTRKHNLEHHQLGQMGLDLEKYLELQGKTAEEFETETREAAVKGIKTQFVLDELVKQENLNVSQEELTEHLMRRASSSGMSPDQFAQAVVEQGQVPLLVGEVARGKALAAVVEKATVKDTNGEIVDLDDEEDEEPETVEAAATESADAEQADEKADDKADDKAGKAEEKTEG Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06354 Trp operon leader peptide MSPERRRFENQRSRSPAQDYGVGTGAHGRAQRMRRAAHSGARPGWGTLPAMFAHPIQNWWWTAHPAAH Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06395 Type 2 lantipeptide synthetase LanM MSDVQVATDARPATGPTAAADAHVVTEPQVAVEDFLPFYRNRIPRQVVVDRLRGPLSQAAAPEHAGTLVDQVWEDLVTAVEGHSLRVLIGEFHEFRQSRGLPATAGSDEAISRFRRHIEDPDNCRELLGRYDVLRRRLTVVLDRFLDAYDDLFTAFRDDRPRLVERGLLTDGGDTLASLITTGGDPHNDNRRVVGVRLAGGGRLVFKPRTLAADDFVRDLYAVVDPYLAHSLGGCVPESLSVGDHGWQSFVTPRAMTGPDQPARYFYRFGALCALFGAIGASDLHDENLLAAGEHPCVIDTEMMLRPGSGTGDGSLEQRLNNHVEASVASTMLVPNVRPESPIDVIMAGVGVSGEQVSGKMKKSALQDGGTDALRLRWEPIVYQHKENVPRLGDEKLASVRFYRDIVAGYTDALGAVRERRAIEEVIGRYAELPVRCLIRSTMVYGRFLDAATQPRYLRDAGESERFLGLLKQFPRQLAPEARAFAGEAERVAMDTGNVPYFTGRAGTTELATHTDRLPGAHPSSPADAARAGLALHAAQSDRYHRFVLEECFGELAEAAPDVMSAQSVFAPVLDTPAGEPWWPHIARILQDIQVTYSDADGVQCGWVGGVGPDRGVPTLLPGNYLSFHDNGGIVTFLQDAAEHDPRFAELYRRADRGLSALLQVYDEAQLRAPESVFTGAASMMLTRPRRQDRAWTARLLERVPERIEAGTLEKDLANGPAGLLMAVLARLEAGQDRLMDEEQLGRLCDLVLGQAATPLDRAWYDVAHGDVGMWWAVSRIGRYLGDAALSGEAADRLTERLSAGELPPVPGWCNGSAGVLLVSAEILTSAGRPEVLTGGRLAELLDGATSSRGDRPVDLSVCHGSSGVVQSLIATSRLLEDRSLLGRAAEYREQTARAAGARGFHTGCPGRTSLLGYMFGWSGIGHTDLMLDEALDGRAPAFVPVALTAAGAPEEPAPPRRPGANVRASAAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06400 Type 2 lantipeptide synthetase LanM MRSAINYYPEFDDTEIEETITPLAAFDDEVRAVVSREPQQPAVLPSRPGVVKDWTARAEEYPFQQVVRDIAAGAADGDPLAAFPGLFADRDDALTELLDRAEARIRELYTRPLVAAVNHAREQGSLLGETPRERYRYFVDEAVRGSVASAGGLDFPVLRNLTPVVLAGTVDSVVELCSRLVADRAAIRDTFGIAVEDRLVSFGRPQGDTHHHGRAVCILAFESGTRLVYKPRDVSCEAGFAVLADEFNAAFGTRLHAVTALARDGYGYVEYVETEDVSAISERFLYESGELAAVLYLLNARDMHFENIVPTRRGPVPVDLETVLHPERIHVGPVPEADGNAYGTIGRSVYGVGILPLVMAGRRGDQGGHVDLGFLGGPGRGASPFKQMSFDEPYTDRIRLSLKAQEVSARRTVVGERTEEEILRLGRSMADGFTRTYRAVLAAPGTWTALLRKAADGLRIRYVHNPTALYSQTLRMVTGPSALDDTDTYLALLKRIAIASKTSDRTLIASELRQLAERDVPYFTVSATGTRVCDGDGREVGAAFGSSPLDLALDKAAGLGETDLGEQLRLIRSAFTAQFPDNHLTPARPTEAPSGGGADSGERAALTSLARELTDGLVATSLPDRFAHLPRTWIGPLASAEADRPWPPGVLGYDLYTGRTGIALTLAAAGRVLDDERCLAVARQIFSTTGEILASHRYETRSLQQAGYAGYTGMSGILFCLSAAGRLIGEEAWVSAAQGAVPLVLEQIRAVPVDELPLDVISGLAGVLNCFAAVADPTGSGVAAPEGREAVTEVALLLTRALGRDGALARSVLDQSGFAHGISGVVHALGRAHPLLPAEHRAPVGTALTDLVRRLDTFYDPAERNWSSQLSRQGSFATGWCHGATSVALALSGAAGVLGHETVAARRDQAVENTLRLGFGRNLTWCHGDLGNHGALRFIAGPDGSPLHDEVRQKERQWLRPEVMRRKLADPDSRYAHTNSLMVGSAGLALHLLNRIDPGLRLCPLTLTVEGR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06431 UDP-N-acetylmuramate--L-alanine ligase MAPGLPTAMDRPHFIGIGGAGMSGIAKVLAQRGAAVAGSDAKESATAGALRALGATVHIGHAAGHLADDASCVVVSSAIREDNPELARAAELGIPVVHRSDALAALMNGLRPLAVAGTHGKTTTTSMLAVSLSELGLNPSYAIGGDLDEPGSNALHGSGEIFVAEADESDRSFHKYAPEVAIVLNVELDHHANYASMDEIYESFETFADRIVPGGTLVIAADHEGARELTRRLAGTVRTVTYGESEDADVRILSVVPQGLKSEVTVVLDGAELTFGVSVPGRHYAHNAVAALAAGAALGVPAAELAAALAAYTGVKRRLQLKGEAAGVQVVDSYAHHPTEMTADLEAMRAAVGDARILVLFQPHLFSRTQELGKEMGQALALADASVVLDIYPAREDPIPGITSDLIVEAARAAGADVTPVHDKDAASAAVAGMAKAGDLVLTMGAGDVTDLGPRILDELSSQANQ Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06436 UDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligase MTYPGPPRPVRISATPLAELADQLGVTAPDSSAGVTGITHDSRAVRPGDLYAALPGARVHGADFATQAAGLGAAAVLTDPAGAERVSAAGLPALVVDDPRARMGELAATIYGHPGRDLLQIGITGTSGKTTTAYLVEGGLRTEKSTGLIGTVEMRIGDERIKSERTTPEATDLQALFSVMRERGTEAVAMEVSSHALVLGRVDACVFDVAVFTNLSPEHMEFHSGMEDYFQAKAQLFTPARSRLGVVNVDDEYGRRLAKEATVPVVTYSAEGHPDADWRADEVEVGPLDSTFTVLGPKGERIAAKSPLAGPFNVANTLAAIVSLAAAGLDPQTAADGVAAVPGVPGRLERVDEGQPFFAVVDYAHKTDAVESVLRALRKVTEGKLHAVLGCGGDRDTTKREPMGAAVARFADTAVLTSDNPRSEDPLAILAVMLQGAASVPAHERGEVQVFEDRAAAIAAAVARAEPGDTVVVAGKGHEQGQDIAGVVRPFDDREVLREAIQRSKA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06441 UDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase MITLSLAEIADVVGGRMHDIPDASAQVTGPVVRDSREAGPGSLFVAFVGERVDGHDFAPAVVGAGAVAVLGSRPVGVPAIVVDDVQAALGALARHVVRRLGTTLVALTGSAGKTSTKDLIAQVLRRKAPTVFTPGSLNNEIGLPLTALTATGETRFLVLEMGARGIGHIRYLCELTPPRIGLVLNVGSAHIGEFGGREQIAQAKGELVEALPPAGEGGTAVLNADDPLVRAMASRTTAKVLLFGESGEADVRAENVRLTDSGQPSFSLHTPSGASDVTMRLYGEHHVSNALAAAAVAHELGMSADEIATALSEADSLSRWRMEVTERPDGVTVVNDAYNANPESMKAALRALVAIGGASRARGGRTWAVLGEMAELGDEALAEHDAVGRLAVRLNVSKLVAVGGREAQWLQLGAYNEGSWGEESVHVSDAQAAVDLLRSELRPGDVVLVKASRSVGLESVATALLETGTEGEVAAR Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06446 UDP-N-acetylmuramoylalanine--D-glutamate ligase MPSEFSGKHVTVAGLGVSGVPAAKVLHGLGAHVTVVNDGADERARTQAAELEALGVTVRLGDGTASDSGSAAGLPEGTELIVTAPGWKPTKPLFTAAEQAGVPVWGDVELAWRLRGHGGRKAAPWLAVTGTNGKTTTVQMLASILAAAGLRTAAVGNIGVSLLDAVTGDTEYDVLAVELSSYQLHWAPSLRAHSAVVLNLAADHLDWHGSMEAYAADKGRVYEGNQVACVYNAADRATEDLVRAADVEEGCRAVGFTLGTPGPSQLGVVEGLLVDRAFVEDRHKNAQELAEVSDVNPPAPHNIANALAAAALARAYGVPAAAVRDGLRAFTPDAHRIAHVADVDGVAYVDDSKATNTHAAEASLAAYEPIVWIAGGLAKGATFDELVAGAAKRLRGAVLIGADRALIREALARHAPEVPVVDLDRTDTGAMPQAVREARRLAEPGDTVLLAPACASMDMFTNYNKRGDAFAEAVRELGA Streptomyces sp. VN1 Not specified Cytotoxicity assay HCT116 Colon cancer IC50 : 123.7 µM
dbacp06550 Z1 KAAKKWAKAAKKWAKAWKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : > 211 µM
dbacp06553 Z10 AAKKWAKAKWAKAKKWAKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : > 211 µM
dbacp06556 Z2 KAAKKWAKAWKKAAKAWKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : > 211 µM
dbacp06569 Z3 KAAKKAWKAWKKAAKAAWKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : >211 µM
dbacp06572 Z4 KAAKKAWKAAKKAAKWWKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 173 µM
dbacp06585 Z5 KAAKKAWKWAKKAAKWAKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 67 µM
dbacp06588 Z6 KWWKKAAKAAKKAAKAAKKWA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 31 µM
dbacp06591 Z7 KAAKKAWKAAKKAWKAAKKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 21 µM
dbacp06594 Z8 AWKKWAKAWKWAKAKWWAKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 23 µM
dbacp06597 Z9 AAWKWAWAKKWAKAKKWAKAA Synthetic Disruption of cell membrane MTT/MTS assay HT-29 Colon cancer EC50 : 13 µM
dbacp06605 αs1-casein f(90_95) RYLGYL Bovine milk Regulation of immune response; Apoptosis inducing MTT/MTS assay AZ-97 Colon cancer Inhibition at 12 - 15 g/l
dbacp06606 β-Casomorphins 5 f(60_64) YPFPG Bovine milk Regulation of immune response; Apoptosis inducing MTT/MTS assay AZ-97 Colon cancer Inhibition at 9 - 11 g/l
dbacp06608 Maculatin 1.3 GLLGLLGSVVSHVVPAIVGHF Fringed Tree Frog, Australia Disruption of either cancer or bacterial cell membrane integrity Not specified Not specified Colon cancer IC50 : 10−5 to 10−6 M
dbacp06654 LUNA18 Not Available Synthetic Not available CellTiter-Glo Cell Viability assay LS 180 Colon Cancer IC50 = 2.7 ± 0.4 nmol/L
dbacp06657 LfcinB (21-25)Pal RWQWRWQWR LfcinB Apoptosis inducing MTT assay HT-29 Colon Cancer IC50 = 100 μM
dbacp06659 Ahx-[Pal] Ahx-RWQWRWQWR Synthetic Apoptosis inducing MTT assay HT-29 Colon Cancer IC50 = 119 μM
dbacp06661 9[Orn] [Pal] RWQWRWQWO Synthetic Apoptosis inducing MTT assay HT-29 Colon Cancer IC50 = 109 μM
dbacp06672 Crabrolin FLPLILRKIVTAL European hornet (Vespa crabro) Not available MTT assay HCT-116 Colon Cancer IC50 = 8.539 μM
dbacp06677 Crabrolin-4R FLPRILRKIVTAL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 47.02 μM
dbacp06682 Crabrolin-4K FLPKILRKIVTAL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 42.88 μM
dbacp06687 Crabrolin-TR FLPRILRKIVRAL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 2.810 μM
dbacp06692 Crabrolin-FR RLPRILRKIVRAL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 30.29 μM
dbacp06697 Crabrolin-AR RLPRILRKIVRRL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 29.90 μM
dbacp06702 Crabrolin-PR RLRRILRKIVRRL Synthetic Analog of Crabrolin Not available MTT assay HCT-116 Colon Cancer IC50 = 16.29 μM
dbacp06737 Aurein 1.2_mutant (Aurm) GLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 51.63% cell viability
dbacp06738 Aurein 1.2_mutant (Aurm) GLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay HT-29 Colon Cancer 66.10% cell viability
dbacp06739 Aurein 1.2_R5 (R5-Aur) RRRRRGLFDIIKKIAESF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 43.89% cell viability
dbacp06740 Aurein 1.2_R5 (R5-Aur) RRRRRGLFDIIKKIAESF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay HT-29 Colon Cancer 61.56% cell viability
dbacp06741 Aurein 1.2_mutant_R5 (R5-Aurm) RRRRRGLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay SW-480 Colon Cancer 40.62% cell viability
dbacp06742 Aurein 1.2_mutant_R5 (R5-Aurm) RRRRRGLFDIIKKIIKSF Synthetic Necrotic activity via cell membrane lysis and apoptotic activity through disrupting mitochondrial membrane MTT assay HT-29 Colon Cancer 54.22% cell viability
dbacp06759 p28 LSTAADMQGVVTDGMASGLDKDYLKPDD Pseudomonas aeruginosa Apoptosis inducing MTT assay HT-29 Colon Cancer IC50 ~ 200 μg/ml
dbacp06767 M1-21 rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF Synthetic FOXM1 inhibitor Cell Viability assay HCT-116 Colon Cancer IC50 = 9.08 µM
dbacp06854 WP1 RLLRLMRLRMLLRM Derived from RLL peptide Apoptosis inducing Cell Viability assay HT-29 Colon Cancer IC50 = 54.6 ± 2.1 μM
dbacp06858 WP2 RLLRLLRLRRLLRL Derived from RLL peptide Apoptosis inducing Cell Viability assay HT-29 Colon Cancer IC50 = 42.6 ± 4.0 μM
dbacp06860 ALA-A2 KLWCKSSQVPQSR Alpha-Lactalbumin Not available MTT assay HT-29 Colon Cancer ~50% cell viability
dbacp07012 Sansalvimide A LXVLF Fusarium sp. Not Available Not Available HCT-116 Colon Cancer IC50 = 9.8 µg/ml
dbacp07013 Sansalvimide A LXVLF Fusarium sp. Not Available Not Available Colo-205 Colon Cancer IC50 = 3.5 µg/ml
dbacp07085 HB43 FAKLLAKLAKKLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 12 ± 4 μM
dbacp07086 HB43 FAKLLAKLAKKLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-620 Colon Cancer IC50 = 10 ± 1 μM
dbacp07087 HB43 FAKLLAKLAKKLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay HT-29 Colon Cancer IC50 = 11 ± 1 μM
dbacp07089 HB43-mut2 FAKLLAKLAKLLK Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 34 ± 2 μM
dbacp07090 HB43-mut2 FAKLLAKLAKLLK Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-620 Colon Cancer IC50 = 40 ± 3 μM
dbacp07091 HB43-mut2 FAKLLAKLAKLLK Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay HT-29 Colon Cancer IC50 = 50 ± 3 μM
dbacp07093 HB43-mut3 FAKLLAKLARRLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-480 Colon Cancer IC50 = 8 ± 1 μM
dbacp07094 HB43-mut3 FAKLLAKLARRLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay SW-620 Colon Cancer IC50 = 9 ± 1 μM
dbacp07095 HB43-mut3 FAKLLAKLARRLL Synthetic Motif-driven membrane insertion triggers cytotoxicity AlamarBlue assay HT-29 Colon Cancer IC50 = 9 ± 1 μM
dbacp07278 LCP-2 WAHT Laminaria japonica Mitochondrial apoptosis via p53 activation. MTT assay CaCo-2 Colon Cancer IC50 = 100 ± 11.6 μM
dbacp07282 LCP-3 WHLV Laminaria japonica Mitochondrial apoptosis via p53 activation. MTT assay CaCo-2 Colon Cancer IC50 = 68.2 ± 7.11 μM
dbacp07316 B1OS-L FLPLIASLAGNVVPKIFCKITKRC B-1OS Not Available MTT assay HCT-116 Colon Cancer IC50 = 11.03 µM
dbacp07321 B1OS-D-L FlPLIASLAGNVVPKIFCKITKRC B-1OS Not Available MTT assay HCT-116 Colon Cancer IC50 = 3.721 µM
dbacp07348 GA - 2 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 70.30 ± 0.9 µg/mL
dbacp07350 GA - 3 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 7.40 ± 0.4 µg/mL
dbacp07352 GA - 4 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 73.0 ± 1.4 µg/mL
dbacp07354 GA - 5 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 5.2 ± 0.8 µg/mL
dbacp07356 GA - 7 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 3.0 ± 1.1 µg/mL
dbacp07359 GA - 8 Structure given in figure Synthetic (glycyrrhetinic acid (GA)-based peptides) Apoptosis induction, Bax/p53/caspase activation MTT assay HCT-116 Colon Cancer IC50 = 60.70 ± 0.6 µg/mL
dbacp07374 HPRP-A1 FKKLKKLFSKLWNWK N-terminal region of Helicobacter pylori ribosomal protein L1 Apoptosis induction, p53-mediated cell cycle arrest MTT assay HT-29 Colon Cancer IC50 ~ 0.5 µg/mL
dbacp07378 Brevinin-2DYd GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC Rana dybowskii Not Available MTT assay LoVo Colon Cancer IC50 = 8.05 µg/ml
dbacp07382 Ranatuerin-2Lb GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC Rana luteiventris Not Available MTT assay LoVo Colon Cancer IC50 = 59.78 µM
dbacp07386 Odorranain-C1 GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC Odorrana grahami Not Available MTT assay LoVo Colon Cancer IC50 = 55.22 µM
dbacp07390 Brevinin-2DYb GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC Rana dybowskii Not Available MTT assay LoVo Colon Cancer IC50 = 35.05 µM
dbacp07394 Ranatuerin-2 GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP Rana catesbeiana Not Available MTT assay LoVo Colon Cancer IC50 = 128 µM
dbacp07424 GP-1 FKEHGY Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay CaCo-2 Colon Cancer IC50 = 104 ± 11.3 µM
dbacp07425 GP-1 FKEHGY Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay Colo-320 Colon Cancer IC50 = 111 ± 12.0 µM
dbacp07427 GP-2 EGFHL Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay CaCo-2 Colon Cancer IC50 = 154 ± 15.8 µM
dbacp07428 GP-2 EGFHL Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay Colo-320 Colon Cancer IC50 = 142 ± 14.9 µM
dbacp07430 GP-3 FSHTYV Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay CaCo-2 Colon Cancer IC50 = 162 ± 17.1 µM
dbacp07431 GP-3 FSHTYV Ginseng Leaf Peptide Mitochondrial apoptosis via p53 activation MTT assay Colo-320 Colon Cancer IC50 = 149 ± 15.2 µM
dbacp07469 Protonectin ILGTILGLLKGL Parachartergus fraternus Cell penetration without toxic accumulation Resazurin dye assay HCT-116 Colon Cancer CC50 = 8.0 ± 0.5 µM
dbacp07471 Protonectin-F IFGTILGFLKGL Protonoectin Cell penetration without toxic accumulation Resazurin dye assay HCT-116 Colon Cancer CC50 = 9.8 ± 1.2 µM
dbacp07474 MzDef MSSSNCANVCQTENFPGGECKAEGATRKCFCKNC Zea mays L. Disulfide-stabilized peptide disrupts pathogens MTT assay HCT-116 Colon Cancer IC50 = 29.85 µg/mL
dbacp07478 (LLKK)4 linear peptide LLKKLLKKLLKKLLKK Synthetic Apoptosis, drug-resistance reversal, tumor suppression MTT assay HCT-116 Colon Cancer Cell Viability (%) ~ 10.73 ± 2.4 at 30 µg/mL
dbacp07482 2-arm branched peptide [LLKKLLKK]2kC Synthetic Apoptosis, drug-resistance reversal, tumor suppression MTT assay HCT-116 Colon Cancer Cell Viability (%) ~ 78.6 ± 10.5 at 30 µg/mL
dbacp07486 4-arm branched peptide {[LLKKLLKK]2kC}2 Synthetic Apoptosis, drug-resistance reversal, tumor suppression MTT assay HCT-116 Colon Cancer Cell Viability (%) ~ 67.6 ± 5.8 at 30 µg/mL
dbacp07504 Brevinin-1Ha FALGAVTCLIRTKCKVLPKLF Analogue of Brevinin-1H α-helix enhances antimicrobial, anticancer activity MTT assay HCT-116 Colon Cancer IC50 = 342.8 µM
dbacp07508 Brevinin-1HY FALGAVTKVLYKLFCLITRKC Analogue of Brevinin-1H α-helix enhances antimicrobial, anticancer activity MTT assay HCT-116 Colon Cancer IC50 = 3.583 µM
dbacp07511 YT12 YFYPKDFTPGCT Arthrospira platensis ROS scavenging induces cancer cell death MTT assay HT-29 Colon Cancer IC50 = 12.5 μM
dbacp07536 AEM-28 LRKLRKRLLRDWLKAFYDKVAEKLKEAF Synthetic LPA reduction suppresses tumor growth MTS assay ID8 Colon Cancer ~60% cell viability at 10 μg/mL
dbacp07539 AEM-28 LRKLRKRLLRDWLKAFYDKVAEKLKEAF Synthetic LPA reduction suppresses tumor growth MTS assay CaCo-2 Colon Cancer ~70% cell viability at 10 μg/mL
dbacp07542 AEM-28–2 Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF Synthetic LPA reduction suppresses tumor growth MTS assay ID8 Colon Cancer ~20% cell viability at 10 μg/mL
dbacp07545 AEM-28–2 Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF Synthetic LPA reduction suppresses tumor growth MTS assay CaCo-2 Colon Cancer ~60% cell viability at 10 μg/mL
dbacp07546 Sur-X YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM Synthetic Disrupts XIAP-survivin, induces apoptosis/necroptosis MTT assay HCT-116 Colon Cancer 20% cell viability at at 20 μM
dbacp07547 Sur-X YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM Synthetic Disrupts XIAP-survivin, induces apoptosis/necroptosis MTT assay HCT-15 Colon Cancer Not Available
dbacp07548 Sur-X YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM Synthetic Disrupts XIAP-survivin, induces apoptosis/necroptosis MTT assay RKO Colon Cancer 25% cell viability at at 20 μM
dbacp07549 Sur-X YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM Synthetic Disrupts XIAP-survivin, induces apoptosis/necroptosis MTT assay HT-29 Colon Cancer Not Available
dbacp07551 NMANF2 KAIGLVIPEIDGKLDGGAQRV Staphylococcus hominis strain MANF2 GAPDH-like protein disrupts survival MTT assay HT-29 Colon Cancer IC50 = 48.9 µg/mL
dbacp07802 Longicalycinin A cyclic analogue 18 FSPAG Synthetic Analogue of Longicalycinin A Cyclization enhances apoptosis via lysosomes MTT assay HT-29 Colon Cancer 22.8% Cell death at 100 µg/ml
dbacp07890 H-58 IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 1.29 ± 0.08 μM
dbacp07893 H-57 IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 1.29 ± 0.08 μM
dbacp07896 H-18 IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 1.11 ± 0.21 μM
dbacp07899 H-21 IKLSKS5TKKS5LKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 3.05 ± 0.21 μM
dbacp07902 H-20 IKLSPS5TKKS5LKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 2.63 ± 0.35 μM
dbacp07905 H-19 IKLSKETKKNLKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 1.78 ± 0.35 μM
dbacp07908 H-17 IKLSKS5TKKS5LKKVLKGAIKGAIAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 1.49 ± 0.45 μM
dbacp07911 H-16 IKLSPS5TKKS5LKKVLKGAIKGAIAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 2.65 ± 0.35 μM
dbacp07914 H-15 IKLSKS5TKDS5LKKVLKGAIKGAIAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 2.95 ± 0.25 μM
dbacp07917 H-10 IKLSPS5TKDS5LKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 3.51 ± 0.37 μM
dbacp07920 H-5 IKLSPETKDNLKKVLKGS5IKGS5IAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 4.16 ± 0.21 μM
dbacp07923 H-2 IKLSPS5TKDS5LKKVLKGAIKGAIAVAKMV Synthetic Cell entry, DNA damage, apoptosis. MTT assay HCT-116 Colon Cancer IC50 = 3.54 ± 0.72 μM
dbacp08018 Peptide4 Gonearrestide ADAPGNYPLDARGKSYYC Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay HCT-116 Colon Cancer Not Available
dbacp08019 Peptide4 Gonearrestide ADAPGNYPLDARGKSYYC Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay DLD-1 Colon Cancer Not Available
dbacp08020 Peptide4 Gonearrestide ADAPGNYPLDARGKSYYC Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay HKe-3 Colon Cancer Not Available
dbacp08021 Peptide4 Gonearrestide ADAPGNYPLDARGKSYYC Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay Dks8 Colon Cancer Not Available
dbacp08023 Peptide6 Gonearrestide KLSAIISKIRDE Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay HCT-116 Colon Cancer Not Available
dbacp08024 Peptide6 Gonearrestide KLSAIISKIRDE Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay DLD-1 Colon Cancer Not Available
dbacp08025 Peptide6 Gonearrestide KLSAIISKIRDE Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay HKe-3 Colon Cancer Not Available
dbacp08026 Peptide6 Gonearrestide KLSAIISKIRDE Androctonus australis Gonearrestide induces G1 cell-cycle arrest MTT assay Dks8 Colon Cancer Not Available
dbacp08028 Peptide10 Gonearrestide NDADKDEMQSVYRGKANDDNSRGSKTNHRF Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay HCT-116 Colon Cancer Not Available
dbacp08029 Peptide10 Gonearrestide NDADKDEMQSVYRGKANDDNSRGSKTNHRF Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay DLD-1 Colon Cancer Not Available
dbacp08030 Peptide10 Gonearrestide NDADKDEMQSVYRGKANDDNSRGSKTNHRF Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay HKe-3 Colon Cancer Not Available
dbacp08031 Peptide10 Gonearrestide NDADKDEMQSVYRGKANDDNSRGSKTNHRF Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay Dks8 Colon Cancer Not Available
dbacp08033 Peptide13 Gonearrestide WCYKLPDRVSIKEKGRCN Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay HCT-116 Colon Cancer IC50 ~ 100 μM/L
dbacp08034 Peptide13 Gonearrestide WCYKLPDRVSIKEKGRCN Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay DLD-1 Colon Cancer Not Available
dbacp08035 Peptide13 Gonearrestide WCYKLPDRVSIKEKGRCN Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay HKe-3 Colon Cancer Not Available
dbacp08036 Peptide13 Gonearrestide WCYKLPDRVSIKEKGRCN Androctonus mauritanicus Gonearrestide induces G1 cell-cycle arrest MTT assay Dks8 Colon Cancer Not Available
dbacp08043 Silk Fibroin peptide Not Available Silkworm Cocoons SFP induces S-phase cell-cycle arrest MTT assay HT-29 Colon Cancer IC50 = 11.55 ± 3.33 mg/ml
dbacp08060 TAT-327 RKKRRQRRREFLDCFQKF Peptide-327 Peptide 327 blocks Eps8–EGFR CCK-8 assay Colo-320 Colon Cancer EC50 = 68.40 ± 0.42 μM
dbacp08061 TAT-327 RKKRRQRRREFLDCFQKF Peptide-327 Peptide 327 blocks Eps8–EGFR CCK-8 assay HT-29 Colon Cancer EC50 = 74.08 ± 0.63 μM
dbacp08114 FR-15 FRRFFKWFRRFFKFF Synthetic Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 6.7 μM
dbacp08118 FR4P FRRPFKWFRRFFKFF Analogue of FR-15 Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 9.4 μM
dbacp08122 FR8P FRRFFKWPRRFFKFF Analogue of FR-15 Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 10.8 μM
dbacp08126 FR11P FRRFFKWFRRPFKFF Analogue of FR-15 Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 12.9 μM
dbacp08130 FR4,8P FRRPFKWPRRFFKFF Analogue of FR-15 Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 15.3 μM
dbacp08134 FR8,11P FRRFFKWPRRPFKFF Analogue of FR-15 Proline-substituted AMP triggers mitochondrial apoptosis MTT assay DLD-1 Colon Cancer IC50 = 22 μM
dbacp08172 Peptide - 1 GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKK Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 = 5.4 µM
dbacp08173 Peptide - 1 GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKK Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08184 Peptide - 2 GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRR Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 = 6.6 µM
dbacp08185 Peptide - 2 GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRR Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 = 6.4 µM
dbacp08192 Peptide - 3 GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- Orn Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 = 3.2 µM
dbacp08193 Peptide - 3 GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- Orn Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 = 6.2 µM
dbacp08200 Peptide - 4 GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-Dab Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 = 6.4 µM
dbacp08201 Peptide - 4 GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-Dab Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 = 2.6 µM
dbacp08208 Peptide - 6 GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 > 7.5 µM
dbacp08209 Peptide - 6 GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08216 Peptide - 7 GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRR Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 > 7.5 µM
dbacp08217 Peptide - 7 GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRR Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08224 Peptide - 8 GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKK Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 > 7.5 µM
dbacp08225 Peptide - 8 GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKK Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08232 Peptide - 9 GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKK Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 > 7.5 µM
dbacp08233 Peptide - 9 GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKK Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08240 Peptide - 10 GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 > 7.5 µM
dbacp08241 Peptide - 10 GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKK Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08248 Peptide - 11 KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c) Synthetic Not Available CellTiter-Glo assay COLO-205 Colon Cancer IC50 = 6.7 µM
dbacp08249 Peptide - 11 KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c) Synthetic Not Available CellTiter-Glo assay DLD-1 Colon Cancer IC50 > 7.5 µM
dbacp08259 Tr3 Not Available Protein extraction from Spirulina platensis Not Available MTT assay HT-29 Colon Cancer IC50 = 112.89 μg/mL
dbacp08262 HR HVLSRAPR Fraction identified from Tr1 Not Available MTT assay HT-29 Colon Cancer IC50 = 99.88 μg/mL