438 result(s) have been found!
| Accession | Name | Sequence | Source/Organism | Mechanism | Assay Type | Cell Line | Cancer Type | Activity |
|---|---|---|---|---|---|---|---|---|
| dbacp00051 | Enkephalins7 analogue-8 | YA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 2.4% inhibition at 10-5 M |
| dbacp00052 | Enkephalins7 analogue-8 | YA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 7.5% inhibition at 10-4 M |
| dbacp00075 | Enkephalins7 analogue-9 | YSA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 1.1% inhibition at 10-5 M |
| dbacp00076 | Enkephalins7 analogue-9 | YSA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 1.2% inhibition at 10-4 M |
| dbacp00077 | Enkephalins7 analogue-9 | YSA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 17.8% inhibition at 10-3 M |
| dbacp00096 | Enkephalins7 analogue-10 | YSA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 7.7% inhibition at 10-4 M |
| dbacp00097 | Enkephalins7 analogue-10 | YSA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 18.7% inhibition at 10-3 M |
| dbacp00149 | Enkephalins7 analogue-15 | YSA*G | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 21.2% inhibition at 10-3 M |
| dbacp00182 | Enkephalins7 analogue-16 | YRA*G | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 15.6% inhibition at 10-3 M |
| dbacp00216 | Enkephalins7 analogue-17 | YA*GFM | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 22.8% inhibition at 10-3 M |
| dbacp00250 | Enkephalins7 analogue-18 | YA*GFM | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 9.6% inhibition at 10-4 M |
| dbacp00251 | Enkephalins7 analogue-18 | YA*GFM | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 29.9% inhibition at 10-3 M |
| dbacp00288 | Enkephalins7 analogue-23 | YGGFMA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 2.2% inhibition at 10-6 M |
| dbacp00289 | Enkephalins7 analogue-23 | YGGFMA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 7.1% inhibition at 10-5 M |
| dbacp00290 | Enkephalins7 analogue-23 | YGGFMA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 6.9% inhibition at 10-4 M |
| dbacp00291 | Enkephalins7 analogue-23 | YGGFMA* | Synthetic Peptide | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | 25.9% inhibition at 10-3 M |
| dbacp00304 | Temporin-SHf | FFFLSRIF* | Sahara frog | Apoptosis inducing | MTT assay | MCF-7 | Not specified | IC50 : 32.76 ± 1.528 µM |
| dbacp00342 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 29.0 ± 3.7 μM |
| dbacp00343 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 29.0 ± 3.7 μM |
| dbacp00344 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 29.0 ± 3.7 μM |
| dbacp00345 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 29.0 ± 3.7 μM |
| dbacp00346 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 29.0 ± 3.7 μM |
| dbacp00382 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 37.5 ± 3.3 μM |
| dbacp00383 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 37.5 ± 3.3 μM |
| dbacp00384 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 37.5 ± 3.3 μM |
| dbacp00385 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 37.5 ± 3.3 μM |
| dbacp00386 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 37.5 ± 3.3 μM |
| dbacp00460 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 6.7 ± 0.7 μM |
| dbacp00461 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 6.7 ± 0.7 μM |
| dbacp00462 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 6.7 ± 0.7 μM |
| dbacp00463 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 6.7 ± 0.7 μM |
| dbacp00464 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 6.7 ± 0.7 μM |
| dbacp00500 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 15.2 ± 1.9 μM |
| dbacp00501 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 15.2 ± 1.9 μM |
| dbacp00502 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 15.2 ± 1.9 μM |
| dbacp00503 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 15.2 ± 1.9 μM |
| dbacp00504 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 15.2 ± 1.9 μM |
| dbacp00593 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 48.4 ± 0.7 μM |
| dbacp00594 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 48.4 ± 0.7 μM |
| dbacp00595 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 48.4 ± 0.7 μM |
| dbacp00596 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 48.4 ± 0.7 μM |
| dbacp00597 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 48.4 ± 0.7 μM |
| dbacp00666 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 15.1 ± 1.4 μM |
| dbacp00667 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid Leukemia | CC50 : 15.1 ± 1.4 μM |
| dbacp00668 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 15.1 ± 1.4 μM |
| dbacp00669 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 15.1 ± 1.4 μM |
| dbacp00670 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 15.1 ± 1.4 μM |
| dbacp00775 | A12L | KWKSFLKTFKSLKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 5 µMo/L |
| dbacp00783 | A12L/A20L | KWKSFLKTFKSLKKTVLHTLLKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 6.2 µMo/L |
| dbacp00791 | A12L/A20L/A23L | KWKSFLKTFKSLKKTVLHTLLKLISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 5.7 µMo/L |
| dbacp00799 | A20L | KWKSFLKTFKSAKKTVLHTLLKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 5.1 µMo/L |
| dbacp00811 | A4K14-citropin1.1 | GLFAVIKKVASVIKGL | Synthetic construct | Cell membrane disintegration | CCK-8 test | MCF-7 | Prostate cancer | IC50 : 14.16 μM |
| dbacp00812 | A4K14-citropin1.1 | GLFAVIKKVASVIKGL | Synthetic construct | Cell membrane disintegration | CCK-8 test | MCF-7 | Lung cancer | IC50 : 14.16 μM |
| dbacp00819 | AaeAP1 | FLFSLIPSVIAGLVSAIRN | Aeneas fattailed scorpion | Not specified | MTT assay | MCF-7 | Prostate cancer | Not found |
| dbacp00823 | AaeAP1 | FLFSLIPSVIAGLVSAIRN | Venom, Aeneas fattailed scorpion, Africa | Membrane lysis | MTT assay | MCF-7 | Non-tumourigenic mammary gland cancer | MIC : 10−4 to 10−9 M |
| dbacp00827 | AaeAP2 | FLFSLIPSAIAGLVSAIRN | Aeneas fattailed scorpion | Not specified | MTT assay | MCF-7 | Prostate cancer | Not found |
| dbacp00831 | AaeAP2 | FLFSLIPSAIAGLVSAIRN | Venom, Aeneas fattailed scorpion, Africa | Membrane lysis | MTT assay | MCF-7 | Non-tumourigenic mammary gland cancer | MIC : 10−4 to 10−9 M |
| dbacp01142 | Amphipathic peptide CT1 | MKTQFVILIVAVVLLQLISHSEAFLGALWNVAKSVFGKRGLRNFDDLDDTFEPEMSEADLKYLQDLLR | Scorpions, Morelos, located in South-Central Mexico (Mexican scorpion) | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 6.3-12.5 μM |
| dbacp01163 | Antimicrobial peptide TsAP-1 | MQIKHLITLFFLVLIVADQCSAFLSLIPSLVGGSISAFKGRRKREISAQIEQYKDLQKREAELEELLDRLPMY | Brazilian scorpion | Membrane disruption | MTT Cell viability assay | MCF-7 | Human breast carcinoma | IC50 : 0.83 - 2.0 μM |
| dbacp01187 | APQQ | NA | Synthetic construct | Cell metatstasis inhibition | Transwell assay | MCF-7 | Breast cancer | Not found |
| dbacp01391 | Aurein-3.3 [Cleaved into: Aurein-3.3.1] | GLFDIVKKIAGHIVSSI | Southern bell frog | Cell membrane disintegration | One-dose and five-dose assay | MCF7 | Breast cancer | IC50 : 5 μM |
| dbacp01919 | BR-C | CKLKNFAKGVAQSLLNKASKLSGQC | Not found | Inducing apoptosis | Not specified | MCF-7 | Not specified | IC50 : 45.72 μg/ml |
| dbacp01921 | BR-D | KLKNFAKGVAQSLLNKASCKLSGQC | Not found | Inducing apoptosis | Not specified | MCF-7 | Not specified | IC50 : 67.52 μg/ml |
| dbacp01974 | Brevinin-2R | KLKNFAKGVAQSLLNKASCKLSGQC | Skin, Marsh frog, Europe | Activates the lysosomal-mitochondrial death pathway; Involves autophagy-like cell death | MTT-assay | MCF-7 | Breast adenocarcinoma | LD50 : 10 – 15μg/ml |
| dbacp01975 | Brevinin-2R | KLKNFAKGVAQSLLNKASCKLSGQC | Skin, Marsh frog, Europe | Activates the lysosomal-mitochondrial death pathway; Involves autophagy-like cell death | MTT-assay | MCF-7 | Breast adenocarcinoma | LD50 : 20 – 25 μg/ml |
| dbacp01976 | Brevinin-2R | KLKNFAKGVAQSLLNKASCKLSGQC | Skin, Marsh frog, Europe | Activates the lysosomal-mitochondrial death pathway; Involves autophagy-like cell death | MTT-assay | MCF-7 | Breast adenocarcinoma | LD50 : 30 – 40 μg/ml |
| dbacp01983 | Brevinin-2R | KLKNFAKGVAQSLLNKASCKLSGQC | Skin, Marsh frog, Europe | Activates the lysosomal-mitochondrial death pathway; Involves autophagy-like cell death | MTT-assay | MCF-7 | Breast adenocarcinoma | LD50 : 10 – 15 µg/ml |
| dbacp01984 | Brevinin-2R (BR-2R) | KLKNFAKGVAQSLLNKASCKLSGQC | Not found | Inducing apoptosis | Not specified | MCF-7 | Not specified | IC50 : 24.11 μg/ml |
| dbacp01995 | Buforin IIb | RAGLQFPVGRLLRRLLRRLLR | Histone H2A | Inducing mitochondria-dependent apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 15.1 µg/ml |
| dbacp02053 | Buforin Iib | RAGLQFPVGRLLRRLLRRLLR | Not found | Inducing apoptosis | MTT/MTS assay | MCF-7 | Not specified | IC50 : 15.1 µg/ml |
| dbacp02112 | cMastoparan-C(cMP-C) | CLNLKALLAVAKKILC | Synthetic construct | Apoptosis | MTT assay | MCF-7 | Human breast cancer | IC50 : 13.66 μM |
| dbacp02284 | Cancer stem-like cells CD44 peptide-specific CTLs | YIFYTFSTV,LILAVCIAV,SLLALALIL,IILASLLAL,WLIILASLL,VLLQTTTRM,GLVEDLDRT,TVGDSNSNV | Cancer stem-like cells CD44 peptide-specific CTLs | Cell membrane penetrating | Not specified | MCF-7 | Breast cancer | Not found |
| dbacp02285 | Cancer stem-like cells EpCAM peptide-CTLs | VVAGIVVLV,GLKAGVIAV,VLAFGLLLA,RTYWIIIEL,SMCWCVNTA,SMQGLKAGV,ILYENNVIT,LLLAAATAT | Cancer stem-like cells EpCAM peptide-CTLs | Inhibit tumor growth and induce specific immune response | Not specified | MCF-7 | Hepatoma cancer | Not found |
| dbacp02298 | Carcinoembryonic antigen glypican-3 GPC3(298-306) | EYILSLEEL | Carcinoembryonic antigen glypican-3 GPC3(298-306) | Immune response to tumor cell recognition | Cytotoxicity assay | MCF-7 | Not specified | Not found |
| dbacp02366 | Cecropin B | KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL | Silkmoth | Pore formation at the cytoplasmic membrane | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 42.5 µM |
| dbacp02369 | Cecropin B | KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL | Silkmoth | Pore formation at the cytoplasmic membrane | MTT/MTS assay | MCF-7R | Breast cancer | IC50 : 24.5 µM |
| dbacp02415 | cGm (Derived from Gm) | GCRRLCYKQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Epithelial cancer | CC50 : 15.3 ± 1.4 μM |
| dbacp02416 | cGm (Derived from Gm) | GCRRLCYKQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Chronic myeloid leukemia | CC50 : 15.3 ± 1.4 μM |
| dbacp02417 | cGm (Derived from Gm) | GCRRLCYKQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Gastric cancer | CC50 : 15.3 ± 1.4 μM |
| dbacp02418 | cGm (Derived from Gm) | GCRRLCYKQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Breast cancer | CC50 : 15.3 ± 1.4 μM |
| dbacp02419 | cGm (Derived from Gm) | GCRRLCYKQRCVTYCRGR | Synthetic construct | Target and destroy tumor cell membranes | Cell viability assay | MCF-7 | Cervical cancer | CC50 : 15.3 ± 1.4 μM |
| dbacp02475 | Chickpea peptide | ADLPGLK | Plant sources | Inducing apoptosis | SRB assay | MCF-7 | Human endometrial cancer | IC50 : 110.3 ± 2.97µM |
| dbacp02546 | Conotoxin Cl14.1a (Conotoxin Cal14.1a) | MNVTAMFIVLLLTMPLTDGFNIRAINGGELFGLVQRDAGNALDHGFYRRGDCPPWCVGARCRAEKC | California cone | Apoptosis | Not specified | MCF-7 | Breast cancer | Not found |
| dbacp02629 | D-SVS-1 | kvkvkvkvPptkvkvkvk | Synthetic peptide | Disruption of cell membranes | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 4.7 ± 0.4 µM |
| dbacp02637 | Decoralin | SLLSLIRKLI | Solitary eumenine wasp | Mediate necrosis | MTT assay | MCF-7 | Breast cancer | IC50 : 12.5 μmolL−1 |
| dbacp02645 | Defensin-like protein (Sesquin) | KTCENLADTY | Yard-Long bean | Anti-proliferative action | MTT assay | MCF-7 | Leukemia | MIC : 0.25 μg/ml |
| dbacp02654 | Dermaseptin PS4 | MDILKKSIFLVLFLGLVSLSICEEEKRENEDEEKQEDDEQSEEKRALWKTLLKHVGKAAGKAALNAVTDMVNQGEQ | Sauvage's leaf frog | Membrane disruption | Lactate dehydrogenase (LDH) cytotoxicity assay, MTT assay | MCF-7 | Breast cancer | MIC : 10−9 to 10−4 M |
| dbacp02660 | Dermaseptin-B3 | ALWKnMLKGIGKLAGQAALGAVKTLVGA | South American frog, Giant leaf frog | Apoptosis inducing | Thymidine Incorporation assay | MCF-7 | Breast cancer | Not found |
| dbacp02661 | Dermaseptin-B4 | ALWKDILKNVGKAAGKAVLNTVTDMVNQ | Giant leaf frog | Apoptosis inducing | Thymidine Incorporation assay | MCF-7 | Breast cancer | Not found |
| dbacp02678 | Dermaseptin-PH | ALWKEVLKNAGKAALNEINNLVQ | Northern orange-legged leaf frog | Cell membrane permeabilization | Bioactivity assessment assay, MTT cell proliferation assay | MCF-7 | Not specified | IC50 : 0.69 μM |
| dbacp02683 | Dermaseptin-PH | ALWKEVLKNAGKAALNEINNLV | Orange-legged leaf frog, Northern orange-legged leaf frog, South America | Cell membrane permeabilization | MTT cell proliferation assay | MCF-7 | Lung cancer | IC50 : 0.69 μM |
| dbacp02689 | Dermaseptin-PH | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay, Lactate dehydrogenase (LDH) assay | MCF-7 | Breast cancer | IC50 : 17.44 - 49.51 μM |
| dbacp02693 | Dermaseptin-PH (DRS-PH) | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Brain tumor | IC50 : 7.44 μM |
| dbacp02694 | Dermaseptin-PH (DRS-PH) | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Breast cancer | IC50 : 7.44 μM |
| dbacp02695 | Dermaseptin-PH (DRS-PH) | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | pancreatic cancer | IC50 : 7.44 μM |
| dbacp02696 | Dermaseptin-PH (DRS-PH) | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Lung cancer | IC50 : 7.44 μM |
| dbacp02697 | Dermaseptin-PH (DRS-PH) | MDILKKSLFLILFLGVVSLSICEEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Prostate cancer | IC50 : 7.44 μM |
| dbacp02730 | Dermaseptin-PS4 | ALWKTLLKHVGKAAGKAALNAVTDMVNQ | Waxy monkey tree frog | Membrane disruption | Lactate dehydrogenase (LDH) cytotoxicity assay, MTT assay | MCF-7 | Breast cancer | MIC : 10−9 to 10−4 M |
| dbacp02732 | Dermaseptin-PT9 | GLWSKIKDAAKTAGKAALGFVNEMV | Brownbelly leaf frog | Disruption of cell membranes | MTT assay, Lactate dehydrogenase (LDH) assay | MCF-7 | Breast cancer | IC50 : 8.64 - 18.51 μM |
| dbacp02737 | Dermaseptin-PT9 | GLWSKIKDAAKTAGKAALGFVNEMV | Skin secretion, Brownbelly leaf frog, Purchased in Peru, South America | Disruption of cell membranes | MTT assay, Lactate dehydrogenase (LDH) assay | MCF-7 | Breast cancer | IC50 : 8.64 - 18.51 μM |
| dbacp02745 | Dex-(KW)3 | KWKWKW | Synthetic | Cell membrane disruption | MTT/MTS assay | MCF-7 | Breast cancer | At 10 µM 35-40% viablity |
| dbacp02759 | Dimer of peptide-paclitaxel conjugate | (K-Aib-C(CH2CO-2'-Pac))2 | Synthetic peptide paclitaxel conjugate | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 0.62 nM |
| dbacp02815 | DRS B3 | ALWKnMLKGIGKLAGQAALGAVKTLVGA | Dermaseptins B | Apoptosis inducing | Thymidine incorporation assay | MCF-7 | Breast cancer | Cytotoxicity :12 µM |
| dbacp02816 | DRS B4 | ALWKDILKNVGKAAGKAVLNTVTDMVNQ | Dermaseptins B | Apoptosis inducing | Thymidine incorporation assay | MCF-7 | Breast cancer | Cytotoxicity :15 µM |
| dbacp02817 | DRS S1 | ALWKTMLKKLGTMALHAGKAALGAAADTISQGTQ | Dermaseptins B | Apoptosis inducing | Thymidine incorporation assay | MCF-7 | Breast cancer | Not found |
| dbacp02829 | Elastin derived peptide | VGVAPG | Elastin derived | Apoptosis inducing | Cell viability assay | MCF-7 | Breast cancer | Not found |
| dbacp02931 | Figainin 1 | FIGTLIPLALGALTKLFK | Chaco tree frog | Membrane disruption and cell lysis | MTT/MTS assay | MCF | Murine Melanoma | IC50 : 13.7 µM |
| dbacp02939 | Figainin 1 | MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG | Chaco tree frog | Anti-proliferative action | MTT/MTS assay | MCF | Skin cancer | IC50 : 13.7 µM |
| dbacp02940 | Figainin 1 | MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG | Chaco tree frog | Anti-proliferative action | MTT/MTS assay | MCF | Breast cancer | IC50 : 13.7 µM |
| dbacp02941 | Figainin 1 | MAFLKKSLFLVLFLGLVSLSIGEEEKREEEEKNEEGANQEENAENKEKRFIGTLIPLALGALTKLFKG | Chaco tree frog | Anti-proliferative action | MTT/MTS assay | MCF | Cervical cancer | IC50 : 13.7 µM |
| dbacp02947 | Figainin 1 | FIGTLIPLALGALTKLFK | Skin secretions, Chaco tree frog, South America | Membrane disruption | MTT/MTS assay | MCF | Murine melanoma | IC50 : 13.7 µM |
| dbacp02950 | Figainin 2 | FLGAILKIGHALAKTVLPMVTNAFKPKQ | Skin secretions, Chaco tree frog, South America | Cell membrane interaction; Necrosis; Apoptosis | MTT/MTS assay | MCF-7 | Murien melanoma | IC50 : 15.3 µM |
| dbacp02953 | Figainin 2 | MAFLKKSLFLVLFLGIVSLSVCEEEKREGEEKEEKREEEEGKEENEDGNEEHKEKRFLGAILKIGHALAKTVLPMVTNAFKPKQ | Chaco tree frog | Necrosis; Apoptosis | MTT/MTS assay | MCF-7 | Skin cancer | IC50 : 15.3 µM |
| dbacp02954 | Figainin 2 | MAFLKKSLFLVLFLGIVSLSVCEEEKREGEEKEEKREEEEGKEENEDGNEEHKEKRFLGAILKIGHALAKTVLPMVTNAFKPKQ | Chaco tree frog | Necrosis; Apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 15.3 µM |
| dbacp03035 | Galaxamide derivative (Compound 3) | cyclo(WnMLLLnML) | Marine invertebrates | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 1.72 ± 0.85 μg/mL |
| dbacp03039 | Galaxamide derivative Compound 1 | cyclo(FnMLLLnML) | Marine invertebrates | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 4.76 ± 1.36 μg/mL |
| dbacp03043 | Galaxamide derivative Compound 2 | cyclo(NAl-nMLLLnML) | Marine invertebrates | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 3.16 ± 0.92 μg/mL |
| dbacp03061 | GGN6 | FLPLLAGLAANFLPTIICKISYKC | Skin of a Korean frog, wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 4.88 µg/ml |
| dbacp03292 | HECI | TVLRGCWTFSFPPKPCI | Hylarana erythraea | Cell membrane disintegration | MTT anti-proliferation assay | MCF-7 | Breast cancer | MIC : 1µM |
| dbacp03367 | Ichthyophthirius multifiliis (strain G5) B4 | LKKLFKKILKYL | White spot disease (strain G5) B4 | Apoptosis inducing; Penetration of the cell membrane | MTT assay | MCF-7 | Breast cancer | MIC : 5 μM |
| dbacp03369 | Ichthyophthirius multifiliis (strain G5) B8 | LKKLFKKILKY | White spot disease (strain G5) B8 | Apoptosis inducing; Penetration of the cell membrane | MTT assay | MCF-7 | Breast cancer | MIC : 7 μM |
| dbacp03371 | Ichthyophthirius multifiliis BP100 | KKLFKKILKYL | White spot disease BP100 | Apoptosis inducing; Penetration of the cell membrane | MTT assay | MCF-7 | Breast cancer | MIC : 25 μM |
| dbacp03485 | K8, 23-DPT9 | MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Brain tumor | IC50 : 8.64μM |
| dbacp03486 | K8, 23-DPT9 | MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Breast cancer | IC50 : 8.64μM |
| dbacp03487 | K8, 23-DPT9 | MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Pancreatic cancer | IC50 : 8.64μM |
| dbacp03488 | K8, 23-DPT9 | MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Lung cancer | IC50 : 8.64μM |
| dbacp03489 | K8, 23-DPT9 | MDILKKSKFLILFLGVVSLSICKEEKRENEEEMEQDDEQSEMKRALWKEVLKNAGKAALNEINNLVQGGQ | Northern orange-legged leaf frog | Disruption of cell membranes | MTT assay | MCF-7 | Prostate cancer | IC50 : 8.64μM |
| dbacp03533 | L-amino acid oxidase (CC-LAAO) (LAO) (EC 1.4.3.2) | MNVFFMFSLLFLAALESCADDKNPLEEEFFEADYEEFLLIAKNGLQQTSNPKRVVIVGAGMSGLSAAYVLAKTGHEVILLEASERVGGRVSTYRNDQEGWYANLGPMRLPERHRIVREYIRKFGLQLNEFSQENENAWYFIKNIRKRVGEVNKDPGVLEYPVKPSEKGKSAPQLYRDSLQKIIEEYGRSNCSYILNKYDTYSTKDYLIKEGNLSPGAVDMVGDLLNEDSGYYVSFIESLKPDDIFAYENRFDEIVGGFDKLPTSMYQAIQEKVRLNVRVIKIQQDVKEVTVTYQTPAKNLSYVTADYVIVCTTSGAARRIKFEPPLPLKKAHALRSVHYRSGTKIFLTCTKKFWEDDGIHGGKSITDRPSRLIHYPNHNFPNGIGVLVIFTIADDADFFLALDNKTIADIVIHDLSLIHQLPKEKIRDLCYVSMIQKWSLDKYAMGGITTFTPYQFQHFSEALTAPVDRIYFAGEYTAQAHGWIDSTIKSGLTAARDVNRASENPSGIHLSNDNEL | Horned desert vip | Cytotoxic effects | MTT assay | MCF-7 | Not found | IC50 : 4 µg/mL |
| dbacp03572 | L17A | KWKSFLKTFKSAKKTVAHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : > 83.6 µMo/L |
| dbacp03580 | L17A/L21A | KWKSFLKTFKSAKKTVAHTAAKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : > 83.6 µMo/L |
| dbacp03591 | L21A | KWKSFLKTFKSAKKTVAHTAAKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 70.8 µMo/L |
| dbacp03615 | L6A | KWKSFAKTFKSAKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 62.3 µMo/L |
| dbacp03623 | L6A/L17A | KWKSFAKTFKSAKKTVAHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : >83.6 µMo/L |
| dbacp03742 | LfcinB (Bovine lactoferricin) | FKCRRWQWRM | Not found | Inducing apoptosis | MTT assay | MCF-7 | Leukemia | Not found |
| dbacp03753 | LHRH–BH3 peptide luteinizing hormone-releasing hormone (LHRH) | QHWSYGLRPGMGQVGRQLAIIGDDINRRY | Effectors (BAK, BAX) | Inducing apoptosis | Cytotoxicity assay, MTT assay | MCF-7 | Human breast cancer | Not found |
| dbacp04129 | LK-L1C/K6W/L8C | CKKLLWLCKKLLKLAG | Not found | Inducing apoptosis | MTS assay | MCF-7 | Not specified | Not found |
| dbacp04130 | LK1 (Temporin-1CEa Analog peptide) | FVDLKKIANIINSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 20.97 µM |
| dbacp04133 | LK2(5) (Temporin-1CEa Analog peptide) | FKDLKKIANIINSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 44.7 µM |
| dbacp04136 | LK2(6) (Temporin-1CEa Analog peptide) | FVKLKKIANIINSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 15.54 µM |
| dbacp04139 | LK2(6)A(L) (Temporin-1CEa Analog peptide) | FVKLKKILNIINSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 9.01 µM |
| dbacp04142 | LK2(6)AN(2L) (Temporin-1CEa Analog peptide) | FVKLKKILNIILSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 11 µM |
| dbacp04145 | LK3 (Temporin-1CEa Analog peptide) | FKKLKKIANIINSIFKK | Synthetic construct | Cell membrane disintegration | MTT-assay | MCF-7 | Breast cancer | IC50 : 27.72 µM |
| dbacp04148 | LL 37 | LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES | Also known human cathelicidin | Plasma membrane perturbations | MTT/MTS assay | MCF-7 | Breast cancer | LC50 : 21 at 100 µM |
| dbacp04311 | Lunasin | SKWQHQQDSCRKQLQGVNLTPCEKHIMEKIQGRGDDDDDDDDD | Soyabean | Cell membrane degradation | TUNEL DNA fragmentation assay | MCF-7 | Breast cancer | Not found |
| dbacp04314 | Lunasin | SKWQHQQDSCRKQLQGVNLTPCEKHIMEKIQGRGDDDDDDDDD | Soyabean | Apoptosis inducing; Anti-proliferative | MTT/MTS | MCF-7 | Not specified | IC50 : 431.9 µM |
| dbacp04495 | Magainin 2 | GIGKFLHSAKKFGKAFVGEIMNS | African clawed frog | Dissipate ion gradients; Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | IC50 : >200 µg/ml |
| dbacp04513 | Magainin A | AIGKFLHSAKKFGKAFVGEIMNS | African clawed frog | Dissipate ion gradients; Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | IC50 : 49 µg/ml |
| dbacp04523 | Magainin B | GIGKFLHAAKKFAKAFVAEIMNS | African clawed frog | Dissipate ion gradients; Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | IC50 : 37 µg/ml |
| dbacp04539 | Magainin G | GIGKFLHSAKKFAKAFVAEIMNS | African clawed frog | Dissipate ion gradients; Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | IC50 : 42 µg/ml |
| dbacp04543 | Malanin chain A | DYPKLTFTTS | Plant sources | Inducing apoptosis | MTT assay | MCF-7 | Leukemia | IC50 : 11.20 ± 0.02 nM |
| dbacp04549 | Malanin chain B | DETCTDEEFN | Plant sources | Inducing apoptosis | MTT assay | MCF-7 | Leukemia | IC50 : 11.20 ± 0.02 nM |
| dbacp04553 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : >80% at 25 µM |
| dbacp04554 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : ~50% at 50 µM |
| dbacp04555 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : <40% at 75 µM |
| dbacp04556 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : >20% at 100 µM |
| dbacp04557 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : ~100% at 25 µM |
| dbacp04558 | MAP-04-03 | KWLRRVWRWWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | IC50 :61.5 µM |
| dbacp04559 | MAP-04-04 | KRLRRVWRRWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : > 80% at 50 µM |
| dbacp04560 | MAP-04-04 | KRLRRVWRRWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : > 80% at 75 µM |
| dbacp04561 | MAP-04-04 | KRLRRVWRRWR | Analogs of Ixosin-B amide | Disrupting the integrity of cell membrane | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability : > 80% at 100 µM |
| dbacp04563 | Mastoparan | INLKALAALAKKIL | Venom base | Inducing apoptosis | Not specified | MCF-7 | Not specified | IC50 : 432.5 ± 10.9 µM |
| dbacp04577 | Mastoparan-C | LNLKALLAVAKKIL | European hornet | Apoptosis | MTT assay | MCF-7 | Human Breast cancer | IC50 : 1.4 μM |
| dbacp04582 | Mastoparan-Cimals. XXA; UCLL1c) | LNLKALLAVAKKIL | Venom, the European Hornet | Inducing apoptosis | MTT cell viability assay and Lactate dehydrogenase (LDH) leakage assay | MCF-7 | Breast cancer | MIC : 6.26 - 36.65 μM |
| dbacp04588 | Mastoparan-Cimals. XXA; UCLL1c) | LNLKALLAVAKKIL | Venom, the European Hornet | Inducing apoptosis | MTT cell viability assay and Lactate dehydrogenase (LDH) leakage assay | MCF-7 | Breast cancer | IC50 : < 4 μM |
| dbacp04713 | mt_E17L/L22 W/P27A | LTFSDWWKLLAE | MDM3 | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 15.1 µM |
| dbacp04714 | mt_L22 W/P27A | ETFSDWWKLLAE | MDM2 | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 16.3 µM |
| dbacp04715 | mt_S20A/L22 W/P27A | ETFADWWKLLAE | MDM5 | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 8.7 µM |
| dbacp04716 | mt_T18S/L22 W/P27A | ESFSDWWKLLAE | MDM4 | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 27 µM |
| dbacp04929 | NRC-03 | GRRKRKWLRRIGKGVKIIGGAALDHL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7 | Breast cancer | 70% Cytotoxic at 50 µM |
| dbacp04930 | NRC-03 | GRRKRKWLRRIGKGVKIIGGAALDHL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7-TX400 | Breast cancer | 60-70% Cytotoxic at 50 µM |
| dbacp04931 | NRC-03 | GRRKRKWLRRIGKGVKIIGGAALDHL-NH2 | PseudopWinter flounder | Cell membrane damage | MTT/MTS assay | MCF-7-TX400 | Breast cancer | 60-70% Cytotoxic at 50 µM |
| dbacp04952 | NRC-03 | GRRKRKWLRRIGKGVKIIGGAALDHL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7 | Breast cancer | 70% Cytotoxic at 50 µM |
| dbacp04974 | NRC-07 | RWGKWFKKATHVGKHVGKAALTAYL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7 | Breast cancer | 70% Cytotoxic at 50 µM |
| dbacp04975 | NRC-07 | RWGKWFKKATHVGKHVGKAALTAYL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7-TX400 | Breast cancer | 60-70% Cytotoxic at 50 µM |
| dbacp04996 | NRC-13 | GWRTLLKKAEVKTVGKLALKHYL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7 | Breast cancer | 0% Cytotoxic at 50 µM |
| dbacp04997 | NRC-13 | GWRTLLKKAEVKTVGKLALKHYL | Skin mucous secretion of winter flounder | Cell membrane damage | MTT/MTS assay | MCF-7-TX400 | Breast cancer | ~5% Cytotoxic at 50 µM |
| dbacp04998 | NuBCP-9 | FSRSLHSLL | Not found | Inducing apoptosis | Not specified | MCF-7 | Not specified | Not found |
| dbacp05000 | NuBCP-9 (DR8) | FSRSLHSLLRRRRRRRR | Not found | Inducing apoptosis | XTT assat | MCF-7 | Breast cancer | IC50 : 7.11 μM |
| dbacp05023 | Peptide P | KWKSFLKTFKSAKKTVLHTALKAISS | PeptideV13K | Membrane disruption mechanism | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 15.8 µMo/L |
| dbacp05036 | p120RasGAP (317-326) | WMWVTNLRTD | Not found | Inducing apoptosis | Luciferase assay | MCF-7 | Human malignant mesothelomia | Not found |
| dbacp05037 | P160 | VPWMEPAYQRFL | Not found | Apoptosis inducing | MTT cytotoxicity assay | MCF-7 | Breast cancer | IC50 : 14.2 ± 1.5 μM |
| dbacp05080 | p53-C terminal peptide | GSRAHSSHLKSKKGQSTSRHKK | Not found | Inducing apoptosis | Annexin V-FITC Binding assay | MCF-7 | Breast cancer | Not found |
| dbacp05081 | p53-C terminal peptide | GSRAHSSHLKSKKGQSTSRHKK | Not found | Inducing apoptosis | Annexin V-FITC Binding assay | MCF10-2A | Breast cancer | Not found |
| dbacp05106 | PA10 | RQIKIWFQNRRMKWKKGGGGNNETTSIQIAGSLHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05110 | PA15 | RQIKIWFQNRRMKWKKGGSLSAACHEQWSLGAQHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05114 | PA2 | RQIKIWFQNRRMKWKKGGATRPRVDTQPELCGMHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05118 | PA3 | RQIKIWFQNRRMKWKKGGDCLCISRRARLLRATHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05122 | PA38 | RQIKIWFQNRRMKWKKGGKYNGRFTTHHLLHLLNHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05126 | PA49 | RQIKIWFQNRRMKWKKGGAGVYTFLVGADNRGWEHHHHHH | Synthetic construct | Cell proliferation inhibition; Cell penetration; Apoptosis | Cell viability assay | MCF10A | Breast cancer | MIC : 10 μM |
| dbacp05250 | Pep27 | MRKEFHNVLSSGQLLADKRPARDYNRK | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : > 70 µM |
| dbacp05255 | Pep27 | MRKEFHNVLSSGQLLADKRPARDYNRK | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : > 70 µM |
| dbacp05256 | Pep27 | MRKEFHNVLSSGQLLADKRPARDYNRK | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : > 70 µM |
| dbacp05261 | Pep27 anal1 | MWKWFHNVLSSWQLLADKRPARDYNRK | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 55 µM |
| dbacp05266 | Pep27 anal2 | MWKWFHNVLSWWWLLADKRPARDYNRK | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : < 10 µM |
| dbacp05271 | Pep27 anal3 | MRKWFHNVLSSGQLLADKWPAWDYNRK | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 38 µM |
| dbacp05276 | Pep27 anal4 | MWKEFHNVLSSGQLLADKRWARWYNRW | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : 29 µM |
| dbacp05281 | Pep27 anal5 | MWKWFHNVLSSGQLLADKWWAWWYNWW | Not found | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | IC50 : > 70 µM |
| dbacp05286 | Pep27anal1 | MWKWFHNVLSSWQLLADKRPARDYNRK | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 55 µM |
| dbacp05291 | Pep27anal2 | MWKWFHNVLSWWWLLADKRPARDYNRK | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : < 10 µM |
| dbacp05296 | Pep27anal3 | MRKWFHNVLSSGQLLADKWPAWDYNRK | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 38 µM |
| dbacp05301 | Pep27anal4 | MWKEFHNVLSSGQLLADKRWARWYNRW | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 29 µM |
| dbacp05306 | Pep27anal5 | MWKWFHNVLSSGQLLADKWWAWWYNWW | Pneumococcus | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : >70 µM |
| dbacp05403 | Peptide Glycyrrhetinic Acid Based Derivatives (compound 5) | GGGG | Not found | Inducing apoptosis | Not specified | MCF-7 | Cervical cancer | IC50 : 5.0 ± 0.3 µg/mL |
| dbacp05484 | Pexiganan | GIGKFLKKAKKFGKAFVKILKK | Analog of African clawed frog | Plasma membrane perturbations | MTT/MTS assay | MCF-7 | Breast cancer | LC50 : 8 at 100 µM |
| dbacp05534 | Phylloseptin-PBa1 | FLSLIPHIASGIASLVKNF | Burmeister's leaf frog, Brazil, South America | Disruption of cell membranes | MTT cell viability assay | MCF-7 | Breast cancer | IC50 : approx. 0.29 µM |
| dbacp05545 | Phylloseptin-PBa2 | FLSLLPHIASGIASLVSKF | Burmeister's leaf frog, Brazil, South America | Disruption of cell membranes | MTT cell viability assay | MCF-7 | Breast cancer | IC50 : approx. 0.50 µM |
| dbacp05552 | Phylloseptin-PHa | FLSLIPAAISAVSALANHF | Northern orange-legged leaf frog | Disruption of the membrane | MTT assay, Lactate dehydrogenase (LDH) assay | MCF-7 | Human breast cancer | LD50 : < 5 µM |
| dbacp05665 | Protein GPR15LG (Antimicrobial peptide with 57 amino acid residues) (AP-57) (Antimicrobial peptide-57) (Colon-derived SUSD2 binding factor) (CSBF) (Protein GPR15 ligand) (Protein GPR15L) (Secreted protein C10orf99) | MRLLVLSSLLCILLLCFSIFSTEGKRRPAKAWSGRRTRLCCHRVPSPNSTNLKGHHVRLCKPCKLEPEPRLWVVPGALPQV | Human | Cytotoxic effects | SDS-PAGE assay | MCF-7 | Colorectal cancer | Not found |
| dbacp05712 | PTP1 | LLAGLAANFLPTIICKISYKC | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : >100 µg/ml |
| dbacp05717 | PTP2 | FAGLAANFLPTIICKISYKC | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : >100 µg/ml |
| dbacp05722 | PTP4 | FLKLLKKLAAKFLPTIICKISYKC | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 18.1 µg/ml |
| dbacp05727 | PTP5 | FLKLLKKLAAKLF | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 5.43 µg/ml |
| dbacp05732 | PTP6 | FLKLLKKLAAKLF | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 17.56 µg/ml |
| dbacp05737 | PTP7 | FLGALFKALSKLL | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 5.25 µg/ml |
| dbacp05742 | PTP8 | FLKLLAGLLKNFA | Skin of a Korean frog, Wrinkled frog | Induce apoptosis | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 32.23 µg/ml |
| dbacp05812 | R2PLx-22 | GIMDTVKNAAKNLAGQLLDKLK | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Lung cancer | IC50 : 109.30 µM |
| dbacp05813 | R2PLx-22 | GIMDTVKNAAKNLAGQLLDKLK | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Prostate cancer | IC50 : 109.30 µM |
| dbacp05814 | R2PLx-22 | GIMDTVKNAAKNLAGQLLDKLK | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Breast cancer | IC50 : 109.30 µM |
| dbacp05815 | R2PLx-22 | GIMDTVKNAAKNLAGQLLDKLK | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Glioma | IC50 : 109.30 µM |
| dbacp05863 | RA-V | cyclopeptideRA-V-,cyclo(YAAYAY) | Plant sources | Inducing apoptosis | MTT assay | MCF-7 | Breast cancer | Not found |
| dbacp05873 | Radical SAM domain protein | MEAVLYVTRKCNLSCGHCIVDKEDNSDLPTDKVETLASDYPIDRTILSGGEPFLHDNFEELVALVPEPTVLSNGLVLSDEEYVGENSDMLEELNGIQLSVEGKEETTDARRGEGVWDRVMEAHQNLSEIGVESYLRSTYSREMMEEVGELMEFCDAEGISLVLFPEIGKPPLSPTENASFFDYAVEKGVVVATPDFHSYIGEGGECPAARTRISVDVNGEIYPCQFNWDYCLGEVGDEWGLIESRIERFDRTEPVPRTCSRCDFANKCRGCGVADTWSGCPIARGLSHSESPSRRPLKRVQETMNTLEDVGAPRGCHGC | Uncultured archaeon | Apoptosis inducing | MTT assay | MCF-7 | Breast cancer | MIC : 42% ± 8.1 μM |
| dbacp05893 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCKITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7) | Lung cancer | IC50 : 20.19 µM |
| dbacp05894 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCKITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7) | Prostate cancer | IC50 : 20.19 µM |
| dbacp05895 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCKITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7) | Breast cancer | IC50 : 20.19 µM |
| dbacp05896 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCKITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7) | Glioma | IC50 : 20.19 µM |
| dbacp05905 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCKITAC | Gram-negative purple non-sulfur bacteria | Inducing apoptosis | MTT Cell viability assay and Lactate dehydrogenase (LDH) leakage assay | MCF-7 | Human breast cancer | IC50 : 20.19 µM |
| dbacp05910 | Ranatuerin-2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Skin secretions, the pickerel frog, North America | Inducing apoptosis | MTT Cell viability assay and Lactate dehydrogenase (LDH) leakage assay | MCF-7 | Breast cancer | IC50 : 20.19 µM |
| dbacp05961 | RGD-mda-7 | MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSGAQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQNVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNFVLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAFKQLDVEAALTKALGEVDILLTWMQKFYKL | Derived from wtmda-7/IL-24 by insertion or a glycine residue between Arg(164) and Asp(165). | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability(% of control):0.5 at concentration 4 µg/ml |
| dbacp05963 | RGD-mda-7 | MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSGAQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQNVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNFVLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAFKQLDVEAALTKALGEVDILLTWMQKFYKL | Derived from wtmda-7/IL-24 by insertion or a glycine residue between Arg(164) and Asp(165). | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | Apoptotic rate(%): >70% at concentration of 8 µg/ml |
| dbacp06000 | S−24-R2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Lung cancer | IC50 : 316.90 µM |
| dbacp06001 | S−24-R2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Prostate cancer | IC50 : 316.90 µM |
| dbacp06002 | S−24-R2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Breast cancer | IC50 : 316.90 µM |
| dbacp06003 | S−24-R2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Not found | Inducing apoptosis | MTT and LDH assay | MCF-7 | Glioma | IC50 : 316.90 µM |
| dbacp06119 | SK84 | SQLGDLGSGAGQGGGGGGSIRAAGGAFGKLEAAREEEFFYKKQKEQLERLKNDQIHQAEFHHQQIKEHEEAIQRHKDFLNNLHK | Fruit fly | Cell membrane disintegration | MTS/PES colorimetric assay | MCF-7 | Liver cancer | IC50 : 50 μM |
| dbacp06120 | SK84 | SQLGDLGSGAGQGGGGGGSIRAAGGAFGKLEAAREEEFFYKKQKEQLERLKNDQIHQAEFHHQQIKEHEEAIQRHKDFLNNLHK | Fruit fly | Cell membrane disintegration | MTS/PES colorimetric assay | MCF-7 | Breast cancer | IC50 : 50 μM |
| dbacp06125 | SK84 | SQLGDLGSGAGQGGGGGGSIRAAGGAFGKLEAAREEEFFYKKQKEQLERLKNDQIHQAEFHHQQIKEHEEAIQRHKDFLNNLHK | Fruit fly | Destroying the cell membranes | Cell proliferation assay | MCF-7 | Breast cancer | MIC : 4 – 8 mM |
| dbacp06140 | SP22 | ACHWPWCHGWHSACDLPMHPMC | Not found | Inducing apoptosis | Tunnel assay | MCF-7 | Breast cancer | Not found |
| dbacp06171 | SVS-1 | KVKVKVKVpPTKVKVKVK | Synthetic peptide | Disruption of cell membranes | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 8.1 ± 0.8 µM |
| dbacp06175 | SVS-2 | KVKVKVKVPPTKVKVKVK | Synthetic peptide | Disruption of cell membranes | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : >100 µM |
| dbacp06187 | t Mastoparan-C(tMP-C, Tat (49-57)-Mastoparan-C) | RKKRRQRRRLNLKALLAVAKKIL | Synthetic construct | Apoptosis inducing | MTT assay | MCF-7 | Human breast cancer | IC50 : 3.70 μM |
| dbacp06220 | TAT-RasGAP (317-326) From p120RasGAP | GRKKRRQRRRGGWMWVTNLRTD | Not found | Inducing apoptosis | Luciferase assay | MCF-7 | Human malignant mesothelomia | Not found |
| dbacp06233 | Temporin-1CEa | FVDLKKIANIINSIF | Chinese brown frog | Membrane disruption | MTT/MTS assay | MCF-7 | Breast cancer | 61% cell viability at 40 µM |
| dbacp06234 | Temporin-1CEa | FVDLKKIANIINSIF | Chinese brown frog | Membrane disruption | LDH leakage assay | MCF-7 | Breast cancer | 32% cytotoxicity at 40 µM |
| dbacp06237 | Temporin-1CEa | FVDLKKIANIINSIF | Chinese brown frog | Membrane disruption | MTT/MTS assay | MCF-7 | Breast cancer | MIC : 40 µM |
| dbacp06238 | Temporin-1CEa | FVDLKKIANIINSIF | Chinese brown frog | Membrane disruption | LDH leakage assay | MCF-7 | Breast cancer | MIC : 40 µM |
| dbacp06242 | Temporin-1RNa | ILPIRSLIKKLL | The black-spotted frog, Northeastern China, Asia | Disruption of membrane | Cytotoxicity assay, MTT/MTS assay | MCF 7 | Breast cancer | IC50 : 23.4 ± 5.2 µM |
| dbacp06244 | Temporin-1RNb | FLPLKKLRFGLL | The black-spotted frog, Northeastern China, Asia | Disruption of membrane | Cytotoxicity assay, MTT/MTS assay | MCF 7 | Breast cancer | IC50 : 11.4 ± 2.3 µM |
| dbacp06295 | Tetramer of peptide-paclitaxel conjugate | (K-Aib-C(CH2CO-2'-Pac))4 | Synthetic peptide paclitaxel conjugate | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 0.64 nM |
| dbacp06327 | Transactivator of transcript-DV1-Bcl-2, AT-DV1-BH3 | RRRQRRKKRGGGGLGASWHRPDK | Transactivator of transcript-DV1-Bcl-2 TAT-DV1-BH4 | Apoptosis inducing | Cell viability assay, Transwell invasion assay | MCF-7 | Breast cancer | Not specified |
| dbacp06348 | Trimer of peptide-paclitaxel conjugate | (K-Aib-C(CH2CO-2'-Pac))3 | Synthetic peptide paclitaxel conjugate | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 3.00 nM |
| dbacp06362 | TsAP-2 | FLGMIPGLIGGLISAFK | Venom-derived cDNAlibrary of the Brazilian yellow scorpion | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 6.4 µM |
| dbacp06370 | TsAP-S1 | FLSLIPKLVKKIIKAFK | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 1.8 µM |
| dbacp06378 | TsAP-S2 | FLGMIPKLIKKLIKAFK | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | Not specified | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 1.8 µM |
| dbacp06416 | U3 | NGSIPATWASL | Date palm | Cell proliferation inhibition | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 555 μM |
| dbacp06419 | U7 | NCSIHGDIPAY | Date palm | Cell proliferation inhibition | MTT/MTS assay | MCF-7 | Breast cancer | IC50 : 554 μM |
| dbacp06534 | wtmda-7/IL-24 | MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSGAQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQNVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNFVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAFKQL | Not found | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | Cell viability (% of control):0.5 at concentration 7 µg/ml |
| dbacp06536 | wtmda-7/IL-24 | MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSGAQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQNVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNFVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAFKQL | Not found | Apoptosis inducing | MTT/MTS assay | MCF-7 | Breast cancer | Apoptotic rate(%) : > 50% at concentration of 8 µg/ml |
| dbacp06543 | XLAsp-P1 | DEDDD | Skin, African clawed frog, Africa | Destruction of the cell membrane | MTT assay | MCF-7 cells | Breast cancer | LC50 : < 5 μg/mL |
| dbacp06565 | Z24 | ALSKALSKALSKALSKALSKALSK | African clawed frog | Dissipate ion gradients; Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | Not found |
| dbacp06581 | Z44 | ALSKALSKALSKALSKALSKALSK | African clawed frog | Dissipate ion gradients;Induce osmotic lysis; Membrane damage | Trypan blue assay | MCF-7 | Breast cancer | Not found |
| dbacp06616 | LA3IK | LAIAVK | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 90.23 ± 7.32 µM |
| dbacp06620 | D-LA3IK | laiavk | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 91.2 ± 8.21 µM |
| dbacp06624 | LA3IK-SCR | LAKAVI | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 133 ± 9.52 µM |
| dbacp06628 | RP-7 | RPPCVIL | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 110.12 ± 4.23 µM |
| dbacp06632 | D-RP-7 | rppcvil | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 90 ± 10.31 µM |
| dbacp06636 | RP7 SCR | RPPLVIC | Migration and invasion enhancer 1 (MIEN1) | Targeting the MIEN1 signaling pathway | MTT assay | MCF-7 | Breast Cancer | IC50 = 150 ± 10.32 µM |
| dbacp06641 | C-Mel | CGIGAVLKVLTTGLPALISWIKRKRQQ | Synthetic analogue | Plasma memberane pore formation | MTT assay | MCF-7 | Breast Cancer | IC50 = 110.59 µg/mL |
| dbacp06644 | CM–FA | CGIGAVLKVLTTGLPALISWIKRKRQQ | Synthetic analogue | Plasma memberane pore formation | MTT assay | MCF-7 | Breast Cancer | IC50 = 10.38 µg/mL |
| dbacp06647 | Mel-C | GIGAVLKVLTTGLPALISWIKRKRQQC | Synthetic analogue | Plasma memberane pore formation | MTT assay | MCF-7 | Breast Cancer | IC50 = 160.62 µg/mL |
| dbacp06650 | MC–FA | GIGAVLKVLTTGLPALISWIKRKRQQC | Synthetic analogue | Plasma memberane pore formation | MTT assay | MCF-7 | Breast Cancer | IC50 = 12.63 µg/mL |
| dbacp06673 | Crabrolin | FLPLILRKIVTAL | European hornet (Vespa crabro) | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 26.49 μM |
| dbacp06678 | Crabrolin-4R | FLPRILRKIVTAL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 20.26 μM |
| dbacp06683 | Crabrolin-4K | FLPKILRKIVTAL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 23.18 μM |
| dbacp06688 | Crabrolin-TR | FLPRILRKIVRAL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 3.459 μM |
| dbacp06693 | Crabrolin-FR | RLPRILRKIVRAL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 33.85 μM |
| dbacp06698 | Crabrolin-AR | RLPRILRKIVRRL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 32.51 μM |
| dbacp06703 | Crabrolin-PR | RLRRILRKIVRRL | Synthetic Analog of Crabrolin | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 12.29 μM |
| dbacp06722 | GE18 | GAGIVVASIDTGVRVSHE | Aphanomyces invadans | Not available | MTT assay | MCF-7 | Breast Cancer | IC50 = 35.34 µM |
| dbacp06744 | M1-20 | grrrqrrkkrlgpfsidllikslsdnmtdl | Synthetic | Inhibits FOXM1 transcriptional activities | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 31.05 µM |
| dbacp06791 | PS9 | PSRKVMLWS | Aphanomyces invadans | Reactive Oxygen Species and Apoptotic Pathways | Neutral Red Uptake assay | MCF-7 | Breast Cancer | IC50 value range between 25.27 - 43.28 μM |
| dbacp06792 | PS9 | PSRKVMLWS | Aphanomyces invadans | Reactive Oxygen Species and Apoptotic Pathways | LDH leakage assay | MCF-7 | Breast Cancer | 71.25 ± 1.3% LDH release at 40 μM |
| dbacp06796 | LHRH-BinBC | QHWSYGLRPGGRGPKDAVRAVKGSALLPCIIVHDPNLNNSDKMKFNTYYLLEYKEYWHQLWSQIIPAHQTVKIQERTGISEVVQNSMIEDLNMYIGADFGMYFYLRSSGFKEQITRGLNRPLSQTTTQLGERVEEMEYYNSNDLDVRYVKYALAREFTLKRVNGEIVKNWVAVDYRMAGIQSYPNAPITNPLTLT | Synthetic | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 10.96 μM |
| dbacp06797 | LHRH-BinBC | QHWSYGLRPGGRGPKDAVRAVKGSALLPCIIVHDPNLNNSDKMKFNTYYLLEYKEYWHQLWSQIIPAHQTVKIQERTGISEVVQNSMIEDLNMYIGADFGMYFYLRSSGFKEQITRGLNRPLSQTTTQLGERVEEMEYYNSNDLDVRYVKYALAREFTLKRVNGEIVKNWVAVDYRMAGIQSYPNAPITNPLTLT | Synthetic | Apoptosis inducing | LDH leakage assay | MCF-7 | Breast Cancer | 40% LDH efflux at 16 µM |
| dbacp06806 | [C/U, G1K, L5Y, K8R]cGm | KURRYUYRQRUVTYURGR | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 29.0 ± 3.7 μM |
| dbacp06812 | [G1K, L5Y, K8R]cGm | KCRRYCYRQRCVTYCRGR | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 15.2 ± 1.9 μM |
| dbacp06822 | [C/U]cGm | GURRLUYKQRUVTYURGR | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 37.5 ± 3.3 μM |
| dbacp06828 | [G1K, K8R]cGm | KCRRLCYRQRCVTYCRGR | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 6.7 ± 0.7 μM |
| dbacp06834 | [R4A, R18A]cGm | GCRALCYKQRCVTYCRGA | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 48.4 ± 0.7 μM |
| dbacp06840 | [Y7W, K8R, Y14W]cGm | GCRRLCWRQRCVTWCRGR | Synthetic Analogue of Gomesin | Cell membrane penetration | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 15.1 ± 1.4 μM |
| dbacp06870 | LfcinB(21-25)Pal | RWQWRWQWR | LfcinB | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 81 µM |
| dbacp06871 | RR-1-RR | RRWQWRWQWRR | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 58 µM |
| dbacp06873 | R-1-RR | RWQWRWQWRR | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 122 µM |
| dbacp06875 | RR-1-R | RRWQWRWQWR | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 68 µM |
| dbacp06877 | 1 | WQWRWQW | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 105 µM |
| dbacp06879 | R-1 | RWQWRWQW | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 58 µM |
| dbacp06881 | 1-R | WQWRWQWR | Synthetic analogue of LfcinB(21-25)Pal | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 130 µM |
| dbacp06925 | #2(D33-N52) | RRRRRRRRGGDRDYKKFWAGLQGLTIYFYN | STAP-2 PH domain–derived peptide | Inhibition of cell signalling | CellTiter-Glo assay | MCF-7 | Breast Cancer | Graph figure 1-B |
| dbacp06928 | #6(M108-L127) | RRRRRRRRGGMWKGFILTVVELRVPTDLTL | STAP-2 PH domain–derived peptide | Inhibition of cell signalling | CellTiter-Glo assay | MCF-7 | Breast Cancer | Graph figure 1-B |
| dbacp06978 | C16-E4Y | EEEEY | Synthetic | Inhibition of cell signalling | WST-8 assay | MCF-7 | Breast Cancer | 50 % cell viability at 0.05 wt % |
| dbacp07007 | ST101 | vaeareelerlearlgqargelkkwkmrrnqfwlklqr | Synthetic | Prevents C/EBPβ dimerization, induces degradation | Annexin V/ PI staining assay | MCF-7 | Breast Cancer | mean EC50 value of 2.1 ± 0.4 μmol/L |
| dbacp07023 | [G10a]-SHa | FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MCF-7 | Breast Cancer | IC50 = 15.05 ± 8.51 µM |
| dbacp07030 | [G10a]2-SHa | FLSGIVGMLaKLFKFLKaLMFLSGIVG | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MCF-7 | Breast Cancer | IC50 = 5.69 ± 1.46 µM |
| dbacp07037 | [G10a]3-SHa | FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MCF-7 | Breast Cancer | IC50 = 3.77 ± 0.12 µM |
| dbacp07044 | Jeff-[G10a]2-SHa | FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF | Analog of temporin SHa | Dendrimerization enhances stability, selectivity, anticancer efficacy | Resazurin dye assay | MCF-7 | Breast Cancer | IC50 = 35.71 ± 8.50 µM |
| dbacp07110 | Nigrocin-M1 | GLLGKILGAGKKVLLGVSGLL | Synthetic | Membrane disruption mediates selective cytotoxicity. | MTT assay | MCF-7 | Breast Cancer | IC50 = 24.60 μM |
| dbacp07113 | Galaxamide | (N-Me-L)L(N-Me-L)LL | Galaxaura filamentosa | Cell-cycle arrest induces apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 11.33 ± 2.95 µg/ml |
| dbacp07117 | Z-1 | L(N-Me-L)LPL | Synthetic | Cell-cycle arrest induces apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 5.85 ± 1.28 µg/ml |
| dbacp07243 | RB4 | MADSERLSAPGCWAACTNFSRTRK | Derived from protein PLP2 | F-actin modulation induces necrotic death. | MTT assay | MCF-7 | Breast Cancer | EC50 = 0.724 ± 0.340 mol/L × 10-3 |
| dbacp07283 | AtMP1 | THPPTTTTTTTTTTTTTAAPATTT | Anabastestudineus skin mucus fraction 2 | p53-mediated Bax/Bcl-2 apoptosis activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 8.25 ± 0.14 μg/ml |
| dbacp07285 | AtMP2 | TGIATSGLATFTLHTGSLAPAT | Anabastestudineus skin mucus fraction 2 | p53-mediated Bax/Bcl-2 apoptosis activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 5.89 ± 0.14 μg/ml |
| dbacp07310 | LyeTxI-b | IWLTALKFLGKNLGKLAKQQLAKL | Synthetic | Apoptosis induction and immune modulation. | MTT assay | MCF-7 | Breast Cancer | IC50 = 7.34 ± 3.09 µM |
| dbacp07315 | B1OS-L | FLPLIASLAGNVVPKIFCKITKRC | B-1OS | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 8.883 µM |
| dbacp07320 | B1OS-D-L | FlPLIASLAGNVVPKIFCKITKRC | B-1OS | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 3.17 µM |
| dbacp07347 | GA - 2 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 7.70 ± 1.3 µg/mL |
| dbacp07349 | GA - 3 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 5.1 ± 0.7 µg/mL |
| dbacp07351 | GA - 4 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 6.10 ± 0.4 µg/mL |
| dbacp07353 | GA - 5 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 5.0 ± 0.3 µg/mL |
| dbacp07355 | GA - 7 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 3.70 ± 0.2 µg/mL |
| dbacp07358 | GA - 8 | Structure given in figure | Synthetic (glycyrrhetinic acid (GA)-based peptides) | Apoptosis induction, Bax/p53/caspase activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 6.90 ± 1.1 µg/mL |
| dbacp07363 | Pal-N-Ter-TAT | Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ | Analogue of N-terminal fragment of the VDAC1 protein | Mitochondrial targeting, VDAC1-HKII dissociation | MTT assay | MCF-7 | Breast Cancer | IC50 = 27.26 μM |
| dbacp07376 | Brevinin-2DYd | GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC | Rana dybowskii | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 25.74 µg/ml |
| dbacp07380 | Ranatuerin-2Lb | GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC | Rana luteiventris | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 45.25 µM |
| dbacp07384 | Odorranain-C1 | GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC | Odorrana grahami | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 41.21 µM |
| dbacp07388 | Brevinin-2DYb | GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC | Rana dybowskii | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 37.84 µM |
| dbacp07392 | Ranatuerin-2 | GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP | Rana catesbeiana | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 > 128 µM |
| dbacp07397 | Pugnin A | RLMRIFRILKLAR | Synthetic | Membrane disruption induces necrotic death | MTT assay | MCF-7 | Breast Cancer | 12% Cytotoxicity at 100 µM |
| dbacp07399 | Pugnin B | RMMRIFWVIKLAR | Synthetic | Membrane disruption induces necrotic death | MTT assay | MCF-7 | Breast Cancer | 5% Cytotoxicity at 100 µM |
| dbacp07403 | Pep | GKLRLIKKLWVKKWKKKGWKA | Synthetic | Membrane disruption induces necrotic death | MTT assay | MCF-7 | Breast Cancer | IC50 = 2 µM |
| dbacp07411 | Si1 | (KLAKLAK)2 | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 124.1 ± 8.12 µM |
| dbacp07413 | Si3 | KL(Beta-A)KL(Beta-A)AK | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 176.3 ± 4.66 µM |
| dbacp07414 | Si2 | KL(Beta-A)KL(Beta-A)K | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 662.9 ± 20.02 µM |
| dbacp07417 | Si11 | KL(Beta-A)KLAK | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 228.8 ± 7.18 µM |
| dbacp07418 | Si13 | KnLAKnLAK | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 1704 ± 112 µM |
| dbacp07419 | Si14 | KnLAKnLAK | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 593.3 ± 60.3 µM |
| dbacp07421 | Si15 | KnLAKnLAK | Synthetic | Membrane disruption induces cancer apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 140.3 ± 7.12 µM |
| dbacp07432 | [Arg]3-VmCT1 | FLRALWNVAKSVF | Synthetic | Membrane disruption via cationic interaction | MTT assay | MCF-7 | Breast Cancer | IC50 = 20.6 ± 3.1 μmol/L |
| dbacp07433 | [Arg]7-VmCT1 | FLGALWRVAKSVF | Synthetic | Membrane disruption via cationic interaction | MTT assay | MCF-7 | Breast Cancer | IC50 = 18.0 ± 2.7 μmol/L |
| dbacp07434 | [Arg]11-VmCT1 | FLGALWNVAKRVF | Synthetic | Membrane disruption via cationic interaction | MTT assay | MCF-7 | Breast Cancer | IC50 = 25.8 ± 5.2 μmol/L |
| dbacp07440 | A4K14 - Citropin 1.1 - Sp 7 | GLFAVR8KKVASVS5KGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 12.1 µM |
| dbacp07444 | A4K14 - Citropin 1.1 - Sp 6 | GR8FAVIKKS5ASVIKGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 23.78 µM |
| dbacp07448 | A4K14 - Citropin 1.1 - Sp 5 | GLFAVIKKVAS5VIKS5L | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 12.42 µM |
| dbacp07452 | A4K14 - Citropin 1.1 - Sp 4 | GLFAVIKKS5ASVS5KGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 10.49 µM |
| dbacp07456 | A4K14 - Citropin 1.1 - Sp 3 | GLFAVS5KKVS5SVIKGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 11.92 µM |
| dbacp07460 | A4K14 - Citropin 1.1 - Sp 2 | GLFAS5IKKS5ASVIKGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 12.65 µM |
| dbacp07464 | A4K14 - Citropin 1.1 - Sp 1 | GS5FAVS5KKVASVIKGL | Synthetic | Stapled peptide enhances helical apoptosis | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 11.26 µM |
| dbacp07473 | MzDef | MSSSNCANVCQTENFPGGECKAEGATRKCFCKNC | Zea mays L. | Disulfide-stabilized peptide disrupts pathogens | MTT assay | MCF-7 | Breast Cancer | IC50 = 14.85 µg/mL |
| dbacp07475 | Latcripin-7A | MTTESKVKNATTLLHSGKVKERQEGLSALRNIFSQNSSIERFYNVAGRDGRKPSHEIWAPILDGLQTCIRSEKSAFVTAKKSTDVIEKRLAAAAGTYRWFVEKSMMHFAKKTVLEICHFLYREMKVRETLIPSVALDFIKAYECVASHPPHLARLEEDEIEWEE | Lentinula edodes | Cell-cycle arrest, apoptosis, autophagy induction | CCK-8 assay | MCF-7 | Breast Cancer | IC50 = 91 μg/mL |
| dbacp07491 | Figainin 1 | FIGTLIPLALGALTKLFK | Boana raniceps | Membrane disruption, α-helix mediated | MTT assay | MCF-7 | Breast Cancer | IC50 = 13.7 µM |
| dbacp07496 | RA-3 | RWrGGGGGLFDIIKKIAESF | Synthetic | Integrin-targeting, α-helix mediated lysis | MTT assay | MCF-7 | Breast Cancer | IC50 = 44.14 μM |
| dbacp07500 | Mambalgin-1 | LKCYQHGKVVTCHRDMKFCYHNTGMPFRNLKLILQGCSSSCSETENNKCCSTDRCNK | Dendroaspis polylepsis | ASIC inhibition suppresses cancer proliferation | MTT assay | MCF-7 | Breast Cancer | 22.43% cytotoxicity at 10 µg/mL |
| dbacp07510 | cyclic dipeptide - 2b | WA | Synthetic | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 45.6 µM |
| dbacp07513 | Dermaseptin-PP | ALWKDMLKGIGKLAGKAALGAVKTLV | Phyllomedusa palliata | Membrane disruption triggers dual apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 2.92 μM |
| dbacp07534 | rCT-II | LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN | Naja naja | Apoptosis via intrinsic (mitochondrial) and extrinsic (death receptor) pathways | MTT assay | MCF-7 | Breast Cancer | IC50 = 3.66 µg/mL |
| dbacp07552 | macrocyclic pyridoheptapeptide derivative 1a | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 15.329 ± 0.672 μM |
| dbacp07554 | macrocyclic pyridoheptapeptide derivative 1b | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 10.904 ± 0.534 μM |
| dbacp07556 | macrocyclic pyridoheptapeptide derivative 1c | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 34.894 ± 1.273 μM |
| dbacp07559 | macrocyclic pyridoheptapeptide derivative 2b | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 20.697 ± 0.974 μM |
| dbacp07561 | macrocyclic pyridoheptapeptide derivative 2c | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 24.943 ± 1.082 μM |
| dbacp07563 | macrocyclic pyridoheptapeptide derivative 3a | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 10.316 ± 0.546 μM |
| dbacp07565 | macrocyclic pyridoheptapeptide derivative 3b | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 9.911 ± 0.491 μM |
| dbacp07567 | macrocyclic pyridoheptapeptide derivative 3c | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 22.864 ± 0.992 μM |
| dbacp07569 | macrocyclic pyridoheptapeptide derivative 4a | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 9.304 ± 0.536 μM |
| dbacp07571 | macrocyclic pyridoheptapeptide derivative 4b | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 9.188 ± 0.545 μM |
| dbacp07573 | macrocyclic pyridoheptapeptide derivative 4c | Structure given in Scheme 1 | Synthetic | Macrocyclic peptides disrupt cancer growth | MTT assay | MCF-7 | Breast Cancer | IC50 = 19.552 ± 1.032 μM |
| dbacp07638 | branched tetrapeptide Schiff bases derivative 4a | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07639 | branched tetrapeptide Schiff bases derivative 4b | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07640 | branched tetrapeptide Schiff bases derivative 4c | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07641 | branched tetrapeptide Schiff bases derivative 5c | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07642 | branched tetrapeptide Schiff bases derivative 5d | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07643 | branched tetrapeptide Schiff bases derivative 5e | Figure given in Scheme 1 | Synthetic | p53 stabilization and LDHA inhibition | MTT assay | MCF-7 | Breast Cancer | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM |
| dbacp07647 | AP1-Z1 | FLFSLIPHAISGLISAFK | AcrAP1 from the venom of the Arabian scorpion | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 7.222 μM |
| dbacp07650 | AP1-Z5a | FLFKLIPKAIKGLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | Graph Figure 2A |
| dbacp07653 | AP1-Z5b | FLFKLIKHAIKGLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 1.037 μM |
| dbacp07656 | AP1-Z3a | FLFSLIKHAIKGLISAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | Graph Figure 2A |
| dbacp07659 | AP1-Z3b | FLFSLIKHAISKLISAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | Graph Figure 2A |
| dbacp07662 | AP1-Z7 | FLFKLIKKAIKKLIKAFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | Graph Figure 2A |
| dbacp07665 | AP1-Z9 | FLFKLIKKKIKKLIKKFK | Mutant of APR-Z1 | Charge–hydrophobicity balance drives apoptosis | MTT assay | MCF-7 | Breast Cancer | Graph Figure 2A |
| dbacp07808 | cT1 | KWCFRVCYRGICYRRCRG | Synthetic | Not Available | Resazurin dye assay | MCF-7 | Breast Cancer | CC50 = 6.4 ± 0.6 µM |
| dbacp07849 | Dermaseptin-PT9 | GLWSKIKDAAKTAGKAALGFVNEMV | Phyllomedusa tarsius | Membrane disruption and cationic enhancement | MTT assay | MCF-7 | Breast Cancer | IC50 = 7.44 µM |
| dbacp07854 | K8, 23-DPT9 | GLWSKIKKAAKTAGKAALGFVNKMV | Synthetic | Membrane disruption and cationic enhancement | MTT assay | MCF-7 | Breast Cancer | IC50 = 8.64 µM |
| dbacp07859 | HN-1 | FALGAVTKLLPSLLCMITRKC | Amolops hainanensis | Apoptosis induction and immune activation | MTT assay | MCF-7 | Breast Cancer | IC50 = 6.9 μM |
| dbacp07887 | ICD-85 | Not Available | Active fractions from Gloydius halys and Hemiscorpius lepturus | Caspase-9 mediated apoptotic death | MTT assay | MCF-7 | Breast Cancer | IC50 = 36.45 ± 0.38 μg/mL |
| dbacp07888 | ICD-85 | Not Available | Active fractions from Gloydius halys and Hemiscorpius lepturus | Caspase-9 mediated apoptotic death | Neutral Red Uptake assay | MCF-7 | Breast Cancer | IC50 = 21.97 ± 0.63 μg/mL |
| dbacp07931 | myristoyl-CM4 | GRWKIFKKIEKVGQNIRDGIVKAGPAVAVVGQAATI | Bombyx mori | Cell penetration, Mitochondrial dysfunction, Apoptosis pathway activation | MTT assay | MCF-7 | Breast cancer | IC50 = 6 μM |
| dbacp07944 | TC22 | MTVVLLLIVLPLLGGVHSSGIL | Tribolium castaneum | ROS, p53, mitochondrial apoptosis activation | MTT assay | MCF-7 | Breast Cancer | Fig 4a |
| dbacp07955 | S-24-R2PLx | GIMDTVKNAAKNLAGQLLDKLKCSITAC | Synthetic Analogue of Ranatuerin-2PLx | R2PLx induces caspase-dependent apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 316.90 µM |
| dbacp07958 | Compound 2a | Structure in scheme 1 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 31.64 ± 1.30 µM |
| dbacp07960 | Compound 2b | Structure in scheme 1 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 32.58 ± 1.50 µM |
| dbacp07964 | Compound 3b | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 25.33 ± 1.18 µM |
| dbacp07966 | Compound 3c | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 29.55 ± 2.06 µM |
| dbacp07969 | Compound 4b | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 10.45 ± 1.33 µM |
| dbacp07971 | Compound 4c | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 29.15 ± 1.39 µM |
| dbacp07973 | Compound 5a | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 12.67 ± 2.40 µM |
| dbacp07975 | Compound 5b | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 11.32 ± 1.15 µM |
| dbacp07977 | Compound 5c | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 9.41 ± 1.25 µM |
| dbacp07979 | Compound 6a | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 11.83 ± 1.62 µM |
| dbacp07981 | Compound 6b | Structure in scheme 2 | Synthetic | 5c inhibits cancer via kinase blockade | Not Available | MCF-7 | Breast Cancer | IC50 = 10.87 ± 1.10 µM |
| dbacp07993 | [G10a]SHa | FLSGIVGMLaKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 16.2 ± 2.2 µM |
| dbacp07996 | [G10a]SHa-BCTP | FLSGIVGMLaKLFLFKQYAELW | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 26.85 ± 1.85 µM |
| dbacp07999 | [G4a]SHa | FLSaIVGMLGKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 17.9 ± 1.1 µM |
| dbacp08002 | [G7a]SHa | FLSGIVaMLGKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 =22.4 ± 2.2 µM |
| dbacp08005 | [G4,7a]SHa | FLSaIVaMLGKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 29.5 ± 6.03 µM |
| dbacp08008 | [G4,7,10a]SHa | FLSaIVaMLaKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 26.33 ± 5.8 µM |
| dbacp08011 | [G7,10a]SHa | FLSGIVaMLaKLF | Synthetic analogue of Temporin-1SHa | Enhanced cationicity/hydrophobicity increases cytotoxicity | MTT assay | MCF-7 | Breast Cancer | IC50 = 21.3 ± 1.13 µM |
| dbacp08081 | Peptide 3a | YD | Synthetic | Inhibit COX-2 enzyme | MTT assay | MCF-7 | Breast Cancer | IC50 = 17.5 ± 0.04 µM |
| dbacp08086 | L-K6 | IKKILSKIKKLLK | Temporin 1CEb analogue | L-K6 binds, internalizes, damages nucleus | MTT assay | MCF-7 | Breast Cancer | IC50 = 31 μM |
| dbacp08090 | B1 | KKLFKKILKYLK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 15.7 ± 1.5 μM |
| dbacp08091 | B1 | KKLFKKILKYLK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 18.2 ± 1.3 μM |
| dbacp08094 | B2 | KKLFKKILKYLKK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 30.8 ± 3.4 μM |
| dbacp08095 | B2 | KKLFKKILKYLKK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 36.1 ± 6.7 μM |
| dbacp08098 | B3 | KKLFKKILKYLKKL | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 25.3 ± 3.2 μM |
| dbacp08099 | B3 | KKLFKKILKYLKKL | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 28.4 ± 3.1 μM |
| dbacp08101 | B5 | LKKLFKKILKYLK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 27.3 ± 2.4 μM |
| dbacp08102 | B5 | LKKLFKKILKYLK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 28.2 ± 2.7 μM |
| dbacp08105 | B6 | LKKLFKKILKYLKK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 18.4 ± 1.5 μM |
| dbacp08106 | B6 | LKKLFKKILKYLKK | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 20.7 ± 1.6 μM |
| dbacp08109 | B9 | KLKKLFKKILKY | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7 | Breast Cancer | IC50 = 38.3 ± 2.5 μM |
| dbacp08110 | B9 | KLKKLFKKILKY | Analogue of BP 100 | Membrane disruption triggers apoptosis | MTT assay | MCF-7/ADM | Breast Cancer | IC50 = 30.6 ± 5.7 μM |
| dbacp08136 | Laterosporulin10 (LS10) | ACVNQCPDAIDRFIVKDKGCHGVEKKYYKQVYVACMNGQHLYCRTEGGPCQL | Brevibacillus sp. strain SKDU10 | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | 40% cytotoxicity at 5 μM concentration |
| dbacp08137 | Laterosporulin10 (LS10) | ACVNQCPDAIDRFIVKDKGCHGVEKKYYKQVYVACMNGQHLYCRTEGGPCQL | Brevibacillus sp. strain SKDU10 | Apoptosis inducing | LDH leakage assay | MCF-7 | Breast Cancer | >80% LDH release at 15 μM |
| dbacp08143 | MccJ25-18-4 | GGAGHVPEYFVGIGTPISFYG-WxEAAYQrFL | Synthetic | Apoptosis inducing | MTT assay | MCF-7 | Breast Cancer | IC50 = 14.2 ± 1.5 μM |
| dbacp08150 | CIGB-552 | HARIKpTFRRlKWKYKGKFW | Synthetic | Not Available | Sulforhodamine B assay | MCF-7 | Breast Cancer | IC50 = 379.1 ± 8.6 µM |
| dbacp08170 | Peptide - 1 | GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKK | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 = 6.2 µM |
| dbacp08182 | Peptide - 2 | GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRR | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 = 7.0 µM |
| dbacp08190 | Peptide - 3 | GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- Orn | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 = 4.6 µM |
| dbacp08198 | Peptide - 4 | GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-Dab | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 = 3.0 µM |
| dbacp08206 | Peptide - 6 | GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKK | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 > 7.5 µM |
| dbacp08214 | Peptide - 7 | GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRR | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 > 7.5 µM |
| dbacp08222 | Peptide - 8 | GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKK | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 > 7.5 µM |
| dbacp08230 | Peptide - 9 | GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKK | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 > 7.5 µM |
| dbacp08238 | Peptide - 10 | GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKK | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 > 7.5 µM |
| dbacp08246 | Peptide - 11 | KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c) | Synthetic | Not Available | CellTiter-Glo assay | MCF-7 | Breast Cancer | IC50 = 7.3 µM |
| dbacp08254 | Tr1 | Not Available | Protein extraction from Spirulina platensis | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 60.12 μg/mL |
| dbacp08256 | Tr2 | Not Available | Protein extraction from Spirulina platensis | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 < 31.25 μg/mL |
| dbacp08260 | Tr4 | Not Available | Protein extraction from Spirulina platensis | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 238.86 μg/mL |
| dbacp08299 | SKACP003 | FPLPCAYKGTYC | Synthetic | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 193 ± 0.5 µM |
| dbacp08380 | IDP-LS13 | RKRRNDLRSRFLALRDQ | Synthetic | Not Available | MTT/Alamamar-Blue/Hexosaminidase activity test | MCF-7 | Breast Cancer | EC50 ~ 10 μM |
| dbacp08424 | 5-2C | NYPQRPCRGDKGPDC | Synthetic | Not Available | MTT assay | MCF-7 | Breast Cancer | IC50 = 9.74 μM |